SE0101327D0 - New crystalline forms - Google Patents

New crystalline forms

Info

Publication number
SE0101327D0
SE0101327D0 SE0101327A SE0101327A SE0101327D0 SE 0101327 D0 SE0101327 D0 SE 0101327D0 SE 0101327 A SE0101327 A SE 0101327A SE 0101327 A SE0101327 A SE 0101327A SE 0101327 D0 SE0101327 D0 SE 0101327D0
Authority
SE
Sweden
Prior art keywords
oxa
crystalline forms
ylüethylcarbamate
tert
butyl
Prior art date
Application number
SE0101327A
Other languages
English (en)
Swedish (sv)
Inventor
Neil Barnwell
Annika Bjoere
Lal Lashkar Singh Cheema
David Cladingboel
Karin Loevqvist
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Priority to SE0101327A priority Critical patent/SE0101327D0/xx
Publication of SE0101327D0 publication Critical patent/SE0101327D0/xx
Priority to TW091106493A priority patent/TWI237025B/zh
Priority to ARP020101189A priority patent/AR035452A1/es
Priority to CA002443470A priority patent/CA2443470A1/en
Priority to MXPA03009206A priority patent/MXPA03009206A/es
Priority to RU2003129231/04A priority patent/RU2286993C2/ru
Priority to PCT/SE2002/000725 priority patent/WO2002083688A1/en
Priority to PT02761972T priority patent/PT1389213E/pt
Priority to ES02761972T priority patent/ES2261721T3/es
Priority to EEP200300504A priority patent/EE200300504A/et
Priority to HU0303487A priority patent/HUP0303487A3/hu
Priority to NZ528560A priority patent/NZ528560A/en
Priority to PL02367179A priority patent/PL367179A1/xx
Priority to US10/474,592 priority patent/US7217708B2/en
Priority to DK02761972T priority patent/DK1389213T3/da
Priority to EP02761972A priority patent/EP1389213B1/en
Priority to SI200230325T priority patent/SI1389213T1/sl
Priority to KR10-2003-7013320A priority patent/KR20030087078A/ko
Priority to EP05007851A priority patent/EP1550663A1/en
Priority to AT02761972T priority patent/ATE323095T1/de
Priority to JP2002581443A priority patent/JP2004525970A/ja
Priority to CNB028116283A priority patent/CN1269823C/zh
Priority to BR0208829-0A priority patent/BR0208829A/pt
Priority to DE60210598T priority patent/DE60210598T2/de
Priority to CZ20032760A priority patent/CZ20032760A3/cs
Priority to IL15825002A priority patent/IL158250A0/xx
Priority to SK1257-2003A priority patent/SK12572003A3/sk
Priority to UA2003098709A priority patent/UA74629C2/uk
Priority to ZA200307759A priority patent/ZA200307759B/en
Priority to IS6980A priority patent/IS6980A/is
Priority to NO20034527A priority patent/NO20034527L/no
Priority to HK04104077A priority patent/HK1061026A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SE0101327A 2001-04-12 2001-04-12 New crystalline forms SE0101327D0 (sv)

Priority Applications (32)

