SE436359B - Analogiforfarande for framstellning av 4-substituerade imidazo/1,2-a/kinoxaliner - Google Patents
Analogiforfarande for framstellning av 4-substituerade imidazo/1,2-a/kinoxalinerInfo
- Publication number
- SE436359B SE436359B SE7800138A SE7800138A SE436359B SE 436359 B SE436359 B SE 436359B SE 7800138 A SE7800138 A SE 7800138A SE 7800138 A SE7800138 A SE 7800138A SE 436359 B SE436359 B SE 436359B
- Authority
- SE
- Sweden
- Prior art keywords
- carbon atoms
- water
- formamide
- quinoxaline
- imidazo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Transplantation (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US75764077A | 1977-01-07 | 1977-01-07 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SE7800138L SE7800138L (sv) | 1978-07-08 |
| SE436359B true SE436359B (sv) | 1984-12-03 |
Family
ID=25048641
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7800138A SE436359B (sv) | 1977-01-07 | 1978-01-05 | Analogiforfarande for framstellning av 4-substituerade imidazo/1,2-a/kinoxaliner |
| SE8300945A SE460477B (sv) | 1977-01-07 | 1983-02-21 | 1-(2-acylaminofenyl)imidazoler till anvaendning sommellanprodukter |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE8300945A SE460477B (sv) | 1977-01-07 | 1983-02-21 | 1-(2-acylaminofenyl)imidazoler till anvaendning sommellanprodukter |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US4160097A (de) |
| JP (2) | JPS5387398A (de) |
| AU (1) | AU521807B2 (de) |
| BE (1) | BE862608A (de) |
| CA (1) | CA1149385A (de) |
| CH (2) | CH636102A5 (de) |
| CS (1) | CS200232B2 (de) |
| DE (2) | DE2858766C2 (de) |
| DK (1) | DK157024C (de) |
| FI (1) | FI64374C (de) |
| FR (1) | FR2376858A1 (de) |
| GB (2) | GB1579499A (de) |
| GR (1) | GR73168B (de) |
| IE (1) | IE46191B1 (de) |
| LU (1) | LU78813A1 (de) |
| NL (1) | NL7800114A (de) |
| SE (2) | SE436359B (de) |
| YU (1) | YU44663B (de) |
| ZA (1) | ZA7827B (de) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE439308B (sv) * | 1978-08-02 | 1985-06-10 | Roussel Uclaf | Imidazo(1,2-a)kinoxaliner och farmaceutiska kompositioner derav |
| JPS5569567A (en) * | 1978-11-21 | 1980-05-26 | Eisai Co Ltd | Novel imidazole compound, and antidepressant containing the same |
| IT1209431B (it) * | 1980-11-28 | 1989-07-16 | Angeli Inst Spa | Imidazolilfenil amidine, processi per la loro preparazione e loro impiego farmaceutico, ed intermedi di preparazione. |
| DE3830054A1 (de) * | 1988-09-03 | 1990-03-15 | Boehringer Mannheim Gmbh | Phenylamide - verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel |
| JPH0349309U (de) * | 1989-09-21 | 1991-05-14 | ||
| US6235740B1 (en) | 1997-08-25 | 2001-05-22 | Bristol-Myers Squibb Co. | Imidazoquinoxaline protein tyrosine kinase inhibitors |
| US6635626B1 (en) | 1997-08-25 | 2003-10-21 | Bristol-Myers Squibb Co. | Imidazoquinoxaline protein tyrosine kinase inhibitors |
| CN1285834A (zh) | 1997-11-11 | 2001-02-28 | 小野药品工业株式会社 | 稠合吡嗪化合物 |
| DE69940808D1 (de) * | 1998-03-04 | 2009-06-10 | Bristol Myers Squibb Co | Heterocyclen substituierte imidazopyrazine als protein- tyrosin-kinase-inhibitoren |
