SG11201906373VA - Chemical compounds as inhibitors of interleukin-1 activity - Google Patents

Chemical compounds as inhibitors of interleukin-1 activity

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Publication number
SG11201906373VA
SG11201906373VA SG11201906373VA SG11201906373VA SG11201906373VA SG 11201906373V A SG11201906373V A SG 11201906373VA SG 11201906373V A SG11201906373V A SG 11201906373VA SG 11201906373V A SG11201906373V A SG 11201906373VA SG 11201906373V A SG11201906373V A SG 11201906373VA
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SG
Singapore
Prior art keywords
international
co7d
california
san diego
pct
Prior art date
Application number
SG11201906373VA
Other languages
English (en)
Inventor
Jeffrey A Stafford
James M Veal
Lynnie Lin Trzoss
Christopher Mcbride
Original Assignee
Genentech Inc
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Publication date
Application filed by Genentech Inc filed Critical Genentech Inc
Publication of SG11201906373VA publication Critical patent/SG11201906373VA/en

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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles
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    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • A61K31/4161,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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SG11201906373VA 2017-01-23 2018-01-22 Chemical compounds as inhibitors of interleukin-1 activity SG11201906373VA (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762449431P 2017-01-23 2017-01-23
US201762492813P 2017-05-01 2017-05-01
PCT/US2018/014728 WO2018136890A1 (en) 2017-01-23 2018-01-22 Chemical compounds as inhibitors of interleukin-1 activity

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