SG11201400974VA - Crystal of 5-hydroxy-1h-imidazole-4-carboxamideˑ3/4 hydrate, method for producing the same and crystal of 5-hydroxy-1h-imidazole-4-carboxamide hydrate - Google Patents

Crystal of 5-hydroxy-1h-imidazole-4-carboxamideˑ3/4 hydrate, method for producing the same and crystal of 5-hydroxy-1h-imidazole-4-carboxamide hydrate

Info

Publication number
SG11201400974VA
SG11201400974VA SG11201400974VA SG11201400974VA SG11201400974VA SG 11201400974V A SG11201400974V A SG 11201400974VA SG 11201400974V A SG11201400974V A SG 11201400974VA SG 11201400974V A SG11201400974V A SG 11201400974VA SG 11201400974V A SG11201400974V A SG 11201400974VA
Authority
SG
Singapore
Prior art keywords
imidazole
hydroxy
crystal
hydrate
producing
Prior art date
Application number
SG11201400974VA
Other languages
English (en)
Inventor
Taisuke Fujimoto
Tomohiro Hashimoto
Katsuyuki Hayashi
Tomoyuki Tanaka
Original Assignee
Fujifilm Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujifilm Corp filed Critical Fujifilm Corp
Publication of SG11201400974VA publication Critical patent/SG11201400974VA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
SG11201400974VA 2011-09-28 2012-09-28 Crystal of 5-hydroxy-1h-imidazole-4-carboxamideˑ3/4 hydrate, method for producing the same and crystal of 5-hydroxy-1h-imidazole-4-carboxamide hydrate SG11201400974VA (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2011213500 2011-09-28
JP2011213501 2011-09-28
PCT/JP2012/075106 WO2013047758A1 (ja) 2011-09-28 2012-09-28 5-ヒドロキシ-1h-イミダゾール-4-カルボキサミド水和物の結晶及び5-ヒドロキシ-1h-イミダゾール-4-カルボキサミド・3/4水和物の結晶及びその製造方法

Publications (1)

Publication Number Publication Date
SG11201400974VA true SG11201400974VA (en) 2014-09-26

Family

ID=47995783

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201400974VA SG11201400974VA (en) 2011-09-28 2012-09-28 Crystal of 5-hydroxy-1h-imidazole-4-carboxamideˑ3/4 hydrate, method for producing the same and crystal of 5-hydroxy-1h-imidazole-4-carboxamide hydrate

Country Status (13)

Country Link
US (2) US9108928B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP2762469B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR101970509B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN103827093B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU2012317424B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BR (1) BR112014007436A2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA2850196A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (2) IL231677A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IN (1) IN2014CN02346A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (1) MX354498B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
RU (2) RU2672560C1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SG (1) SG11201400974VA (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
WO (1) WO2013047758A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2672560C1 (ru) 2011-09-28 2018-11-16 Фуджифилм Корпорэйшн Кристалл гидрата 5-гидрокси-1Н-имидазол-4-карбоксамида и фармацевтическая композиция на его основе
WO2014112529A1 (ja) * 2013-01-15 2014-07-24 富士フイルム株式会社 5-ヒドロキシ-1h-イミダゾール-4-カルボキサミドの硫酸塩
CN105899951B (zh) * 2014-01-10 2019-07-12 富士胶片株式会社 5-羟基-1h-咪唑-4-甲酰胺的有效给予量的预测装置、黄苷一磷酸的量的测定方法
JP6823660B2 (ja) * 2016-09-13 2021-02-03 富士フイルム株式会社 Mll関連白血病の予防または治療のための医薬、方法、使用及び化合物
EP3686189B1 (en) * 2017-10-27 2021-09-01 FUJIFILM Corporation Production method for 5-hydroxy-1h-imidazole-4-carboxamide-3/4hydrate

