SG10201502588UA - Combination, kit and method of reducing intraocular pressure - Google Patents

Combination, kit and method of reducing intraocular pressure

Info

Publication number
SG10201502588UA
SG10201502588UA SG10201502588UA SG10201502588UA SG10201502588UA SG 10201502588U A SG10201502588U A SG 10201502588UA SG 10201502588U A SG10201502588U A SG 10201502588UA SG 10201502588U A SG10201502588U A SG 10201502588UA SG 10201502588U A SG10201502588U A SG 10201502588UA
Authority
SG
Singapore
Prior art keywords
kit
combination
intraocular pressure
reducing intraocular
reducing
Prior art date
Application number
SG10201502588UA
Other languages
English (en)
Inventor
Norman N Kim
William K Mcvicar
Thomas Mccauley
Rudolf A Baumgartner
Original Assignee
Inotek Pharmaceuticals Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44258984&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG10201502588U(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Inotek Pharmaceuticals Corp filed Critical Inotek Pharmaceuticals Corp
Publication of SG10201502588UA publication Critical patent/SG10201502588UA/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
    • A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
SG10201502588UA 2010-01-11 2011-01-11 Combination, kit and method of reducing intraocular pressure SG10201502588UA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US29380610P 2010-01-11 2010-01-11

Publications (1)

Publication Number Publication Date
SG10201502588UA true SG10201502588UA (en) 2015-05-28

Family

ID=44258984

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10201502588UA SG10201502588UA (en) 2010-01-11 2011-01-11 Combination, kit and method of reducing intraocular pressure
SG2012047882A SG182285A1 (en) 2010-01-11 2011-01-11 Combination, kit and method of reducing intraocular pressure

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG2012047882A SG182285A1 (en) 2010-01-11 2011-01-11 Combination, kit and method of reducing intraocular pressure

Country Status (28)

Country Link
US (3) US8877732B2 (es)
EP (1) EP2523669B1 (es)
JP (2) JP2013516495A (es)
KR (1) KR20120115344A (es)
CN (1) CN102711771B (es)
AU (1) AU2011203897B2 (es)
BR (1) BR112012017106A2 (es)
CA (1) CA2784908A1 (es)
CL (1) CL2012001912A1 (es)
CO (1) CO6571924A2 (es)
CY (1) CY1118510T1 (es)
DK (1) DK2523669T3 (es)
EA (1) EA025415B1 (es)
ES (1) ES2613698T3 (es)
HR (1) HRP20170007T1 (es)
HU (1) HUE030566T2 (es)
IL (1) IL220604A (es)
IN (1) IN2012DN06592A (es)
LT (1) LT2523669T (es)
ME (1) ME02608B (es)
MX (1) MX2012007661A (es)
PL (1) PL2523669T3 (es)
PT (1) PT2523669T (es)
RS (1) RS55615B1 (es)
SG (2) SG10201502588UA (es)
SI (1) SI2523669T1 (es)
SM (1) SMT201700017B (es)
WO (1) WO2011085361A1 (es)

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PL2424546T3 (pl) * 2009-05-01 2016-04-29 Inotek Pharmaceuticals Corp Sposób obniżania ciśnienia wewnątrzgałkowego u ludzi
EP2523669B1 (en) 2010-01-11 2016-12-07 Inotek Pharmaceuticals Corporation Combination, kit and method of reducing intraocular pressure
WO2011119969A1 (en) 2010-03-26 2011-09-29 Inotek Pharmaceuticals Corporation Method of reducing intraocular pressure in humans using n6 -cyclopentyladenosine (cpa), cpa derivatives or prodrugs thereof
US9278991B2 (en) 2012-01-26 2016-03-08 Inotek Pharmaceuticals Corporation Anhydrous polymorphs of [(2R,3S,4R,5R)-5-(6-(cyclopentylamino)-9H-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl)} methyl nitrate and processes of preparation thereof
US9522160B2 (en) * 2013-03-15 2016-12-20 Inotek Pharmaceuticals Corporation Ophthalmic formulations
BR112015022044A2 (pt) * 2013-03-15 2017-07-18 Inotek Pharmaceuticals Corp um método de proporcionar neutroproteção ocular
AU2015336458B2 (en) 2014-10-24 2018-05-10 Ono Pharmaceutical Co., Ltd. KCNQ2-5 channel activator
MX2017007318A (es) * 2014-12-03 2017-08-25 Inotek Pharmaceuticals Corp Metodos de prevencion, reduccion o tratamiento de degeneracion macular.

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US9370530B2 (en) 2016-06-21
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US20110172177A1 (en) 2011-07-14
IL220604A (en) 2017-01-31
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DK2523669T3 (en) 2017-02-06
EP2523669A4 (en) 2013-08-28
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US20160367586A1 (en) 2016-12-22
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