SE444679B - Sett att framstella 5(6)-substituerad bensimidazol-(2)-metylkarbamat med antihelmintisk verkan - Google Patents

Sett att framstella 5(6)-substituerad bensimidazol-(2)-metylkarbamat med antihelmintisk verkan

Info

Publication number
SE444679B
SE444679B SE7804305A SE7804305A SE444679B SE 444679 B SE444679 B SE 444679B SE 7804305 A SE7804305 A SE 7804305A SE 7804305 A SE7804305 A SE 7804305A SE 444679 B SE444679 B SE 444679B
Authority
SE
Sweden
Prior art keywords
general formula
give
substituted benzimidazole
antihelmintic
make
Prior art date
Application number
SE7804305A
Other languages
English (en)
Swedish (sv)
Other versions
SE7804305L (sv
Inventor
P Piccardi
G Confalonieri
P G Ramella
Col L Da
Original Assignee
Montedison Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Montedison Spa filed Critical Montedison Spa
Publication of SE7804305L publication Critical patent/SE7804305L/xx
Publication of SE444679B publication Critical patent/SE444679B/sv

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30—Nitrogen atoms not forming part of a nitro radical
    • C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
SE7804305A 1977-04-20 1978-04-17 Sett att framstella 5(6)-substituerad bensimidazol-(2)-metylkarbamat med antihelmintisk verkan SE444679B (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT22645/77A IT1076022B (it) 1977-04-20 1977-04-20 Benzimidazolcarbammati antielmintici

Publications (2)

Publication Number Publication Date
SE7804305L SE7804305L (sv) 1978-10-21
SE444679B true SE444679B (sv) 1986-04-28

Family

ID=11198787

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7804305A SE444679B (sv) 1977-04-20 1978-04-17 Sett att framstella 5(6)-substituerad bensimidazol-(2)-metylkarbamat med antihelmintisk verkan

Country Status (19)

Country Link
US (1) US4182893A (xx)
AR (1) AR219526A1 (xx)
AT (1) AT356672B (xx)
AU (1) AU520133B2 (xx)
BE (1) BE866195A (xx)
BR (1) BR7802445A (xx)
CA (1) CA1104142A (xx)
CH (1) CH639077A5 (xx)
DE (1) DE2816694C2 (xx)
DK (1) DK154076C (xx)
FR (1) FR2387965A1 (xx)
GB (1) GB1581517A (xx)
IE (1) IE46869B1 (xx)
IT (1) IT1076022B (xx)
NL (1) NL7804049A (xx)
NZ (1) NZ187003A (xx)
SE (1) SE444679B (xx)
SU (1) SU764609A3 (xx)
ZA (1) ZA782250B (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4174400A (en) * 1978-09-13 1979-11-13 Merck & Co., Inc. Anthelmintic benzimidazoles
DE2845537A1 (de) * 1978-10-19 1980-04-30 Bayer Ag Benzimidazolylcarbamidsaeureester, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
DK157547C (da) * 1978-12-06 1990-06-25 Montedison Spa Analogifremgangsmaade til fremstilling af 5(6)-substituerede benzimidazolcarbamater.
US4299837A (en) 1979-12-05 1981-11-10 Montedison S.P.A. Anthelmintic benzimidazole-carbamates

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK131821C (da) * 1967-03-22 1976-03-08 Smith Kline French Lab Analogifremgangsmade til fremstilling af en 2-karbalkoksyaminobenzimidazol
US3657267A (en) * 1969-06-20 1972-04-18 Janssen Pharmaceutica Nv Benzimidazole carbamates
BE793358A (fr) * 1971-12-27 1973-06-27 Hoechst Ag Nouveaux derives de 2-carbalcoxy-amino-benzimidazole presentantune activite anthelmintique et leur procede de preparation
US3929821A (en) * 1972-12-29 1975-12-30 Syntex Inc 5 (6)-Benzene ring substituted benzimidazole-2-carbamate derivatives
US3929824A (en) * 1972-12-29 1975-12-30 Syntex Inc 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US3929823A (en) * 1973-11-21 1975-12-30 Syntex Inc 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US3915986A (en) * 1974-06-19 1975-10-28 Smithkline Corp Methyl 5-propylthio-2-benzimidazolecarbamate

Also Published As

Publication number Publication date
DE2816694C2 (de) 1986-02-06
IT1076022B (it) 1985-04-22
AT356672B (de) 1980-05-12
SE7804305L (sv) 1978-10-21
DK166278A (da) 1978-10-21
US4182893A (en) 1980-01-08
FR2387965B1 (xx) 1980-10-10
CA1104142A (en) 1981-06-30
DK154076B (da) 1988-10-10
DE2816694A1 (de) 1978-10-26
AU3519378A (en) 1979-10-25
AU520133B2 (en) 1982-01-14
BE866195A (fr) 1978-10-20
AR219526A1 (es) 1980-08-29
GB1581517A (en) 1980-12-17
DK154076C (da) 1989-02-27
NL7804049A (nl) 1978-10-24
IE780769L (en) 1978-10-20
ATA272878A (de) 1979-10-15
SU764609A3 (ru) 1980-09-15
ZA782250B (en) 1979-04-25
NZ187003A (en) 1981-03-16
IE46869B1 (en) 1983-10-19
FR2387965A1 (fr) 1978-11-17
BR7802445A (pt) 1978-12-19
CH639077A5 (it) 1983-10-31

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