SI9300309A - Novi biolosko ucinkoviti derivati eburnamenina, farmacevtski pripravki, ki jih vsebujejo, in postopek za njihovo pripravo - Google Patents
Novi biolosko ucinkoviti derivati eburnamenina, farmacevtski pripravki, ki jih vsebujejo, in postopek za njihovo pripravo Download PDFInfo
- Publication number
- SI9300309A SI9300309A SI9300309A SI9300309A SI9300309A SI 9300309 A SI9300309 A SI 9300309A SI 9300309 A SI9300309 A SI 9300309A SI 9300309 A SI9300309 A SI 9300309A SI 9300309 A SI9300309 A SI 9300309A
- Authority
- SI
- Slovenia
- Prior art keywords
- formula
- piperazine
- wavy line
- nitrogen
- group
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D461/00—Heterocyclic compounds containing indolo [3,2,1-d,e] pyrido [3,2,1,j] [1,5]-naphthyridine ring systems, e.g. vincamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Cardiology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU9201911A HU209678B (en) | 1992-06-09 | 1992-06-09 | Process for producing biologically active eburnamenin-14-carbonyl-amino derivatives and pharmaceutical compositions containing them |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI9300309A true SI9300309A (sl) | 1993-12-31 |
Family
ID=10982021
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI9300309A SI9300309A (sl) | 1992-06-09 | 1993-06-09 | Novi biolosko ucinkoviti derivati eburnamenina, farmacevtski pripravki, ki jih vsebujejo, in postopek za njihovo pripravo |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US5510345A (ko) |
| EP (1) | EP0644885A1 (ko) |
| JP (1) | JPH07507793A (ko) |
| KR (1) | KR950701924A (ko) |
| AU (1) | AU4352493A (ko) |
| CA (1) | CA2136547A1 (ko) |
| CZ (1) | CZ307994A3 (ko) |
| EE (1) | EE9400070A (ko) |
| FI (1) | FI945780A0 (ko) |
| GR (1) | GR1001597B (ko) |
| HR (1) | HRP930957A2 (ko) |
| HU (1) | HU209678B (ko) |
| IL (1) | IL105942A0 (ko) |
| LT (1) | LT3118B (ko) |
| NZ (1) | NZ253308A (ko) |
| SI (1) | SI9300309A (ko) |
| WO (1) | WO1993025550A1 (ko) |
| ZA (1) | ZA934037B (ko) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1799664A1 (en) | 2004-09-20 | 2007-06-27 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
| BRPI0515505A (pt) | 2004-09-20 | 2008-07-29 | Xenon Pharmaceuticals Inc | derivados heterocìclicos e sua utilização como inibidores da estearoil-coa desaturase |
| EP1799668A1 (en) | 2004-09-20 | 2007-06-27 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as mediators of stearoyl-coa desaturase |
| TW200626138A (en) | 2004-09-20 | 2006-08-01 | Xenon Pharmaceuticals Inc | Heterocyclic derivatives and their use as therapeutic agents |
| CA2580845A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives for inhibiting human stearoyl-coa-desaturase |
| CA2580787A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes |
| CA2580857A1 (en) | 2004-09-20 | 2006-09-28 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
| US7820654B2 (en) * | 2004-09-23 | 2010-10-26 | Dr. Reddy's Laboratories Ltd. | Pyrimidine compounds, process for their preparation and compositions containing them |
| US8541457B2 (en) | 2005-06-03 | 2013-09-24 | Xenon Pharmaceuticals Inc. | Aminothiazole derivatives as human stearoyl-CoA desaturase inhibitors |
| EP2276750A2 (en) * | 2008-03-27 | 2011-01-26 | Auckland Uniservices Limited | Substituted pyrimidines and triazines and their use in cancer therapy |
| CN101928286A (zh) * | 2009-06-18 | 2010-12-29 | 谢开智 | 长春胺衍生物及制备方法 |
| ES2753386T3 (es) | 2013-03-13 | 2020-04-08 | Forma Therapeutics Inc | Derivados de 2-hidroxi-1-{4-[(4-fenil)fenil]carbonil}piperazin-1-il}etano-1-ona y compuestos relacionados como inhibidores de sintasa de ácido graso (FASN) para el tratamiento del cáncer |
| WO2017210545A1 (en) | 2016-06-02 | 2017-12-07 | Cadent Therapeutics, Inc. | Potassium channel modulators |
| SG11201905893WA (en) | 2017-01-23 | 2019-08-27 | Cadent Therapeutics Inc | Potassium channel modulators |