Application Number Priority Date Filing Date Title
SE0101327A SE0101327D0 (sv) 2001-04-12 2001-04-12 New crystalline forms
TW091106493A TWI237025B (en) 2001-04-12 2002-04-01 New crystalline forms of antiarrhythmic compounds
ARP020101189A AR035452A1 (es) 2001-04-12 2002-04-02 Sales farmaceuticamente aceptables de compuestos antiarritmicos, procedimiento para la preparación de estas sales, formulación farmaceutica y el uso de estos compuestos para la manufactura de medicamentos para el uso en la profilaxis o el tratamiento de una arritmia
SK1257-2003A SK12572003A3 (sk) 2001-04-12 2002-04-12 Farmaceutická kompozícia obsahujúca 3,7-diazabicyklo [3.3.1]-deriváty ako účinnú zložku a jej použitie
DK02761972T DK1389213T3 (da) 2001-04-12 2002-04-12 3,7-Diazabicyclo[3.3.1]formuleringer som antiarytmiske forbindelser
EP05007851A EP1550663A1 (en) 2001-04-12 2002-04-12 New crystalline forms of antiarrhythmic compounds
RU2003129231/04A RU2286993C2 (ru) 2001-04-12 2002-04-12 3,7-диазабицикло[3.3.1]-препараты как антиаритмические соединения
PCT/SE2002/000725 WO2002083688A1 (en) 2001-04-12 2002-04-12 3,7-diazabicyclo [3.3.1] formulations as antiarhythmic compounds
PT02761972T PT1389213E (pt) 2001-04-12 2002-04-12 Formulacoes de 3,7-diazabiciclo 3,3,1¿ como compostos antiarritmicos
ES02761972T ES2261721T3 (es) 2001-04-12 2002-04-12 Formulaciones de 3,7-diazabiciclo(3.3.1) como compuestos antiarritmicos.
EEP200300504A EE200300504A (et) 2001-04-12 2002-04-12 3,7-diasabitsüklo[3.3.1]preparaadid, nende valmistamise meetod ja nimetatud preparaatide kasutaminesüdame arütmiate profülaktikas või ravis
HU0303487A HUP0303487A3 (en) 2001-04-12 2002-04-12 Compositions containing 3,7-diazabicyclo [3,3,1] compounds as anthiarhythmic agents and process for preparation of the compounds
NZ528560A NZ528560A (en) 2001-04-12 2002-04-12 3,7-diazabicyclo [3.3.1] formulations as antiarrhythmic compounds
PL02367179A PL367179A1 (en) 2001-04-12 2002-04-12 3,7-diazabicyclo [3.3.1] formulations as antiarhythmic compounds
US10/474,592 US7217708B2 (en) 2001-04-12 2002-04-12 3,7-Diazabicyclo [3.3.1] formulations as anti-arrhythmic compounds
CA002443470A CA2443470A1 (en) 2001-04-12 2002-04-12 3,7-diazabicyclo [3.3.1] formulations as antiarhythmic compounds
EP02761972A EP1389213B1 (en) 2001-04-12 2002-04-12 3,7-diazabicyclo 3.3.1| formulations as antiarhythmic compounds
SI200230325T SI1389213T1 (sl) 2001-04-12 2002-04-12 3,7-diazabiciklo(3.3.1)formulacije kot antiaritmicne spojine
KR10-2003-7013320A KR20030087078A (ko) 2001-04-12 2002-04-12 항부정맥 화합물로서의 3,7-디아자비시클로[3.3.1] 조성물
MXPA03009206A MXPA03009206A (es) 2001-04-12 2002-04-12 FORMULACIONES DE 3,7-DIAZABICICLO [3.3.1] COMO COMPUESTOS ANTIARRiTMICOS.
AT02761972T ATE323095T1 (de) 2001-04-12 2002-04-12 3,7-diazabicycloc3.3.1)-formulierungen als antiarrhythmika
JP2002581443A JP2004525970A (ja) 2001-04-12 2002-04-12 抗不整脈化合物としての3,7−ジアザビシクロ[3.3.1]製剤
CNB028116283A CN1269823C (zh) 2001-04-12 2002-04-12 作为抗心律不齐化合物的3,7-二氮杂双环[3.3.1]制剂
BR0208829-0A BR0208829A (pt) 2001-04-12 2002-04-12 Sal farmaceuticamente aceitável, composto, processos para a preparação de um sal, de um composto e de uma forma cristalina dos compostos, formulação farmacêutica, uso de um composto, e, método de profilaxia ou tratamento de uma arritmia
DE60210598T DE60210598T2 (de) 2001-04-12 2002-04-12 3,7-DIAZABICYCLOc3.3.1Ü-FORMULIERUNGEN ALS ANTIARRHYTHMIKA
CZ20032760A CZ20032760A3 (cs) 2001-04-12 2002-04-12 Farmaceutická kompozice obsahující 3,7-diazabicyklo[3.3.1]-deriváty jako účinnou složku a její použití
IL15825002A IL158250A0 (en) 2001-04-12 2002-04-12 3,7-diazabicyclo [3.3.1] formulations as antiarrhythmic compounds
UA2003098709A UA74629C2 (en) 2001-04-12 2002-12-04 A derivative of 3,7-diazabicyclo [3,3,1] compounds , pharmaceutically acceptable salts thereof, a method for producing and composition based thereon as antiarrhythmic agents
ZA200307759A ZA200307759B (en) 2001-04-12 2003-10-03 3,7-diazabicyclo[3.3.1]formulations as antiarrhythmic compounds.
IS6980A IS6980A (is) 2001-04-12 2003-10-08 3,7-díasabísýkló [3.3.1] blöndur sem efnasambönd gegn sláttarglöpum
NO20034527A NO20034527L (no) 2001-04-12 2003-10-09 3,7-diazabicyklo(3,3,1) formuleringer som antiarytmiforbindelser
HK04104077A HK1061026A1 (en) 2001-04-12 2004-06-08 3,7-Diazabicyclo 3.3.1Ü formulations as antiarhythmic compounds

