SI9200402A - Substituted benzimidazoles, process for their preparation and their use - Google Patents

Substituted benzimidazoles, process for their preparation and their use Download PDF

Info

Publication number
SI9200402A
SI9200402A SI19929200402A SI9200402A SI9200402A SI 9200402 A SI9200402 A SI 9200402A SI 19929200402 A SI19929200402 A SI 19929200402A SI 9200402 A SI9200402 A SI 9200402A SI 9200402 A SI9200402 A SI 9200402A
Authority
SI
Slovenia
Prior art keywords
methyl
compound
formula
compounds
pyridinyl
Prior art date
Application number
SI19929200402A
Other languages
English (en)
Slovenian (sl)
Inventor
Karl Bjoern Christer Holstein
Gunnel Elisabeth Sunden
Original Assignee
Aktiebolaget Astra
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aktiebolaget Astra filed Critical Aktiebolaget Astra
Publication of SI9200402A publication Critical patent/SI9200402A/sl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SI19929200402A 1991-12-19 1992-12-18 Substituted benzimidazoles, process for their preparation and their use SI9200402A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9103776A SE9103776D0 (sv) 1991-12-19 1991-12-19 New compounds

Publications (1)

Publication Number Publication Date
SI9200402A true SI9200402A (en) 1993-06-30

Family

ID=20384667

Family Applications (1)

Application Number Title Priority Date Filing Date
SI19929200402A SI9200402A (en) 1991-12-19 1992-12-18 Substituted benzimidazoles, process for their preparation and their use

Country Status (25)

Country Link
EP (1) EP0628049A1 (esLanguage)
JP (1) JPH07502503A (esLanguage)
KR (1) KR940703840A (esLanguage)
CN (1) CN1031827C (esLanguage)
AP (1) AP397A (esLanguage)
AU (1) AU665043B2 (esLanguage)
CA (1) CA2124689A1 (esLanguage)
CZ (1) CZ146794A3 (esLanguage)
FI (1) FI942912A0 (esLanguage)
HR (1) HRP921400A2 (esLanguage)
HU (1) HUT68270A (esLanguage)
IL (1) IL104025A0 (esLanguage)
IS (2) IS4079A (esLanguage)
MA (1) MA22746A1 (esLanguage)
MX (1) MX9207269A (esLanguage)
NO (1) NO942230D0 (esLanguage)
NZ (1) NZ246220A (esLanguage)
SE (1) SE9103776D0 (esLanguage)
SI (1) SI9200402A (esLanguage)
SK (1) SK73594A3 (esLanguage)
TN (1) TNSN92115A1 (esLanguage)
TW (1) TW224100B (esLanguage)
WO (1) WO1993012124A1 (esLanguage)
YU (1) YU101692A (esLanguage)
ZA (1) ZA928836B (esLanguage)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19645974C1 (de) * 1996-11-07 1998-08-13 Andreas Johannes Kesel (Z)-5-[[3-Hydroxy-2-methyl-5-[(phosphonooxy)methyl]-4-pyridinyl]methylen]-2-thioxo-4- thiazolidinon, Verfahren zu dessen Herstellung und Verwendung
AU754965B2 (en) * 1997-12-31 2002-11-28 University Of Kansas, The Water soluble prodrugs of tertiary amine containing drugs and methods of making thereof
CA2616512A1 (en) 2005-07-28 2007-02-08 Intervet International B.V. Novel benzimidazole (thio) carbamates with antiparasitic activity and the synthesis thereof
TWI385169B (zh) 2005-10-31 2013-02-11 Eisai R&D Man Co Ltd 經雜環取代之吡啶衍生物及含有彼之抗真菌劑
KR101403135B1 (ko) 2006-06-14 2014-06-19 인터벳 인터내셔널 비.브이. 벤지미다졸 카르바메이트 및 폴리솔베이트를 포함하는 현탁물
TW200841879A (en) 2007-04-27 2008-11-01 Eisai R&D Man Co Ltd Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same
US8513287B2 (en) 2007-12-27 2013-08-20 Eisai R&D Management Co., Ltd. Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same
US8188119B2 (en) 2008-10-24 2012-05-29 Eisai R&D Management Co., Ltd Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same
MX365051B (es) * 2014-11-26 2019-05-09 Univ Mexico Nac Autonoma Nuevos compuestos hidrosolubles derivados del bencimidazol, utiles para el tratamiento de la fasciolosis.

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ234564A (en) * 1986-11-21 1991-04-26 Haessle Ab 1-substituted benzimidazoles and pharmaceutical compositions
SE8801907D0 (sv) * 1988-05-20 1988-05-20 Haessle Ab Novel pharmacological compounds
SE9002206D0 (sv) * 1990-06-20 1990-06-20 Haessle Ab New compounds
WO1991019712A1 (en) * 1990-06-20 1991-12-26 Aktiebolaget Astra Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use

Also Published As

Publication number Publication date
TW224100B (esLanguage) 1994-05-21
SE9103776D0 (sv) 1991-12-19
YU101692A (sh) 1995-10-03
CA2124689A1 (en) 1993-06-24
AU3175293A (en) 1993-07-19
CZ146794A3 (en) 1996-02-14
AU665043B2 (en) 1995-12-14
HU9401840D0 (en) 1994-09-28
IS4079A (is) 1993-06-20
NO942230L (no) 1994-06-14
FI942912L (fi) 1994-06-17
FI942912A7 (fi) 1994-06-17
SK73594A3 (en) 1995-02-08
HUT68270A (en) 1995-06-28
IL104025A0 (en) 1993-05-13
NZ246220A (en) 1996-02-27
JPH07502503A (ja) 1995-03-16
MA22746A1 (fr) 1993-07-01
NO942230D0 (no) 1994-06-14
WO1993012124A1 (en) 1993-06-24
CN1073446A (zh) 1993-06-23
TNSN92115A1 (fr) 1993-06-08
AP9200463A0 (en) 1993-01-31
HRP921400A2 (en) 1994-08-31
KR940703840A (ko) 1994-12-12
AP397A (en) 1995-08-14
FI942912A0 (fi) 1994-06-17
EP0628049A1 (en) 1994-12-14
ZA928836B (en) 1993-07-05
IS3960A (is) 1993-06-20
MX9207269A (es) 1993-06-01
CN1031827C (zh) 1996-05-22

Similar Documents

Publication Publication Date Title
EP0593463B1 (en) Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
US7189744B2 (en) Crystals of benzimidazole compounds
CA1302891C (en) Pharmaceutical formulations of acid labile substances for oral use
US7569697B2 (en) Benzimidazole compound crystal
JPH0739412B2 (ja) 新規なスルホキシド
EP0449940A1 (en) NOVEL THERAPEUTICALLY ACTIVE COMPOUND AND PREPARATION METHOD THEREOF.
RO110493B1 (ro) Derivati de benzimidazol si procedee pentru prepararea acestora
JP2793907B2 (ja) 治療上活性な置換されたベンズイミダゾールおよびその製法
CA2005980C (en) Benzimidazole derivative with gastric acid inhibitory effect and process for its preparation
AP397A (en) Substituted benzimidazoles, process for their preparation as well as their use.