SI1691808T1 - Farmacevtski sestavek za oralno dajanje derivata pirazol-3-karboksamida - Google Patents

Farmacevtski sestavek za oralno dajanje derivata pirazol-3-karboksamida

Info

Publication number
SI1691808T1
SI1691808T1 SI200431173T SI200431173T SI1691808T1 SI 1691808 T1 SI1691808 T1 SI 1691808T1 SI 200431173 T SI200431173 T SI 200431173T SI 200431173 T SI200431173 T SI 200431173T SI 1691808 T1 SI1691808 T1 SI 1691808T1
Authority
SI
Slovenia
Prior art keywords
pyrazol
pharmaceutical composition
oral administration
carboxamide derivative
carboxamide
Prior art date
Application number
SI200431173T
Other languages
English (en)
Inventor
Thierry Breul
Jean Claude Gautier
Olivier Saslawski
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of SI1691808T1 publication Critical patent/SI1691808T1/sl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Dispersion Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SI200431173T 2003-11-10 2004-11-09 Farmacevtski sestavek za oralno dajanje derivata pirazol-3-karboksamida SI1691808T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0313259A FR2861992B1 (fr) 2003-11-10 2003-11-10 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3-carboxamide.
EP04805418A EP1691808B1 (fr) 2003-11-10 2004-11-09 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3-carboxamide
PCT/FR2004/002875 WO2005046690A1 (fr) 2003-11-10 2004-11-09 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3­carboxamide

Publications (1)

Publication Number Publication Date
SI1691808T1 true SI1691808T1 (sl) 2009-10-31

Family

ID=34508418

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200431173T SI1691808T1 (sl) 2003-11-10 2004-11-09 Farmacevtski sestavek za oralno dajanje derivata pirazol-3-karboksamida

Country Status (28)

Country Link
US (2) US20060264469A1 (sl)
EP (1) EP1691808B1 (sl)
JP (1) JP4767171B2 (sl)
KR (1) KR20060108668A (sl)
CN (1) CN100528158C (sl)
AR (1) AR047237A1 (sl)
AT (1) ATE429227T1 (sl)
AU (1) AU2004289086A1 (sl)
BR (1) BRPI0416341A (sl)
CA (1) CA2544413A1 (sl)
CY (1) CY1110478T1 (sl)
DE (1) DE602004020797D1 (sl)
DK (1) DK1691808T3 (sl)
ES (1) ES2325373T3 (sl)
FR (1) FR2861992B1 (sl)
HK (1) HK1102021A1 (sl)
HR (1) HRP20090393T1 (sl)
IL (1) IL175556A (sl)
MA (1) MA28419B1 (sl)
NO (1) NO20062609L (sl)
NZ (1) NZ547763A (sl)
PL (1) PL1691808T3 (sl)
PT (1) PT1691808E (sl)
RU (1) RU2321404C1 (sl)
SI (1) SI1691808T1 (sl)
TW (1) TWI280129B (sl)
WO (1) WO2005046690A1 (sl)
ZA (1) ZA200604451B (sl)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1880715A1 (en) 2006-07-19 2008-01-23 Abbott GmbH & Co. KG Pharmaceutically acceptable solubilizing composition and pharmaceutical dosage form containing same
EP1920767A1 (en) * 2006-11-09 2008-05-14 Abbott GmbH & Co. KG Melt-processed imatinib dosage form
CN101784259B (zh) * 2007-08-21 2013-03-27 巴斯利尔药物股份公司 抗真菌组合物
MY158809A (en) * 2010-09-22 2016-11-15 Craun Res Sdn Bhd Pharmaceutical compositions for calanolides, their derivatives and analogues, and process for producing the same
US20130317117A1 (en) * 2010-11-24 2013-11-28 Pharmaceutics International, Inc. Self micro-emulsifying drug delivery system with increased bioavailability

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5059691A (en) * 1990-01-22 1991-10-22 American Cyanamid Company N-((dialkylamino)methylene)-substituted pyrazolo (1,5-A)-pyrimidine-3-carboxamides and N-((dialkylamino)methylene)-substituted-4,5-dihydropyrazolo-(1,5-A)-pyrimidine-3-carboxamides
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
SI1033128T2 (sl) * 1993-09-28 2012-02-29 Scherer Gmbh R P Izdelava mehke Ĺľelatinaste kapsule
GB9405304D0 (en) * 1994-03-16 1994-04-27 Scherer Ltd R P Delivery systems for hydrophobic drugs
AU692255B2 (en) * 1995-04-24 1998-06-04 Yissum Research Development Company Of The Hebrew University Of Jerusalem Self-emulsifiable formulation producing an oil-in-water emulsion
CA2221145A1 (en) * 1995-05-19 1996-11-21 Abbott Laboratories Self-emulsifying formulations of lipophilic drugs
US5993858A (en) * 1996-06-14 1999-11-30 Port Systems L.L.C. Method and formulation for increasing the bioavailability of poorly water-soluble drugs
CN1092659C (zh) * 1997-03-14 2002-10-16 大塚制药株式会社 新型嘧啶衍生物
FR2761265B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique pour l'administration orale d'un derive du n-piperidino-3-pyrazolecarboxamide, de ses sels et de leurs solvates
FR2761266B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
US6617426B1 (en) * 1999-06-22 2003-09-09 Merck & Co Inc Cysteinyl protease inhibitors
JP2001151669A (ja) * 1999-11-24 2001-06-05 Nippon Kayaku Co Ltd 経口用自己乳化製剤
MXPA02006324A (es) * 1999-12-23 2002-12-13 Pfizer Prod Inc Composiciones farmaceuticas que proporcionan concentraciones potenciadas de farmaco.
GB0001928D0 (en) * 2000-01-27 2000-03-22 Novartis Ag Organic compounds
FR2831883B1 (fr) * 2001-11-08 2004-07-23 Sanofi Synthelabo Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
ATE359779T1 (de) * 2002-03-01 2007-05-15 Novagali Pharma Sa Selbstemulgierende systeme zur abgabe von taxoiden
GB0216700D0 (en) * 2002-07-18 2002-08-28 Astrazeneca Ab Process

