SI9300005A - Process for the preparation of substituted steroidal benzoesters and substituted steroidal benzoacids - Google Patents

Process for the preparation of substituted steroidal benzoesters and substituted steroidal benzoacids Download PDF

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Publication number
SI9300005A
SI9300005A SI19939300005A SI9300005A SI9300005A SI 9300005 A SI9300005 A SI 9300005A SI 19939300005 A SI19939300005 A SI 19939300005A SI 9300005 A SI9300005 A SI 9300005A SI 9300005 A SI9300005 A SI 9300005A
Authority
SI
Slovenia
Prior art keywords
compound
formula
reaction
process according
steroidal
Prior art date
Application number
SI19939300005A
Other languages
English (en)
Slovenian (sl)
Inventor
Neil Howard Baine
Michael Maguire
Original Assignee
Smithkline Beecham Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corporation filed Critical Smithkline Beecham Corporation
Publication of SI9300005A publication Critical patent/SI9300005A/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J51/00Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
    • HELECTRICITY
    • H10SEMICONDUCTOR DEVICES; ELECTRIC SOLID-STATE DEVICES NOT OTHERWISE PROVIDED FOR
    • H10NELECTRIC SOLID-STATE DEVICES NOT OTHERWISE PROVIDED FOR
    • H10N30/00Piezoelectric or electrostrictive devices
    • H10N30/20Piezoelectric or electrostrictive devices with electrical input and mechanical output, e.g. functioning as actuators or vibrators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00Preparation of carboxylic acids or their salts, halides or anhydrides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J3/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0094Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Toxicology (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
SI19939300005A 1992-01-06 1993-01-06 Process for the preparation of substituted steroidal benzoesters and substituted steroidal benzoacids SI9300005A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US81718092A 1992-01-06 1992-01-06

Publications (1)

Publication Number Publication Date
SI9300005A true SI9300005A (en) 1993-09-30

Family

ID=25222515

Family Applications (1)

Application Number Title Priority Date Filing Date
SI19939300005A SI9300005A (en) 1992-01-06 1993-01-06 Process for the preparation of substituted steroidal benzoesters and substituted steroidal benzoacids

Country Status (21)

Country Link
EP (1) EP0621866A4 (hu)
JP (1) JPH07503008A (hu)
KR (1) KR940704064A (hu)
CN (1) CN1077200A (hu)
AP (1) AP361A (hu)
AU (1) AU3434793A (hu)
BG (1) BG98888A (hu)
BR (1) BR9305707A (hu)
CA (1) CA2127274A1 (hu)
FI (1) FI943213A0 (hu)
HU (1) HUT67566A (hu)
IL (1) IL104303A0 (hu)
MA (1) MA22762A1 (hu)
MX (1) MX9300026A (hu)
NO (1) NO942531D0 (hu)
OA (1) OA09959A (hu)
RU (1) RU94037761A (hu)
SI (1) SI9300005A (hu)
SK (1) SK80194A3 (hu)
WO (1) WO1993014107A1 (hu)
ZA (1) ZA938B (hu)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1993022333A1 (en) * 1992-04-30 1993-11-11 Smithkline Beecham Corporation 17α AND 17β-SUBSTITUTED ESTRA-1,3,5(10)-TRIENE-3-CARBOXYLIC ACID
GB9411103D0 (en) * 1994-06-03 1994-07-27 Smithkline Beecham Corp Compounds
GB9608045D0 (en) * 1996-04-18 1996-06-19 Pharmacia Spa Process for preparing steroids having a carboxamide side-chain
JP2000309599A (ja) 1999-04-13 2000-11-07 Kyowa Hakko Kogyo Co Ltd エストラ−1,3,5(10),16−テトラエン誘導体
JP5793996B2 (ja) * 2011-06-29 2015-10-14 セントラル硝子株式会社 フルオロ硫酸芳香環エステル類の製造方法
EP4295841A3 (en) 2014-06-06 2024-03-13 The Scripps Research Institute Sulfur (vi) fluoride compounds and their use in click-reaction

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4954446A (en) * 1988-05-25 1990-09-04 Smithkline Beecham Corporation Aromatic steroid 5-α-reductase inhibitors
US4937237A (en) * 1988-12-23 1990-06-26 Smithkline Beckman Corporation Phosphinic acid substituted aromatic steroids as inhibitors of steroid 5-60 -reductase
US4970205A (en) * 1988-12-23 1990-11-13 Smithkline Beecham Corporation Sulfonic acid substituted aromatic steroids as inhibitors of steroid 5-α-reductase

Also Published As

Publication number Publication date
ZA938B (en) 1994-06-16
AP9300474A0 (en) 1993-01-31
MA22762A1 (fr) 1993-10-01
BR9305707A (pt) 1996-12-31
NO942531L (no) 1994-07-05
MX9300026A (es) 1993-12-01
BG98888A (en) 1995-05-31
CA2127274A1 (en) 1993-07-22
NO942531D0 (no) 1994-07-05
RU94037761A (ru) 1997-05-27
WO1993014107A1 (en) 1993-07-22
AU3434793A (en) 1993-08-03
HU9402029D0 (en) 1994-09-28
SK80194A3 (en) 1994-12-07
EP0621866A4 (en) 1996-03-20
HUT67566A (en) 1995-04-28
FI943213A (fi) 1994-07-05
JPH07503008A (ja) 1995-03-30
FI943213A0 (fi) 1994-07-05
KR940704064A (ko) 1994-12-12
CN1077200A (zh) 1993-10-13
IL104303A0 (en) 1993-05-13
AP361A (en) 1994-09-09
OA09959A (en) 1995-12-11
EP0621866A1 (en) 1994-11-02

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