SE8204640L - Aminosyraderivat - Google Patents
AminosyraderivatInfo
- Publication number
- SE8204640L SE8204640L SE8204640A SE8204640A SE8204640L SE 8204640 L SE8204640 L SE 8204640L SE 8204640 A SE8204640 A SE 8204640A SE 8204640 A SE8204640 A SE 8204640A SE 8204640 L SE8204640 L SE 8204640L
- Authority
- SE
- Sweden
- Prior art keywords
- radical
- acid
- aminophosphonoheptanoic
- isomers
- stands
- Prior art date
Links
- 150000003862 amino acid derivatives Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 239000002253 acid Substances 0.000 abstract 2
- 125000004432 carbon atom Chemical group C* 0.000 abstract 2
- WBMSPCNOBZLEOF-UHFFFAOYSA-N 2-[aminooxy(hydroxy)phosphoryl]heptanoic acid Chemical compound CCCCCC(C(O)=O)P(O)(=O)ON WBMSPCNOBZLEOF-UHFFFAOYSA-N 0.000 abstract 1
- ABLZXFCXXLZCGV-UHFFFAOYSA-N Phosphorous acid Chemical compound OP(O)=O ABLZXFCXXLZCGV-UHFFFAOYSA-N 0.000 abstract 1
- 230000002378 acidificating effect Effects 0.000 abstract 1
- 125000004450 alkenylene group Chemical group 0.000 abstract 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- ZADPBFCGQRWHPN-UHFFFAOYSA-N boronic acid Chemical compound OBO ZADPBFCGQRWHPN-UHFFFAOYSA-N 0.000 abstract 1
- 210000003169 central nervous system Anatomy 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- BDHFUVZGWQCTTF-UHFFFAOYSA-N sulfonic acid Chemical compound OS(=O)=O BDHFUVZGWQCTTF-UHFFFAOYSA-N 0.000 abstract 1
- 150000003536 tetrazoles Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
- C07F9/3808—Acyclic saturated acids which can have further substituents on alkyl
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
- C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
- C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8124899 | 1981-08-14 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SE8204640D0 SE8204640D0 (sv) | 1982-08-10 |
| SE8204640L true SE8204640L (sv) | 1983-02-15 |
Family
ID=10523950
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE8204640A SE8204640L (sv) | 1981-08-14 | 1982-08-10 | Aminosyraderivat |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US4477391A (sv) |
| JP (1) | JPS58131957A (sv) |
| BE (1) | BE894116A (sv) |
| CH (1) | CH656613A5 (sv) |
| DE (1) | DE3229893A1 (sv) |
| FR (1) | FR2511378B1 (sv) |
| HK (1) | HK56085A (sv) |
| IT (1) | IT1201955B (sv) |
| LU (1) | LU84335A1 (sv) |
| MY (1) | MY8600145A (sv) |
| NL (1) | NL8203167A (sv) |
| SE (1) | SE8204640L (sv) |
| SG (1) | SG35385G (sv) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4906621A (en) * | 1985-05-24 | 1990-03-06 | Ciba-Geigy Corporation | Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade |
| US5217963A (en) * | 1985-05-24 | 1993-06-08 | Ciba-Geigy Corporation | Certain phosphonic acid quinoline-2-carboxylic acids, esters or amides useful for treatment of disorders responsive to N-methyl D-aspartate receptor blockade |
| US5175344A (en) * | 1986-02-13 | 1992-12-29 | Ciba-Geigy Corporation | Unsaturated amino acids |
| US5051413A (en) * | 1986-02-13 | 1991-09-24 | Ciba-Geigy Corporation | Unsaturated amino acids |
| ES2038690T3 (es) * | 1986-02-13 | 1993-08-01 | Ciba-Geigy Ag | Aminoacidos insaturados. |
| US4746653A (en) * | 1986-02-28 | 1988-05-24 | Ciba-Geigy Corporation | Certain hetero phosphonic acid derivatives of 2-piperidine or 2-tetrahydropyridinecarboxylates and esters thereof which are useful for the treatment of disorders responsive to blockade of the NMDA receptor in mammals |
| US4761405A (en) * | 1987-03-04 | 1988-08-02 | Nova Pharmaceutical Corporation | Antagonists of specific excitatory amino acid neurotransmitter receptors having increased potency |
| EP0391850B1 (de) * | 1989-04-07 | 1994-09-28 | Ciba-Geigy Ag | Ungesättigte Aminodicarbonsäurederivate |
