SG43809A1 - 2-benzyl-polycyclic guanine derivatives and process for preparing them - Google Patents

2-benzyl-polycyclic guanine derivatives and process for preparing them

Info

Publication number
SG43809A1
SG43809A1 SG1996001116A SG1996001116A SG43809A1 SG 43809 A1 SG43809 A1 SG 43809A1 SG 1996001116 A SG1996001116 A SG 1996001116A SG 1996001116 A SG1996001116 A SG 1996001116A SG 43809 A1 SG43809 A1 SG 43809A1
Authority
SG
Singapore
Prior art keywords
benzyl
preparing
guanine derivatives
polycyclic guanine
polycyclic
Prior art date
Application number
SG1996001116A
Other languages
English (en)
Inventor
Deen Tulsian
Brian A Mckittrick
Yan Xia
Samuel Chackalamannil
Dinesh Gala
Donald J Dibenedetto
Max Kugelman
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of SG43809A1 publication Critical patent/SG43809A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52Two oxygen atoms
    • C07D239/54Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/40Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
SG1996001116A 1993-02-26 1994-02-24 2-benzyl-polycyclic guanine derivatives and process for preparing them SG43809A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2354993A 1993-02-26 1993-02-26
US2459993A 1993-02-26 1993-02-26

Publications (1)

Publication Number Publication Date
SG43809A1 true SG43809A1 (en) 1997-11-14

Family

ID=26697306

Family Applications (1)

Application Number Title Priority Date Filing Date
SG1996001116A SG43809A1 (en) 1993-02-26 1994-02-24 2-benzyl-polycyclic guanine derivatives and process for preparing them

Country Status (14)

Country Link
US (1) US5939419A (xx)
EP (1) EP0686157A1 (xx)
JP (1) JPH08507068A (xx)
KR (1) KR960701058A (xx)
CN (1) CN1118600A (xx)
AU (1) AU681875B2 (xx)
CA (1) CA2156918A1 (xx)
FI (1) FI953981A0 (xx)
HU (1) HUT72640A (xx)
IL (1) IL108754A0 (xx)
NZ (1) NZ262797A (xx)
SG (1) SG43809A1 (xx)
TW (1) TW270118B (xx)
WO (1) WO1994019351A1 (xx)

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US11464781B2 (en) 2009-02-25 2022-10-11 Intra-Cellular Therapies, Inc. PDE1 inhibitors for ophthalmic disorders
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Also Published As

Publication number Publication date
WO1994019351A1 (en) 1994-09-01
CA2156918A1 (en) 1994-09-01
TW270118B (xx) 1996-02-11
IL108754A0 (en) 1994-06-24
JPH08507068A (ja) 1996-07-30
CN1118600A (zh) 1996-03-13
AU6268794A (en) 1994-09-14
NZ262797A (en) 1997-08-22
FI953981A (fi) 1995-08-24
KR960701058A (ko) 1996-02-24
HU9502464D0 (en) 1995-10-30
HUT72640A (en) 1996-05-28
FI953981A0 (fi) 1995-08-24
AU681875B2 (en) 1997-09-11
EP0686157A1 (en) 1995-12-13
US5939419A (en) 1999-08-17

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