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0101327A SE0101327D0 (sv) 2001-04-12 2001-04-12 New crystalline forms

Publications (1)

Publication Number Publication Date
SE0101327D0 true SE0101327D0 (sv) 2001-04-12

Family

ID=20283783

Family Applications (1)

Application Number Title Priority Date Filing Date
SE0101327A SE0101327D0 (sv) 2001-04-12 2001-04-12 New crystalline forms

Country Status (30)

Country Link
US (1) US7217708B2 (et)
EP (2) EP1550663A1 (et)
JP (1) JP2004525970A (et)
KR (1) KR20030087078A (et)
CN (1) CN1269823C (et)
AR (1) AR035452A1 (et)
AT (1) ATE323095T1 (et)
BR (1) BR0208829A (et)
CA (1) CA2443470A1 (et)
CZ (1) CZ20032760A3 (et)
DE (1) DE60210598T2 (et)
DK (1) DK1389213T3 (et)
EE (1) EE200300504A (et)
ES (1) ES2261721T3 (et)
HK (1) HK1061026A1 (et)
HU (1) HUP0303487A3 (et)
IL (1) IL158250A0 (et)
IS (1) IS6980A (et)
MX (1) MXPA03009206A (et)
NO (1) NO20034527L (et)
NZ (1) NZ528560A (et)
PL (1) PL367179A1 (et)
PT (1) PT1389213E (et)
RU (1) RU2286993C2 (et)
SE (1) SE0101327D0 (et)
SK (1) SK12572003A3 (et)
TW (1) TWI237025B (et)
UA (1) UA74629C2 (et)
WO (1) WO2002083688A1 (et)
ZA (1) ZA200307759B (et)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI259836B (en) * 2001-04-12 2006-08-11 Astrazeneca Ab Modified release formulation suitable for antiarrhythmic compounds
SE0401539D0 (sv) * 2004-06-15 2004-06-15 Astrazeneca Ab New compounds
SE0401540D0 (sv) * 2004-06-15 2004-06-15 Astrazeneca Ab New compounds
AR057064A1 (es) * 2005-06-13 2007-11-14 Astrazeneca Ab Compuestos para el tratamiento de arritmias cardiacas, formulacion farmaceutica y preparacion del compuesto
MX2007016496A (es) * 2005-06-20 2008-03-06 Astrazeneca Ab Proceso para la preparacion de oxabispidinas n-n' -disustituidas.
AR053901A1 (es) * 2005-06-20 2007-05-23 Astrazeneca Ab Formas fisicas de oxabispidinas n,n'- disustituidas
TW200734342A (en) * 2005-12-15 2007-09-16 Astrazeneca Ab New compounds for the treatment of cardiac arrhythmias
CA2644613A1 (en) * 2006-03-07 2007-09-13 Endacea, Inc. Compositions and methods for treating respiratory disorders
JP5113838B2 (ja) 2006-06-26 2013-01-09 アケビア セラピューティックス, インコーポレイテッド プロリルヒドロキシラーゼ阻害剤および使用方法
MX2013014310A (es) 2011-06-06 2014-01-23 Akebia Therapeutics Inc Compuestos y composiciones para estabilizar el factor-2 alfa inducible por hipoxia como un metodo para tratar el cancer.
NO2686520T3 (et) 2011-06-06 2018-03-17
SG11201509998WA (en) 2013-06-13 2016-01-28 Akebia Therapeutics Inc Compositions and methods for treating anemia
TW201946625A (zh) 2013-11-15 2019-12-16 美商阿克比治療有限公司 {[5-(3-氯苯基)-3-羥基吡啶-2-羰基]胺基}乙酸之固體型式,其組合物及用途
WO2016118858A1 (en) 2015-01-23 2016-07-28 Akebia Therapeutics, Inc. Solid forms of 2-(5-(3-fluorophenyl)-3-hydroxypicolinamido)acetic acid, compositions, and uses thereof
DK3277270T3 (da) 2015-04-01 2021-12-06 Akebia Therapeutics Inc Sammensætninger og fremgangsmåder til behandling af anæmi
CN112088155A (zh) 2018-05-09 2020-12-15 阿克比治疗有限公司 用于制备2-[[5-(3-氯苯基)-3-羟基吡啶-2-羰基]氨基]乙酸的方法
US11524939B2 (en) 2019-11-13 2022-12-13 Akebia Therapeutics, Inc. Solid forms of {[5-(3-chlorophenyl)-3-hydroxypyridine-2-carbonyl]amino} acetic acid