Also Published As

Publication number Publication date
KR20060108668A (ko) 2006-10-18
US20090004261A1 (en) 2009-01-01
NZ547763A (en) 2009-08-28
IL175556A (en) 2010-11-30
CY1110478T1 (el) 2015-04-29
AU2004289086A1 (en) 2005-05-26
DE602004020797D1 (de) 2009-06-04
ATE429227T1 (de) 2009-05-15
MA28419B1 (fr) 2007-02-01
PL1691808T3 (pl) 2009-09-30
EP1691808A1 (fr) 2006-08-23
ZA200604451B (en) 2007-10-31
CN100528158C (zh) 2009-08-19
JP4767171B2 (ja) 2011-09-07
BRPI0416341A (pt) 2007-02-27
EP1691808B1 (fr) 2009-04-22
RU2006120447A (ru) 2007-12-20
DK1691808T3 (da) 2009-08-03
WO2005046690A1 (fr) 2005-05-26
CN1925856A (zh) 2007-03-07
FR2861992B1 (fr) 2007-07-20
AR047237A1 (es) 2006-01-11
PT1691808E (pt) 2009-07-14
TWI280129B (en) 2007-05-01
FR2861992A1 (fr) 2005-05-13
RU2321404C1 (ru) 2008-04-10
ES2325373T3 (es) 2009-09-02
NO20062609L (no) 2006-06-06
JP2007516960A (ja) 2007-06-28
US20060264469A1 (en) 2006-11-23
HRP20090393T1 (en) 2009-08-31
IL175556A0 (en) 2008-04-13
HK1102021A1 (en) 2007-11-02
TW200524597A (en) 2005-08-01
CA2544413A1 (fr) 2005-05-26

Similar Documents

Publication Publication Date Title
ZA200605631B (en) Directly compressible pharmaceutical composition for the oral administration of CCI-779
PL368636A1 (en) Pharmaceutical dosage forms of epothilones for oral administration
IL166489A (en) Oral dosage form in single-dose administration containing at least two layers for the administration and use of flipridone
PL356358A1 (en) Solid dosage form of someticone for oral administration
EP1757273A4 (en) PREPARATION FOR ORAL ADMINISTRATION
HK1107768A1 (en) Solid drug for oral use
AU2003303633A8 (en) Fast dissolving films for oral administration of drugs
AU2003246978A1 (en) Pharmaceutical compositions comprising cyclosporin for oral administration
PL372773A1 (en) Oral administration of epothilones
IL166337A0 (en) Oral administration of calctionin
AU2003245504A1 (en) Pharmaceutical compositions for drugs having ph-dependentsolubility
IL161143A0 (en) A flash-melt pharmaceutical oral dosage composition
HK1072194A1 (en) Oral dosage form for controlled drug release
EP1683525A4 (en) PREPARATION OF SUSTAINED RELEASE PHENYLALANINE DERIVATIVES FOR ORAL ADMINISTRATION
HK1102021A1 (en) Pharmaceutical composition for oral administration of a pyrazol-3- carboxamide derivative
HK1083768A1 (en) Sustained-release pharmaceutical composition for lung administration
AU2003284786A8 (en) Microemulsion composition for oral administration of biphenyldimethyldicarboxylate
EP1626697A4 (en) PHARMACEUTICAL COMPOSITIONS FOR ORAL ADMINISTRATION WITH LITHIUM CARBONATE
AU2003251643A1 (en) Pharmaceutical compositions containing keto-acids for endoperitoneal administration
ZA200603126B (en) Pharmaceutical compositions for therapeutic use
PL373776A1 (en) Oral pharmaceutical compound
AU2003244092A1 (en) 1ss-METHYLCARBAPENEM DERIVATIVE FOR ORAL ADMINISTRATION
HU0203985D0 (en) Use of a pharmaceutical composition for alleviating side effect of a disease
AU2003254672A8 (en) Dual-spike release formulation for oral drug delivery
GB0218994D0 (en) Oral pharmaceutical compositions