| MX2021004647A (es) | 2018-10-22 | 2021-08-16 | Novartis Ag | Formas cristalinas de moduladores de los canales de potasio. |
| CN113382633A (zh) | 2018-10-29 | 2021-09-10 | 福马治疗股份有限公司 | (4-(2-氟-4-(1-甲基-1H-苯并[d]咪唑-5-基)苯甲酰基)哌嗪-1-基)(1-羟基环丙基)甲酮的固体形式 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2176516B1 (ko) * | 1972-03-22 | 1975-03-14 | Synthelabo | |
| HU171663B (hu) * | 1975-09-01 | 1978-02-28 | Richter Gedeon Vegyeszet | Sposob poluchenija novykh proizvodnykh 14-skobka-zamehhennogo metil-skobka zakryta-vinkana |
| US4547505A (en) * | 1983-03-25 | 1985-10-15 | Degussa Aktiengesellschaft | N-Phenyl-N-'-cycloalkylalkanoylpiperazine useful as analgetics and process for its production |
| US5099019A (en) * | 1985-09-12 | 1992-03-24 | Upjohn Company | Amines useful in producing pharmaceutically active CNS compounds |
| WO1987001706A2 (en) | 1985-09-12 | 1987-03-26 | The Upjohn Company | C20 through c26 amino steroids |
| AU7580187A (en) | 1986-06-23 | 1988-01-12 | Upjohn Company, The | Androstane-type and cortical aminoesters |
| KR890700581A (ko) | 1987-04-03 | 1989-04-25 | 로버어트 에이 아미테이지 | 아미노 -9,10-세코스테로이드 |
| CA1338012C (en) | 1987-04-27 | 1996-01-30 | John Michael Mccall | Pharmaceutically active amines |
| FR2644788B1 (fr) | 1989-03-22 | 1995-02-03 | Roussel Uclaf | Nouveaux steroides 3-ceto comportant une chaine en 17 amino-substituee, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant |
| FR2644787B1 (fr) | 1989-03-22 | 1995-02-03 | Roussel Uclaf | Nouveaux steroides 21 aminosubstitues, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant |
| FR2644789B1 (fr) | 1989-03-22 | 1995-02-03 | Roussel Uclaf | Nouveaux steroides 19-nor, 3-ceto comportant une chaine en 17 aminosubstituee, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant |
| AU642711B2 (en) | 1990-01-26 | 1993-10-28 | Upjohn Company, The | 5-oxygenated-2,4,6-triaminopyrimidines |
-
1992
- 1992-06-09 HU HU9201911A patent/HU209678B/hu not_active IP Right Cessation
-
1993
- 1993-06-02 LT LTIP599A patent/LT3118B/lt not_active IP Right Cessation
- 1993-06-08 NZ NZ253308A patent/NZ253308A/en unknown
- 1993-06-08 WO PCT/HU1993/000036 patent/WO1993025550A1/en not_active Application Discontinuation
- 1993-06-08 HR HR930957A patent/HRP930957A2/xx not_active Application Discontinuation
- 1993-06-08 JP JP6501317A patent/JPH07507793A/ja active Pending
- 1993-06-08 CZ CZ943079A patent/CZ307994A3/cs unknown
- 1993-06-08 EP EP93913456A patent/EP0644885A1/en not_active Withdrawn
- 1993-06-08 US US08/351,447 patent/US5510345A/en not_active Expired - Fee Related
- 1993-06-08 ZA ZA934037A patent/ZA934037B/xx unknown
- 1993-06-08 AU AU43524/93A patent/AU4352493A/en not_active Abandoned
- 1993-06-08 GR GR930100233A patent/GR1001597B/el unknown
- 1993-06-08 CA CA002136547A patent/CA2136547A1/en not_active Abandoned
- 1993-06-08 IL IL105942A patent/IL105942A0/xx unknown
- 1993-06-09 SI SI9300309A patent/SI9300309A/sl unknown
-
1994
- 1994-06-29 EE EE9400070A patent/EE9400070A/xx unknown
- 1994-12-08 FI FI945780A patent/FI945780A0/fi not_active Application Discontinuation
- 1994-12-09 KR KR1019940704495A patent/KR950701924A/ko not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| US5510345A (en) | 1996-04-23 |
| ZA934037B (en) | 1994-01-06 |
| WO1993025550A1 (en) | 1993-12-23 |
| AU4352493A (en) | 1994-01-04 |
| HU9201911D0 (en) | 1992-09-28 |
| NZ253308A (en) | 1995-11-27 |
| CZ307994A3 (en) | 1995-07-12 |
| CA2136547A1 (en) | 1993-12-23 |
| LT3118B (en) | 1994-12-27 |
| GR1001597B (el) | 1994-06-30 |
| KR950701924A (ko) | 1995-05-17 |
| JPH07507793A (ja) | 1995-08-31 |
| HRP930957A2 (en) | 1995-02-28 |
| FI945780A (fi) | 1994-12-08 |
| LTIP599A (en) | 1994-07-15 |
| EP0644885A1 (en) | 1995-03-29 |
| HU209678B (en) | 1994-10-28 |
| IL105942A0 (en) | 1993-10-20 |
| FI945780A0 (fi) | 1994-12-08 |
| EE9400070A (et) | 1995-12-15 |
| HUT64540A (en) | 1994-01-28 |
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