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3732094A1 (de) * 1987-09-24 1989-04-06 Basf Ag Bispidinderivate als klasse iii-antiarrhythmika
US5110933A (en) * 1989-11-13 1992-05-05 Board Of Regents Of Oklahoma State University Salts of 3-azabicyclo[3.3.1]nonanes as antiarrhythmic agents, and precursors thereof
SE9704709D0 (sv) * 1997-12-17 1997-12-17 Astra Ab Pharmaceutically active compounds
SE9902268D0 (sv) 1999-06-16 1999-06-16 Astra Ab Pharmaceutically active compounds
SE9903759D0 (sv) * 1999-10-18 1999-10-18 Astra Ab Pharmaceutically active compounds

Also Published As

Publication number Publication date
NZ528560A (en) 2005-05-27
CA2443470A1 (en) 2002-10-24
TWI237025B (en) 2005-08-01
ZA200307759B (en) 2005-01-03
MXPA03009206A (es) 2004-01-29
RU2286993C2 (ru) 2006-11-10
EP1389213A1 (en) 2004-02-18
PT1389213E (pt) 2006-07-31
AR035452A1 (es) 2004-05-26
RU2003129231A (ru) 2005-04-10
KR20030087078A (ko) 2003-11-12
DE60210598D1 (de) 2006-05-24
DK1389213T3 (da) 2006-07-10
SK12572003A3 (sk) 2004-07-07
WO2002083688A1 (en) 2002-10-24
BR0208829A (pt) 2004-03-09
CZ20032760A3 (cs) 2004-01-14
DE60210598T2 (de) 2007-02-08
HUP0303487A2 (hu) 2004-01-28
HK1061026A1 (en) 2004-09-03
IL158250A0 (en) 2004-05-12
CN1514837A (zh) 2004-07-21
US7217708B2 (en) 2007-05-15
EP1389213B1 (en) 2006-04-12
NO20034527L (no) 2003-12-10
EP1550663A1 (en) 2005-07-06
EE200300504A (et) 2003-12-15
JP2004525970A (ja) 2004-08-26
HUP0303487A3 (en) 2005-04-28
UA74629C2 (en) 2006-01-16
IS6980A (is) 2003-10-08
NO20034527D0 (no) 2003-10-09
US20040143000A1 (en) 2004-07-22
ATE323095T1 (de) 2006-04-15
ES2261721T3 (es) 2006-11-16
PL367179A1 (en) 2005-02-21
CN1269823C (zh) 2006-08-16

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