SG172735A1 - Method of modulating neurite outgrowth by the use of a galanin-3 receptor antagonist - Google Patents
Method of modulating neurite outgrowth by the use of a galanin-3 receptor antagonist Download PDFInfo
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- SG172735A1 SG172735A1 SG2011047032A SG2011047032A SG172735A1 SG 172735 A1 SG172735 A1 SG 172735A1 SG 2011047032 A SG2011047032 A SG 2011047032A SG 2011047032 A SG2011047032 A SG 2011047032A SG 172735 A1 SG172735 A1 SG 172735A1
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- aryl
- branched
- alkyl
- straight chained
- galanin
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- GPKUICFDWYEPTK-UHFFFAOYSA-N methoxycyclohexatriene Chemical class COC1=CC=C=C[CH]1 GPKUICFDWYEPTK-UHFFFAOYSA-N 0.000 description 1
- ZBELDPMWYXDLNY-UHFFFAOYSA-N methyl 9-(4-bromo-2-fluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate Chemical compound C12=C3SC(C(=N)OC)=NC3=CC=C2N=CN=C1NC1=CC=C(Br)C=C1F ZBELDPMWYXDLNY-UHFFFAOYSA-N 0.000 description 1
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- SLFVYFOEHHLHDW-UHFFFAOYSA-N n-(trifluoromethyl)aniline Chemical compound FC(F)(F)NC1=CC=CC=C1 SLFVYFOEHHLHDW-UHFFFAOYSA-N 0.000 description 1
- 125000004108 n-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])([H])C([H])([H])* 0.000 description 1
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- 230000003285 pharmacodynamic effect Effects 0.000 description 1
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- 125000005545 phthalimidyl group Chemical group 0.000 description 1
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- 239000000256 polyoxyethylene sorbitan monolaurate Substances 0.000 description 1
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- 239000000843 powder Substances 0.000 description 1
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- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 description 1
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- 102000004169 proteins and genes Human genes 0.000 description 1
- 108090000623 proteins and genes Proteins 0.000 description 1
- 125000001042 pteridinyl group Chemical group N1=C(N=CC2=NC=CN=C12)* 0.000 description 1
- 125000000561 purinyl group Chemical group N1=C(N=C2N=CNC2=C1)* 0.000 description 1
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- 125000004076 pyridyl group Chemical group 0.000 description 1
- 125000000714 pyrimidinyl group Chemical group 0.000 description 1
- 125000000168 pyrrolyl group Chemical group 0.000 description 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US81668206P | 2006-06-26 | 2006-06-26 |
Publications (1)
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|---|---|
| SG172735A1 true SG172735A1 (en) | 2011-07-28 |
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| Application Number | Title | Priority Date | Filing Date |
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| SG2011047032A SG172735A1 (en) | 2006-06-26 | 2007-06-26 | Method of modulating neurite outgrowth by the use of a galanin-3 receptor antagonist |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20080039496A1 (enExample) |
| EP (1) | EP2032135A2 (enExample) |
| JP (2) | JP2009541493A (enExample) |
| CN (1) | CN101484159A (enExample) |
| AU (1) | AU2007265088B2 (enExample) |
| BR (1) | BRPI0712938A2 (enExample) |
| CA (1) | CA2655829A1 (enExample) |
| IL (1) | IL195903A0 (enExample) |
| MX (1) | MX2008016083A (enExample) |
| SG (1) | SG172735A1 (enExample) |
| WO (1) | WO2008002946A2 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| US7642281B2 (en) * | 2002-08-07 | 2010-01-05 | Helicon Therapeutics, Inc. | Indolone compounds useful to treat cognitive impairment |
| US20100028839A1 (en) * | 2008-07-18 | 2010-02-04 | Tully Timothy P | Methods and systems for evaluating memory agents |
| EP2313098A4 (en) * | 2008-07-18 | 2011-12-21 | Dart Neuroscience Llc | METHOD AND SYSTEMS FOR THE ASSESSMENT OF MEMORY-PROMOTING ACTIVE SUBSTANCES |
| AU2012222869B2 (en) * | 2011-03-02 | 2015-08-13 | Bionomics Limited | Methods of treating a disease or condition of the central nervous system |
| US8277842B1 (en) | 2012-01-20 | 2012-10-02 | Dart Neuroscience (Cayman) Ltd. | Enteric-coated HT-2157 compositions and methods of their use |
| CR20160578A (es) * | 2014-06-26 | 2017-02-21 | Hoffmann La Roche | Derivados de indolin-2-ona o pirrolo-piridin-2-ona |
| CN108349942B (zh) | 2015-11-06 | 2021-03-30 | 豪夫迈·罗氏有限公司 | 用于治疗cns和相关疾病的二氢吲哚-2-酮衍生物 |
| CA3002489C (en) | 2015-11-06 | 2023-11-07 | F.Hoffmann-La Roche Ag | Indolin-2-one derivatives |
| JP6857651B2 (ja) | 2015-11-06 | 2021-04-14 | エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ | Ｃｎｓ疾患の処置に有用なインドリン−２−オン誘導体 |
| WO2017076842A1 (en) | 2015-11-06 | 2017-05-11 | F. Hoffmann-La Roche Ag | Indolin-2-one derivatives |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
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| US7081470B2 (en) * | 2001-01-31 | 2006-07-25 | H. Lundbeck A/S | Use of GALR3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods |
| US7220775B2 (en) * | 2002-08-07 | 2007-05-22 | H. Lundbeck A/S | Compound useful for the treatment of neuropathic pain |
-
2007
- 2007-06-26 MX MX2008016083A patent/MX2008016083A/es not_active Application Discontinuation
- 2007-06-26 SG SG2011047032A patent/SG172735A1/en unknown
- 2007-06-26 CN CNA2007800241434A patent/CN101484159A/zh active Pending
- 2007-06-26 AU AU2007265088A patent/AU2007265088B2/en not_active Ceased
- 2007-06-26 JP JP2009518522A patent/JP2009541493A/ja active Pending
- 2007-06-26 WO PCT/US2007/072166 patent/WO2008002946A2/en not_active Ceased
- 2007-06-26 US US11/768,889 patent/US20080039496A1/en not_active Abandoned
- 2007-06-26 CA CA002655829A patent/CA2655829A1/en not_active Abandoned
- 2007-06-26 BR BRPI0712938-6A patent/BRPI0712938A2/pt not_active IP Right Cessation
- 2007-06-26 EP EP07799059A patent/EP2032135A2/en not_active Withdrawn
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2008
- 2008-12-11 IL IL195903A patent/IL195903A0/en unknown
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2013
- 2013-08-15 JP JP2013168863A patent/JP2013227357A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JP2013227357A (ja) | 2013-11-07 |
| AU2007265088A1 (en) | 2008-01-03 |
| JP2009541493A (ja) | 2009-11-26 |
| EP2032135A2 (en) | 2009-03-11 |
| BRPI0712938A2 (pt) | 2013-03-26 |
| US20080039496A1 (en) | 2008-02-14 |
| WO2008002946A3 (en) | 2008-05-02 |
| MX2008016083A (es) | 2009-03-20 |
| CA2655829A1 (en) | 2008-01-03 |
| IL195903A0 (en) | 2009-09-01 |
| CN101484159A (zh) | 2009-07-15 |
| AU2007265088B2 (en) | 2013-05-23 |
| WO2008002946A2 (en) | 2008-01-03 |
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