SI9300212A - Novel N-acyldipeptides, process for the preparation thereof and pharmaceutical composition containing the same - Google Patents

Novel N-acyldipeptides, process for the preparation thereof and pharmaceutical composition containing the same Download PDF

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Publication number
SI9300212A
SI9300212A SI9300212A SI9300212A SI9300212A SI 9300212 A SI9300212 A SI 9300212A SI 9300212 A SI9300212 A SI 9300212A SI 9300212 A SI9300212 A SI 9300212A SI 9300212 A SI9300212 A SI 9300212A
Authority
SI
Slovenia
Prior art keywords
group
carbon atoms
straight
branched alkyl
hydrogen
Prior art date
Application number
SI9300212A
Other languages
English (en)
Slovenian (sl)
Inventor
Danijel Kikelj
Elizabeta Suhadolc
Slavko Pecar
Alesa Puncuh
Uros Urleb
Gasper Marc
Marija Sollner
Ales Krbavcic
Original Assignee
Univ Ljubljani
Lek Tovarna Farmacevtskih
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Ljubljani, Lek Tovarna Farmacevtskih filed Critical Univ Ljubljani
Priority to SI9300212A priority Critical patent/SI9300212A/sl
Priority to US08/537,782 priority patent/US5824652A/en
Priority to AT94914681T priority patent/ATE167873T1/de
Priority to PCT/SI1994/000003 priority patent/WO1994024152A1/en
Priority to JP6523063A priority patent/JP2886987B2/ja
Priority to EP94914681A priority patent/EP0695308B1/de
Priority to ES94914681T priority patent/ES2120039T3/es
Priority to SI9430187T priority patent/SI0695308T1/xx
Priority to DE69411380T priority patent/DE69411380T2/de
Publication of SI9300212A publication Critical patent/SI9300212A/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
    • C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C07D279/16—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
SI9300212A 1993-04-22 1993-04-22 Novel N-acyldipeptides, process for the preparation thereof and pharmaceutical composition containing the same SI9300212A (en)

Priority Applications (9)

Application Number Priority Date Filing Date Title
SI9300212A SI9300212A (en) 1993-04-22 1993-04-22 Novel N-acyldipeptides, process for the preparation thereof and pharmaceutical composition containing the same
US08/537,782 US5824652A (en) 1993-04-22 1994-04-21 Heterocyclic acyldipeptides, processes for the preparation thereof and pharmaceutical compositions containing the same
AT94914681T ATE167873T1 (de) 1993-04-22 1994-04-21 Neue heterocyclische acyldipeptide, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzung
PCT/SI1994/000003 WO1994024152A1 (en) 1993-04-22 1994-04-21 Novel heterocyclic acyldipeptides, processes for the preparation thereof and pharmaceutical compositions containing the same
JP6523063A JP2886987B2 (ja) 1993-04-22 1994-04-21 新規な複素環式アシルジペプチド、その製造方法及びこれを含有する医薬組成物
EP94914681A EP0695308B1 (de) 1993-04-22 1994-04-21 Neue heterocyclische acyldipeptide, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzung
ES94914681T ES2120039T3 (es) 1993-04-22 1994-04-21 Nuevos acildipeptidos heterociclicos, procedimientos de preparacion y composiciones farmaceuticas que los contienen.
SI9430187T SI0695308T1 (en) 1993-04-22 1994-04-21 Novel heterocyclic acyldipeptides, processes for the preparation thereof and pharmaceutical compositions containing the same
DE69411380T DE69411380T2 (de) 1993-04-22 1994-04-21 Neue heterocyclische acyldipeptide, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzung

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SI9300212A SI9300212A (en) 1993-04-22 1993-04-22 Novel N-acyldipeptides, process for the preparation thereof and pharmaceutical composition containing the same

Publications (1)

Publication Number Publication Date
SI9300212A true SI9300212A (en) 1994-12-31

Family

ID=20431165

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9300212A SI9300212A (en) 1993-04-22 1993-04-22 Novel N-acyldipeptides, process for the preparation thereof and pharmaceutical composition containing the same

Country Status (8)

Country Link
US (1) US5824652A (de)
EP (1) EP0695308B1 (de)
JP (1) JP2886987B2 (de)
AT (1) ATE167873T1 (de)
DE (1) DE69411380T2 (de)
ES (1) ES2120039T3 (de)
SI (1) SI9300212A (de)
WO (1) WO1994024152A1 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2311411B1 (es) * 2007-07-19 2010-01-08 Universidad De Cadiz. Derivados 2-alquil-2h-1, 4-benzoxacin-3(4h)-ona y 2-alcoxicarbonil-2h-1,4-benzoxacin-3(4h)-ona, con actividad fitotoxica.

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2326930A1 (fr) * 1975-10-09 1977-05-06 Anvar Agents hydrosolubles depresseurs non specifiques des reponses immunitaires
US4322341A (en) * 1980-05-13 1982-03-30 Fujisawa Pharmaceutical Co Peptide, process for preparation thereof and use thereof
SI9011830B (sl) * 1990-09-27 1999-12-31 Univerza V Ljubljani, Fakulteta Za Farmacijo Novi N-acildipeptidi, postopki za njihovo pripravo in farmacevtski pripravki, ki jih vsebujejo
US5321216A (en) * 1991-04-09 1994-06-14 Otis Elevator Company Restraining elevator car motion while the doors are open

Also Published As

Publication number Publication date
JP2886987B2 (ja) 1999-04-26
ATE167873T1 (de) 1998-07-15
DE69411380D1 (de) 1998-08-06
EP0695308B1 (de) 1998-07-01
EP0695308A1 (de) 1996-02-07
ES2120039T3 (es) 1998-10-16
US5824652A (en) 1998-10-20
WO1994024152A1 (en) 1994-10-27
JPH09506856A (ja) 1997-07-08
DE69411380T2 (de) 1999-04-01

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