SG11201408491SA - Analogs of glucagon exhibiting gip receptor activity - Google Patents

Analogs of glucagon exhibiting gip receptor activity

Info

Publication number
SG11201408491SA
SG11201408491SA SG11201408491SA SG11201408491SA SG11201408491SA SG 11201408491S A SG11201408491S A SG 11201408491SA SG 11201408491S A SG11201408491S A SG 11201408491SA SG 11201408491S A SG11201408491S A SG 11201408491SA SG 11201408491S A SG11201408491S A SG 11201408491SA
Authority
SG
Singapore
Prior art keywords
lllll
international
indiana
gip receptor
analogs
Prior art date
Application number
SG11201408491SA
Other languages
English (en)
Inventor
Richard D Dimarchi
David L Smiley
Konrad H Bleicher
Eric A Kitas
Original Assignee
Univ Indiana Res & Tech Corp
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Indiana Res & Tech Corp, Hoffmann La Roche filed Critical Univ Indiana Res & Tech Corp
Publication of SG11201408491SA publication Critical patent/SG11201408491SA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Measurement And Recording Of Electrical Phenomena And Electrical Characteristics Of The Living Body (AREA)
  • Measuring Pulse, Heart Rate, Blood Pressure Or Blood Flow (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SG11201408491SA 2012-06-21 2013-06-18 Analogs of glucagon exhibiting gip receptor activity SG11201408491SA (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261662874P 2012-06-21 2012-06-21
US201361787973P 2013-03-15 2013-03-15
PCT/US2013/046229 WO2013192130A1 (en) 2012-06-21 2013-06-18 Analogs of glucagon exhibiting gip receptor activity

Publications (1)

Publication Number Publication Date
SG11201408491SA true SG11201408491SA (en) 2015-01-29

Family

ID=48692696

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201408491SA SG11201408491SA (en) 2012-06-21 2013-06-18 Analogs of glucagon exhibiting gip receptor activity

Country Status (30)

Country Link
US (2) US9868772B2 (sr)
EP (1) EP2864350B1 (sr)
JP (1) JP6300239B2 (sr)
KR (1) KR20150039748A (sr)
CN (1) CN104583233B (sr)
AR (1) AR091478A1 (sr)
AU (1) AU2013277372B2 (sr)
BR (1) BR112014031671A2 (sr)
CA (1) CA2877127A1 (sr)
CL (1) CL2014003421A1 (sr)
CO (1) CO7170125A2 (sr)
CR (1) CR20150015A (sr)
DK (1) DK2864350T3 (sr)
EA (1) EA029025B1 (sr)
ES (1) ES2674946T3 (sr)
HR (1) HRP20180936T1 (sr)
HU (1) HUE039267T2 (sr)
IL (1) IL236386B (sr)
MX (1) MX356000B (sr)
MY (1) MY185217A (sr)
PE (1) PE20150863A1 (sr)
PH (1) PH12014502857A1 (sr)
PL (1) PL2864350T3 (sr)
PT (1) PT2864350T (sr)
RS (1) RS57347B1 (sr)
SG (1) SG11201408491SA (sr)
SI (1) SI2864350T1 (sr)
TR (1) TR201808818T4 (sr)
TW (1) TWI644920B (sr)
WO (1) WO2013192130A1 (sr)

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TWI622596B (zh) 2015-10-26 2018-05-01 美國禮來大藥廠 升糖素受體促效劑
PL3393496T3 (pl) 2015-12-23 2024-04-22 The Johns Hopkins University Długo działający agonista glp-1r jako terapia stanów neurologicznych i neurodegeneracyjnych
EP3398961B1 (en) * 2015-12-31 2022-06-29 Hanmi Pharm. Co., Ltd. Triple activator activating glucagon, glp-1 and gip receptor
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SG11201811697SA (en) 2016-06-29 2019-01-30 Hanmi Pharmaceutical Co Ltd Glucagon derivative, conjugate thereof, composition comprising same and therapeutic use thereof
TW201833132A (zh) 2016-12-02 2018-09-16 法商賽諾菲公司 作為肽類ｇｌｐ１／升糖素／ｇｉｐ三重受體激動劑之新穎化合物
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TW202015735A (zh) 2018-05-30 2020-05-01 法商賽諾菲公司 包含ｇｌｐ－１／升糖素／ｇｉｐ三重受體促效劑、連接子及透明質酸之接合物
US11166910B2 (en) 2019-01-25 2021-11-09 Nordiccan A/S Cannabinoid chewing gum with sugar alcohols
CN114945589B (zh) * 2020-02-24 2024-05-24 深圳市图微安创科技开发有限公司 多肽化合物及其在预防或治疗糖尿病或糖尿病并发症中的应用
CN113493503B (zh) * 2020-04-08 2022-08-05 浙江道尔生物科技有限公司 一种肠促胰岛素类似物及其制备方法和用途
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WO2022156189A1 (zh) * 2021-01-22 2022-07-28 深圳市图微安创科技开发有限公司 多肽化合物在预防或治疗炎症性肠病及其相关的肠纤维化中的应用
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Also Published As

Publication number Publication date
IL236386B (en) 2019-09-26
CN104583233B (zh) 2018-10-23
HRP20180936T1 (hr) 2018-12-14
MY185217A (en) 2021-04-30
CN104583233A (zh) 2015-04-29
US20180105569A1 (en) 2018-04-19
HUE039267T2 (hu) 2018-12-28
MX2014015556A (es) 2015-03-05
DK2864350T3 (en) 2018-05-28
CR20150015A (es) 2015-04-24
US9868772B2 (en) 2018-01-16
AU2013277372A1 (en) 2014-12-11
MX356000B (es) 2018-05-08
TR201808818T4 (tr) 2018-07-23
RS57347B1 (sr) 2018-08-31
EA201590065A1 (ru) 2015-07-30
IL236386A0 (en) 2015-02-26
PH12014502857A1 (en) 2015-02-23
PE20150863A1 (es) 2015-06-11
CL2014003421A1 (es) 2015-05-22
CO7170125A2 (es) 2015-01-28
PL2864350T3 (pl) 2019-01-31
US20150368310A1 (en) 2015-12-24
AU2013277372B2 (en) 2018-03-29
ES2674946T3 (es) 2018-07-05
JP2015528795A (ja) 2015-10-01
EA029025B1 (ru) 2018-01-31
EP2864350A1 (en) 2015-04-29
TWI644920B (zh) 2018-12-21
CA2877127A1 (en) 2013-12-27
BR112014031671A2 (pt) 2018-08-07
AR091478A1 (es) 2015-02-04
SI2864350T1 (en) 2018-08-31
WO2013192130A1 (en) 2013-12-27
EP2864350B1 (en) 2018-03-28
TW201402603A (zh) 2014-01-16
KR20150039748A (ko) 2015-04-13
PT2864350T (pt) 2018-05-14
JP6300239B2 (ja) 2018-03-28

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