| US6869956B2 (en) * | 2000-10-03 | 2005-03-22 | Bristol-Myers Squibb Company | Methods of treating inflammatory and immune diseases using inhibitors of IκB kinase (IKK) |
| DE60117835T2 (de) | 2000-10-03 | 2006-10-19 | Bristol-Myers Squibb Co. | Amino- substituierte tetracyclische Verbindungen,die als entzündungshemmende Mittel nützlich sind, und diese enthaltende Arzneimittel |
| CA2436770A1 (en) * | 2001-02-01 | 2002-08-08 | James R. Burke | Methods of treating inflammatory and immune diseases using inhibitors of ikb kinase (ikk) |
| EP2066642A1 (de) * | 2006-09-25 | 2009-06-10 | Arete Therapeutics, INC. | Lösliche epoxidhydrolaseinhibitoren |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3541109A (en) * | 1968-06-25 | 1970-11-17 | Du Pont | 1-substituted imidazoles useful in acth reserve assay |
| US4011236A (en) * | 1968-09-09 | 1977-03-08 | Merck & Co., Inc. | N-(benzimidazol-2-yl)arylcarboxamides as ultraviolet (uv) light absorbers |
| GB1347493A (en) * | 1971-02-11 | 1974-02-27 | Aspro Nicholas Ltd | Benzazine derivatives |
| US3994893A (en) * | 1975-11-03 | 1976-11-30 | E. R. Squibb & Sons, Inc. | 4-Amino derivatives of pyrozolo[1,5-a]quinoxaline-3-carboxylic acid and esters |
-
1977
- 1977-12-08 US US05/858,515 patent/US4160097A/en not_active Expired - Lifetime
- 1977-12-23 GR GR55051A patent/GR73168B/el unknown
- 1977-12-28 CA CA000293972A patent/CA1149385A/en not_active Expired
- 1977-12-28 JP JP15758177A patent/JPS5387398A/ja active Granted
-
1978
- 1978-01-03 BE BE184085A patent/BE862608A/xx not_active IP Right Cessation
- 1978-01-04 DK DK004278A patent/DK157024C/da not_active IP Right Cessation
- 1978-01-04 FI FI780023A patent/FI64374C/fi not_active IP Right Cessation
- 1978-01-04 NL NL7800114A patent/NL7800114A/xx not_active Application Discontinuation
- 1978-01-04 ZA ZA00780027A patent/ZA7827B/xx unknown
- 1978-01-05 SE SE7800138A patent/SE436359B/sv not_active IP Right Cessation
- 1978-01-05 DE DE2858766A patent/DE2858766C2/de not_active Expired - Fee Related
- 1978-01-05 DE DE19782800480 patent/DE2800480A1/de active Granted
- 1978-01-05 LU LU78813A patent/LU78813A1/xx unknown
- 1978-01-06 FR FR7800308A patent/FR2376858A1/fr active Granted
- 1978-01-06 IE IE37/78A patent/IE46191B1/en unknown
- 1978-01-06 GB GB13335/79A patent/GB1579499A/en not_active Expired
- 1978-01-06 CH CH15278A patent/CH636102A5/fr not_active IP Right Cessation
- 1978-01-06 GB GB492/78A patent/GB1579498A/en not_active Expired
- 1978-01-06 YU YU21/78A patent/YU44663B/xx unknown
- 1978-01-09 CS CS78169A patent/CS200232B2/cs unknown
- 1978-01-11 AU AU32331/78A patent/AU521807B2/en not_active Expired
-
1983
- 1983-01-18 CH CH27483A patent/CH640229A5/fr not_active IP Right Cessation
- 1983-02-21 SE SE8300945A patent/SE460477B/sv not_active IP Right Cessation
-
1986
- 1986-01-17 JP JP61006590A patent/JPS61171470A/ja active Granted
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| NUG | Patent has lapsed |
Ref document number: 7800138-5 Effective date: 19920806 Format of ref document f/p: F |