DE602004020797D1 - Pharmazeutische zusammensetzung für die orale verabreichung eines pyrazol-3-carbonsäurederivats - Google Patents

Pharmazeutische zusammensetzung für die orale verabreichung eines pyrazol-3-carbonsäurederivats

Info

Publication number
DE602004020797D1
DE602004020797D1 DE602004020797T DE602004020797T DE602004020797D1 DE 602004020797 D1 DE602004020797 D1 DE 602004020797D1 DE 602004020797 T DE602004020797 T DE 602004020797T DE 602004020797 T DE602004020797 T DE 602004020797T DE 602004020797 D1 DE602004020797 D1 DE 602004020797D1
Authority
DE
Germany
Prior art keywords
carboxylene
pyrazol
derivative
pharmaceutical composition
oral administration
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602004020797T
Other languages
English (en)
Inventor
Thierry Breul
Jean Claude Gautier
Olivier Saslawski
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi Aventis France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis France filed Critical Sanofi Aventis France
Publication of DE602004020797D1 publication Critical patent/DE602004020797D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
DE602004020797T 2003-11-10 2004-11-09 Pharmazeutische zusammensetzung für die orale verabreichung eines pyrazol-3-carbonsäurederivats Active DE602004020797D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0313259A FR2861992B1 (fr) 2003-11-10 2003-11-10 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3-carboxamide.
PCT/FR2004/002875 WO2005046690A1 (fr) 2003-11-10 2004-11-09 Composition pharmaceutique destinee a l'administration orale d'un derive de pyrazole-3­carboxamide

Publications (1)

Publication Number Publication Date
DE602004020797D1 true DE602004020797D1 (de) 2009-06-04

Family

ID=34508418

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602004020797T Active DE602004020797D1 (de) 2003-11-10 2004-11-09 Pharmazeutische zusammensetzung für die orale verabreichung eines pyrazol-3-carbonsäurederivats

Country Status (28)

Country Link
US (2) US20060264469A1 (de)
EP (1) EP1691808B1 (de)
JP (1) JP4767171B2 (de)
KR (1) KR20060108668A (de)
CN (1) CN100528158C (de)
AR (1) AR047237A1 (de)
AT (1) ATE429227T1 (de)
AU (1) AU2004289086A1 (de)
BR (1) BRPI0416341A (de)
CA (1) CA2544413A1 (de)
CY (1) CY1110478T1 (de)
DE (1) DE602004020797D1 (de)
DK (1) DK1691808T3 (de)
ES (1) ES2325373T3 (de)
FR (1) FR2861992B1 (de)
HK (1) HK1102021A1 (de)
HR (1) HRP20090393T1 (de)
IL (1) IL175556A (de)
MA (1) MA28419B1 (de)
NO (1) NO20062609L (de)
NZ (1) NZ547763A (de)
PL (1) PL1691808T3 (de)
PT (1) PT1691808E (de)
RU (1) RU2321404C1 (de)
SI (1) SI1691808T1 (de)
TW (1) TWI280129B (de)
WO (1) WO2005046690A1 (de)
ZA (1) ZA200604451B (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1880715A1 (de) * 2006-07-19 2008-01-23 Abbott GmbH & Co. KG Pharmazeutisch annehmbare lösungsvermittelnde Zusammensetzung und diese enthaltende pharmazeutische Darreichungsform
EP1920767A1 (de) * 2006-11-09 2008-05-14 Abbott GmbH & Co. KG Schmelzverarbeitete Darreichungsform mit Imatinib
PL2192893T3 (pl) * 2007-08-21 2015-12-31 Basilea Pharmaceutica Ag Kompozycja przeciwgrzybicza
MY158809A (en) * 2010-09-22 2016-11-15 Craun Res Sdn Bhd Pharmaceutical compositions for calanolides, their derivatives and analogues, and process for producing the same
US20130317117A1 (en) * 2010-11-24 2013-11-28 Pharmaceutics International, Inc. Self micro-emulsifying drug delivery system with increased bioavailability

