SI9200095A - Heterocyclic derivatives - Google Patents

Heterocyclic derivatives Download PDF

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Publication number
SI9200095A
SI9200095A SI19929200095A SI9200095A SI9200095A SI 9200095 A SI9200095 A SI 9200095A SI 19929200095 A SI19929200095 A SI 19929200095A SI 9200095 A SI9200095 A SI 9200095A SI 9200095 A SI9200095 A SI 9200095A
Authority
SI
Slovenia
Prior art keywords
formula
compound
methyl
alkyl
group
Prior art date
Application number
SI19929200095A
Other languages
English (en)
Slovenian (sl)
Inventor
Arnold Harry Ratcliffe
Robert James Pearce
Keith Hopkinson Gibson
Robin Wood
Brian Bernard Masek
Original Assignee
Imperial Chemical Industries Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB919111759A external-priority patent/GB9111759D0/en
Priority claimed from GB919116309A external-priority patent/GB9116309D0/en
Application filed by Imperial Chemical Industries Plc filed Critical Imperial Chemical Industries Plc
Publication of SI9200095A publication Critical patent/SI9200095A/sl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Anesthesiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SI19929200095A 1991-05-31 1992-05-29 Heterocyclic derivatives SI9200095A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB919111759A GB9111759D0 (en) 1991-05-31 1991-05-31 Heterocyclic compounds
GB919116309A GB9116309D0 (en) 1991-07-29 1991-07-29 Bicyclic derivatives

Publications (1)

Publication Number Publication Date
SI9200095A true SI9200095A (en) 1992-12-31

Family

ID=26298984

Family Applications (1)

Application Number Title Priority Date Filing Date
SI19929200095A SI9200095A (en) 1991-05-31 1992-05-29 Heterocyclic derivatives

Country Status (21)

Country Link
US (2) US5217976A (zh)
EP (1) EP0516392B1 (zh)
JP (1) JPH05163271A (zh)
KR (1) KR920021545A (zh)
CN (1) CN1073174A (zh)
AT (1) ATE204873T1 (zh)
AU (1) AU1625192A (zh)
CA (1) CA2068946A1 (zh)
CS (1) CS161892A3 (zh)
DE (1) DE69232022D1 (zh)
FI (1) FI922481A (zh)
GB (1) GB2256196B (zh)
HU (1) HUT61303A (zh)
IE (1) IE921506A1 (zh)
IL (1) IL101860A0 (zh)
NO (1) NO922147L (zh)
OA (1) OA09982A (zh)
PL (1) PL294736A1 (zh)
SI (1) SI9200095A (zh)
TW (1) TW213914B (zh)
YU (1) YU56192A (zh)

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US7279487B2 (en) * 2002-01-17 2007-10-09 Merck & Co., Inc. Hydroxynaphthyridinone carboxamides useful as HIV integrase inhibitors
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Also Published As

Publication number Publication date
PL294736A1 (en) 1993-05-31
HUT61303A (en) 1992-12-28
EP0516392A3 (en) 1993-01-27
GB2256196A (en) 1992-12-02
FI922481A (fi) 1992-12-01
DE69232022D1 (de) 2001-10-04
CA2068946A1 (en) 1992-12-01
CN1073174A (zh) 1993-06-16
GB9211211D0 (en) 1992-07-08
ATE204873T1 (de) 2001-09-15
US5217976A (en) 1993-06-08
US5294620A (en) 1994-03-15
YU56192A (sh) 1994-11-15
KR920021545A (ko) 1992-12-18
NO922147D0 (no) 1992-05-29
FI922481A0 (fi) 1992-05-29
HU9201608D0 (en) 1992-08-28
EP0516392B1 (en) 2001-08-29
IL101860A0 (en) 1992-12-30
CS161892A3 (en) 1992-12-16
GB2256196B (en) 1995-05-10
AU1625192A (en) 1992-12-03
TW213914B (zh) 1993-10-01
EP0516392A2 (en) 1992-12-02
OA09982A (fr) 1996-03-29
IE921506A1 (en) 1992-12-02
JPH05163271A (ja) 1993-06-29
NO922147L (no) 1992-12-01

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