SE437516B - Analogiforfarande for framstellning av n-fenyl-n-(4-piperidyl)amidderivat - Google Patents

Analogiforfarande for framstellning av n-fenyl-n-(4-piperidyl)amidderivat

Info

Publication number
SE437516B
SE437516B SE7805110A SE7805110A SE437516B SE 437516 B SE437516 B SE 437516B SE 7805110 A SE7805110 A SE 7805110A SE 7805110 A SE7805110 A SE 7805110A SE 437516 B SE437516 B SE 437516B
Authority
SE
Sweden
Prior art keywords
formula
parts
tetrazol
lower alkyl
dihydrogen
Prior art date
Application number
SE7805110A
Other languages
English (en)
Swedish (sv)
Other versions
SE7805110L (sv
Inventor
F E Janssens
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of SE7805110L publication Critical patent/SE7805110L/xx
Publication of SE437516B publication Critical patent/SE437516B/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04—Five-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
SE7805110A 1977-05-05 1978-05-03 Analogiforfarande for framstellning av n-fenyl-n-(4-piperidyl)amidderivat SE437516B (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79381477A 1977-05-05 1977-05-05
US88618878A 1978-03-13 1978-03-13

Publications (2)

Publication Number Publication Date
SE7805110L SE7805110L (sv) 1978-11-06
SE437516B true SE437516B (sv) 1985-03-04

Family

ID=27121432

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7805110A SE437516B (sv) 1977-05-05 1978-05-03 Analogiforfarande for framstellning av n-fenyl-n-(4-piperidyl)amidderivat

Country Status (26)

Country Link
JP (1) JPS53149980A (enrdf_load_html_response)
AT (1) AT368994B (enrdf_load_html_response)
AU (1) AU514360B2 (enrdf_load_html_response)
CA (1) CA1105464A (enrdf_load_html_response)
CH (1) CH635585A5 (enrdf_load_html_response)
CY (1) CY1253A (enrdf_load_html_response)
DE (1) DE2819873A1 (enrdf_load_html_response)
DK (1) DK152211C (enrdf_load_html_response)
ES (1) ES469473A1 (enrdf_load_html_response)
FI (1) FI64364C (enrdf_load_html_response)
FR (1) FR2389622B1 (enrdf_load_html_response)
GB (1) GB1598872A (enrdf_load_html_response)
HK (1) HK72585A (enrdf_load_html_response)
HU (1) HU179204B (enrdf_load_html_response)
IE (1) IE46836B1 (enrdf_load_html_response)
IL (1) IL54639A (enrdf_load_html_response)
IT (1) IT1105288B (enrdf_load_html_response)
KE (1) KE3429A (enrdf_load_html_response)
LU (1) LU79575A1 (enrdf_load_html_response)
NL (1) NL186861C (enrdf_load_html_response)
NO (1) NO148747C (enrdf_load_html_response)
NZ (1) NZ187164A (enrdf_load_html_response)
PH (1) PH12831A (enrdf_load_html_response)
SE (1) SE437516B (enrdf_load_html_response)
SU (1) SU867304A3 (enrdf_load_html_response)
YU (1) YU40703B (enrdf_load_html_response)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6144294A (ja) * 1984-08-07 1986-03-03 Nippon Denso Co Ltd 熱交換器
US5053411A (en) * 1989-04-20 1991-10-01 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
USRE34201E (en) * 1989-04-20 1993-03-23 Anaquest, Inc. N-aryl-N-[4-(1-heterocyclicalkyl)piperidinyl]amides and pharmaceutical compositions and methods employing such compounds
JPH08193074A (ja) * 1994-11-18 1996-07-30 Nippon Bayeragrochem Kk 除草性１−シクロプロピルテトラゾリノン類
RU2144533C1 (ru) * 1994-12-09 2000-01-20 Такеда Кемикал Индастриз, Лтд. Производные тетразола, способ их получения и фармацевтические композиции на их основе
JP2000327668A (ja) * 1999-05-21 2000-11-28 Nippon Bayer Agrochem Co Ltd テトラゾリノン誘導体
CA2393559C (en) * 1999-12-06 2009-05-26 Mallinckrodt Inc. Methods for the syntheses of alfentanil, sufentanil and remifentanil
US20090030041A1 (en) * 2004-09-14 2009-01-29 Toshihiro Takahashi N-substituted N-(4-piperidinyl) Amide Derivative

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3998834A (en) * 1975-03-14 1976-12-21 Janssen Pharmaceutica N.V. N-(4-piperidinyl)-n-phenylamides and -carbamates

Also Published As

Publication number Publication date
IT1105288B (it) 1985-10-28
IE780901L (en) 1978-11-05
CA1105464A (en) 1981-07-21
DE2819873C2 (enrdf_load_html_response) 1989-05-03
FR2389622B1 (enrdf_load_html_response) 1982-05-21
FI64364C (fi) 1983-11-10
DK152211B (da) 1988-02-08
LU79575A1 (fr) 1978-11-03
YU108578A (en) 1983-01-21
YU40703B (en) 1986-04-30
NO148747C (no) 1983-12-07
NZ187164A (en) 1981-03-16
SU867304A3 (ru) 1981-09-23
CH635585A5 (en) 1983-04-15
FI64364B (fi) 1983-07-29
IL54639A0 (en) 1978-07-31
AT368994B (de) 1982-11-25
ES469473A1 (es) 1979-09-16
NO781559L (no) 1978-11-07
HK72585A (en) 1985-10-04
AU514360B2 (en) 1981-02-05
DK152211C (da) 1988-08-08
IL54639A (en) 1982-02-28
JPS53149980A (en) 1978-12-27
HU179204B (en) 1982-09-28
IE46836B1 (en) 1983-10-05
PH12831A (en) 1979-09-05
NL7804844A (nl) 1978-11-07
FR2389622A1 (enrdf_load_html_response) 1978-12-01
AU3552278A (en) 1979-11-01
DK193778A (da) 1978-11-06
NL186861B (nl) 1990-10-16
CY1253A (en) 1984-08-31
DE2819873A1 (de) 1978-11-09
GB1598872A (en) 1981-09-23
JPS6324995B2 (enrdf_load_html_response) 1988-05-23
FI781398A7 (fi) 1978-11-06
IT7849203A0 (it) 1978-05-04
NO148747B (no) 1983-08-29
NL186861C (nl) 1991-03-18
ATA322078A (de) 1982-04-15
KE3429A (en) 1984-08-10
SE7805110L (sv) 1978-11-06

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