SG170775A1 - 2 -aminopyridine analogs as glucokinase activators - Google Patents

2 -aminopyridine analogs as glucokinase activators

Info

Publication number
SG170775A1
SG170775A1 SG201102157-3A SG2011021573A SG170775A1 SG 170775 A1 SG170775 A1 SG 170775A1 SG 2011021573 A SG2011021573 A SG 2011021573A SG 170775 A1 SG170775 A1 SG 170775A1
Authority
SG
Singapore
Prior art keywords
glucokinase
glucokinase activators
aminopyridine
analogs
aminopyridine analogs
Prior art date
Application number
SG201102157-3A
Other languages
English (en)
Inventor
Thomas Daniel Aicher
Steven Armen Boyd
Mark Joseph Chicarelli
Kevin Ronald Condroski
Ronald Jay Hinklin
Ajay Singh
Original Assignee
Array Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Publication of SG170775A1 publication Critical patent/SG170775A1/en

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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
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  • Child & Adolescent Psychology (AREA)
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  • Gastroenterology & Hepatology (AREA)
SG201102157-3A 2006-03-24 2007-03-23 2 -aminopyridine analogs as glucokinase activators SG170775A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US78546006P 2006-03-24 2006-03-24

Publications (1)

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SG170775A1 true SG170775A1 (en) 2011-05-30

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SG201102157-3A SG170775A1 (en) 2006-03-24 2007-03-23 2 -aminopyridine analogs as glucokinase activators

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US (3) US8022223B2 (pt)
EP (2) EP2543667B1 (pt)
JP (2) JP5377284B2 (pt)
KR (1) KR101440634B1 (pt)
CN (1) CN101437816B (pt)
AU (1) AU2007235558B2 (pt)
BR (1) BRPI0709171A2 (pt)
CA (1) CA2647208C (pt)
DK (1) DK2013204T3 (pt)
ES (1) ES2536547T3 (pt)
HK (1) HK1128130A1 (pt)
HR (1) HRP20150347T1 (pt)
IL (1) IL194160A (pt)
MX (1) MX2008012168A (pt)
MY (1) MY148985A (pt)
NZ (1) NZ571997A (pt)
PL (1) PL2013204T3 (pt)
PT (1) PT2013204E (pt)
RS (1) RS53981B1 (pt)
RU (1) RU2457207C2 (pt)
SG (1) SG170775A1 (pt)
SI (1) SI2013204T1 (pt)
TW (1) TWI393718B (pt)
UA (1) UA103746C2 (pt)
WO (1) WO2007117381A2 (pt)
ZA (1) ZA200809017B (pt)

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US8431713B2 (en) * 2007-01-24 2013-04-30 Array Biopharma, Inc. 2-aminopyridine derivatives as glucokinase activators
WO2008118718A2 (en) * 2007-03-23 2008-10-02 Array Biopharma Inc. 2-aminopyridine analogs as glucokinase activators
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
EP2727910B1 (en) 2007-09-21 2016-03-16 Array Biopharma, Inc. Pyridin-2-yl-thiourea and Pyridin-2-yl-amine derivatives as intermediates for the preparation of Pyridin-2yl-amino-1,2,4-thiadiazole glucokinase activators
BRPI0818658A2 (pt) * 2007-10-09 2015-04-14 Merck Patent Ges Mit Beschränkter Haftung Derivados de piridina úteis como ativadores de glicoquinase
DK2239253T3 (da) * 2008-02-06 2013-09-23 Daiichi Sankyo Co Ltd Hidtil ukendt phenylpyrrolderivat
US7741327B2 (en) 2008-04-16 2010-06-22 Hoffmann-La Roche Inc. Pyrrolidinone glucokinase activators
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
CN105176930B (zh) 2010-03-31 2021-05-04 斯克里普斯研究所 重编程细胞
US8178689B2 (en) 2010-06-17 2012-05-15 Hoffman-La Roche Inc. Tricyclic compounds
WO2011157827A1 (de) 2010-06-18 2011-12-22 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
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