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4181731A (en) * 1976-09-07 1980-01-01 Sumitomo Chemical Company, Limited Novel therapeutic application of 4-carbamoyl-5-hydroxyimidazole
JPS5625165A (en) * 1979-08-08 1981-03-10 Sumitomo Chem Co Ltd Novel imidazole derivative
JPS5824569A (ja) 1981-08-05 1983-02-14 Sumitomo Chem Co Ltd イミダゾ−ル誘導体の精製方法
US4503235A (en) * 1983-03-11 1985-03-05 Warner-Lambert Company Process for producing 4-carbamoyl-1H-imidazolium-5-olate
JPS60185727A (ja) 1984-03-05 1985-09-21 Sumitomo Chem Co Ltd 4−カルバモイルイミダゾリウム−5−オレ−ト製剤の安定化法
US5567816A (en) 1994-07-26 1996-10-22 Syntex (U.S.A.) Inc. Preparation of acyclovir using 1,3 dioxolane
CA2152863A1 (en) 1994-07-26 1996-01-27 Yeun-Kwei Han Preparation of acyclovir
US7002023B2 (en) 2000-09-29 2006-02-21 Basf Aktiengesellschaft Method for producing 1 substituted 5-chloro-4 methly pyrazoles
JP2002265601A (ja) 2001-03-07 2002-09-18 Rikogaku Shinkokai イミド樹脂
EP1874734A1 (en) * 2005-02-16 2008-01-09 Solvay Pharmaceuticals B.V. 1h-imidiazole derivatives as cannabinoid cb2 receptor modulators
CN101395141A (zh) * 2006-02-24 2009-03-25 莱西肯医药有限公司 咪唑基化合物,包含其的组合物和它们的使用方法
JP5266010B2 (ja) 2007-09-14 2013-08-21 富士フイルム株式会社 4−カルバモイル−5−ヒドロキシ−イミダゾール誘導体のスルホン酸塩化合物
KR100982720B1 (ko) * 2008-02-04 2010-09-17 주식회사 파마코스텍 4-카르바모일-1-β-D-리보푸라노실이미다졸륨-5-올레이트의 생산을 위한 중간체로서의 2-아미노말론아미드의제조방법
RU2672560C1 (ru) 2011-09-28 2018-11-16 Фуджифилм Корпорэйшн Кристалл гидрата 5-гидрокси-1Н-имидазол-4-карбоксамида и фармацевтическая композиция на его основе
TWI573791B (zh) 2011-09-28 2017-03-11 富士軟片股份有限公司 5-羥基-1h-咪唑-4-甲醯胺.3/4水合物及其結晶之製造方法

Also Published As

Publication number Publication date
MX2014003638A (es) 2014-05-21
EP2762469A1 (en) 2014-08-06
MX354498B (es) 2018-03-08
AU2012317424A8 (en) 2014-07-03
IL246754A (en) 2017-08-31
US20140275568A1 (en) 2014-09-18
RU2014111810A (ru) 2015-11-10
HK1197406A1 (zh) 2015-01-16
IL231677A0 (en) 2014-05-28
AU2012317424B2 (en) 2017-05-18
KR20140069052A (ko) 2014-06-09
KR101970509B1 (ko) 2019-04-19
US9108928B2 (en) 2015-08-18
RU2630682C2 (ru) 2017-09-12
IN2014CN02346A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 2015-06-19
EP2762469A4 (en) 2015-01-14
RU2672560C1 (ru) 2018-11-16
NZ622928A (en) 2015-04-24
US20150315156A1 (en) 2015-11-05
BR112014007436A2 (pt) 2017-04-04
WO2013047758A1 (ja) 2013-04-04
US9567303B2 (en) 2017-02-14
CA2850196A1 (en) 2013-04-04
CN103827093A (zh) 2014-05-28
AU2012317424A1 (en) 2014-04-17
IL231677A (en) 2017-01-31
CN103827093B (zh) 2016-06-15
EP2762469B1 (en) 2016-11-23

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