| US5294734A (en) * | 1989-09-26 | 1994-03-15 | Ciba-Geigy Corp. | 4-substituted 2-aminoalk-3-enoic acids |
| US5488140A (en) * | 1989-09-26 | 1996-01-30 | Ciba-Geigy Corporation | 4-substituted 2-aminoalk-3-enoic |
| US5157149A (en) * | 1991-06-04 | 1992-10-20 | The United States Of America As Represented By The United States Department Of Energy | Enantioselective synthesis of L-(-)-4- boronophenylalanine (L-BPA) |
| CA2305703A1 (en) * | 1997-10-10 | 1999-04-22 | David W. Christianson | Compositions and methods for inhibiting arginase activity |
| WO1999024015A1 (en) * | 1997-11-12 | 1999-05-20 | Alza Corporation | Buffered drug formulations for transdermal electrotransport delivery |
| US20040063666A1 (en) * | 1998-10-09 | 2004-04-01 | David Christianson | Compositions for inhibiting arginase activity |
| SI2389352T1 (sl) * | 2009-01-26 | 2019-08-30 | The Trustees Of The University Of Pennsylvania, Center For Technology Transfer | Inhibitorji arginaze in postopki uporabe |
| WO2012091757A1 (en) | 2010-12-31 | 2012-07-05 | Corridor Pharmaceuticals, Inc. | Arginase inhibitors and methods of use thereof |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2870201A (en) * | 1955-04-04 | 1959-01-20 | Maxwell A Pollack | Synthesis of amino acids |
| US2934561A (en) * | 1955-09-28 | 1960-04-26 | Du Pont | Optically active salts of lysine and butane-2-sulfonic acid |
| US3405165A (en) * | 1965-10-23 | 1968-10-08 | Parke Davis & Co | Sulfonic acid compound |
| US4001322A (en) * | 1969-05-28 | 1977-01-04 | Eli Lilly And Company | 3-substituted phenylalkyl amines |
| US3977860A (en) * | 1971-08-09 | 1976-08-31 | Monsanto Company | Herbicidal compositions and methods employing esters of N-phosphonomethylglycine |
| US3860636A (en) * | 1972-12-06 | 1975-01-14 | Merck & Co Inc | Substituted indenyl phosphonic acids having anti-inflammatory activity |
| DE2717440C2 (de) * | 1976-05-17 | 1984-04-05 | Hoechst Ag, 6230 Frankfurt | Unkrautbekämpfung mit [(3-Amino-3-carboxy)-propyl-1]-methylphosphinsäure-Derivaten |
| GB1542938A (en) * | 1976-05-21 | 1979-03-28 | Ciba Geigy Ag | Aminophosphonous acids and processes for their preparation |
| JPS5387314A (en) * | 1977-01-07 | 1978-08-01 | Heiichi Sakai | Nn14099substance |
-
1982
- 1982-03-08 US US06/356,036 patent/US4477391A/en not_active Expired - Fee Related
- 1982-08-10 SE SE8204640A patent/SE8204640L/sv unknown
- 1982-08-11 DE DE19823229893 patent/DE3229893A1/de not_active Withdrawn
- 1982-08-12 NL NL8203167A patent/NL8203167A/nl not_active Application Discontinuation
- 1982-08-13 IT IT22834/82A patent/IT1201955B/it active
- 1982-08-13 LU LU84335A patent/LU84335A1/fr unknown
- 1982-08-13 CH CH4869/82A patent/CH656613A5/fr not_active IP Right Cessation
- 1982-08-13 BE BE0/208817A patent/BE894116A/fr not_active IP Right Cessation
- 1982-08-13 FR FR8214108A patent/FR2511378B1/fr not_active Expired
- 1982-08-14 JP JP57141586A patent/JPS58131957A/ja active Pending
- 1982-10-14 US US06/434,361 patent/US4483853A/en not_active Expired - Fee Related
-
1985
- 1985-05-09 SG SG353/85A patent/SG35385G/en unknown
- 1985-07-25 HK HK560/85A patent/HK56085A/xx unknown
-
1986
- 1986-12-30 MY MY145/86A patent/MY8600145A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FR2511378A1 (fr) | 1983-02-18 |
| FR2511378B1 (fr) | 1986-01-24 |
| MY8600145A (en) | 1986-12-31 |
| IT8222834A0 (it) | 1982-08-13 |
| SE8204640D0 (sv) | 1982-08-10 |
| NL8203167A (nl) | 1983-03-01 |
| JPS58131957A (ja) | 1983-08-06 |
| US4483853A (en) | 1984-11-20 |
| LU84335A1 (fr) | 1983-02-28 |
| HK56085A (en) | 1985-08-02 |
| CH656613A5 (fr) | 1986-07-15 |
| SG35385G (en) | 1985-11-15 |
| IT1201955B (it) | 1989-02-02 |
| DE3229893A1 (de) | 1983-03-31 |
| BE894116A (fr) | 1983-02-14 |
| US4477391A (en) | 1984-10-16 |
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