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5059691A (en) * 1990-01-22 1991-10-22 American Cyanamid Company N-((dialkylamino)methylene)-substituted pyrazolo (1,5-A)-pyrimidine-3-carboxamides and N-((dialkylamino)methylene)-substituted-4,5-dihydropyrazolo-(1,5-A)-pyrimidine-3-carboxamides
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
ATE398448T1 (de) * 1993-09-28 2008-07-15 Scherer Gmbh R P Herstellung von weichgelatinekapseln
GB9405304D0 (en) * 1994-03-16 1994-04-27 Scherer Ltd R P Delivery systems for hydrophobic drugs
US5965160A (en) * 1995-04-24 1999-10-12 Yissum Research Development Company Of The Hebrew University Of Jerusalem Self-emulsifiable formulation producing an oil-in-water emulsion
EP0825849A1 (de) * 1995-05-19 1998-03-04 Abbott Laboratories Selbstemulgierbare arzneiformulierungen für lipophile arzneimittel
US5993858A (en) * 1996-06-14 1999-11-30 Port Systems L.L.C. Method and formulation for increasing the bioavailability of poorly water-soluble drugs
BR9808845A (pt) * 1997-03-14 2000-08-01 Otsuka Pharma Co Ltd Derivado de pirimidina, agentes para a cura de uma doença alérgica, da asma e de uma dermatite atópica, agentes para inibição da produção de no de tnf-alfa, de citoquinas e da 5-lipoxigenase, processos para curar uma doença alérgica, a asma e uma dermatite atópica e para inibir a produção de no, de tnf-alfa e de citoquinas e a 5-lipoxigenase e usos de um composto
FR2761265B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique pour l'administration orale d'un derive du n-piperidino-3-pyrazolecarboxamide, de ses sels et de leurs solvates
FR2761266B1 (fr) * 1997-03-28 1999-07-02 Sanofi Sa Composition pharmaceutique formee par granulation humide pour l'administration orale d'un derive du n-piperidino-3- pyrazolecarboxamide, de ses sels et de leurs solvates
US6617426B1 (en) * 1999-06-22 2003-09-09 Merck & Co Inc Cysteinyl protease inhibitors
JP2001151669A (ja) * 1999-11-24 2001-06-05 Nippon Kayaku Co Ltd 経口用自己乳化製剤
JP2003518485A (ja) * 1999-12-23 2003-06-10 ファイザー・プロダクツ・インク 向上された薬物濃度を与える医薬組成物
GB0001928D0 (en) * 2000-01-27 2000-03-22 Novartis Ag Organic compounds
FR2831883B1 (fr) * 2001-11-08 2004-07-23 Sanofi Synthelabo Forme polymorphe du rimonabant, son procede de preparation et les compositions pharmaceutiques en contenant
JP2005523295A (ja) * 2002-03-01 2005-08-04 ノバガリ、ファルマ、エスアー 難溶性薬剤の自己乳化型薬物送達システム
GB0216700D0 (en) * 2002-07-18 2002-08-28 Astrazeneca Ab Process

Also Published As

Publication number Publication date
WO2005046690A1 (fr) 2005-05-26
EP1691808A1 (de) 2006-08-23
DK1691808T3 (da) 2009-08-03
MA28419B1 (fr) 2007-02-01
US20090004261A1 (en) 2009-01-01
RU2006120447A (ru) 2007-12-20
AU2004289086A1 (en) 2005-05-26
IL175556A0 (en) 2008-04-13
US20060264469A1 (en) 2006-11-23
HRP20090393T1 (en) 2009-08-31
JP2007516960A (ja) 2007-06-28
EP1691808B1 (de) 2009-04-22
FR2861992B1 (fr) 2007-07-20
PT1691808E (pt) 2009-07-14
BRPI0416341A (pt) 2007-02-27
CN1925856A (zh) 2007-03-07
ES2325373T3 (es) 2009-09-02
FR2861992A1 (fr) 2005-05-13
CN100528158C (zh) 2009-08-19
IL175556A (en) 2010-11-30
HK1102021A1 (en) 2007-11-02
AR047237A1 (es) 2006-01-11
CA2544413A1 (fr) 2005-05-26
CY1110478T1 (el) 2015-04-29
TWI280129B (en) 2007-05-01
SI1691808T1 (sl) 2009-10-31
RU2321404C1 (ru) 2008-04-10
TW200524597A (en) 2005-08-01
ATE429227T1 (de) 2009-05-15
NZ547763A (en) 2009-08-28
NO20062609L (no) 2006-06-06
ZA200604451B (en) 2007-10-31
KR20060108668A (ko) 2006-10-18
PL1691808T3 (pl) 2009-09-30
JP4767171B2 (ja) 2011-09-07

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