RU94027570A - Способ получения замещенных пиперидинов, способ получения промежуточных продуктов, промежуточные продукты - Google Patents
Способ получения замещенных пиперидинов, способ получения промежуточных продуктов, промежуточные продуктыInfo
- Publication number
- RU94027570A RU94027570A RU94027570/04A RU94027570A RU94027570A RU 94027570 A RU94027570 A RU 94027570A RU 94027570/04 A RU94027570/04 A RU 94027570/04A RU 94027570 A RU94027570 A RU 94027570A RU 94027570 A RU94027570 A RU 94027570A
- Authority
- RU
- Russia
- Prior art keywords
- intermediate products
- obtaining
- substituted piperidines
- piperidines
- products
- Prior art date
Links
- 150000003053 piperidines Chemical class 0.000 title claims 2
- 150000001875 compounds Chemical class 0.000 claims 1
- 239000000543 intermediate Substances 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
Claims (1)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US800667 | 1991-11-27 | ||
US07/800,667 US5364943A (en) | 1991-11-27 | 1991-11-27 | Preparation of substituted piperidines |
PCT/US1992/009929 WO1993011110A1 (en) | 1991-11-27 | 1992-11-24 | Preparation of substituted piperidines |
Publications (2)
Publication Number | Publication Date |
---|---|
RU94027570A true RU94027570A (ru) | 1996-01-10 |
RU2081112C1 RU2081112C1 (ru) | 1997-06-10 |
Family
ID=25179032
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RU9294027570A RU2081112C1 (ru) | 1991-11-27 | 1992-11-24 | Производные пиридина и способы их получения |
Country Status (19)
Country | Link |
---|---|
US (2) | US5364943A (ru) |
EP (1) | EP0619806B1 (ru) |
JP (1) | JP2587903B2 (ru) |
KR (1) | KR0150254B1 (ru) |
AT (1) | ATE132487T1 (ru) |
AU (1) | AU670765B2 (ru) |
BR (1) | BR9206823A (ru) |
CA (1) | CA2124083C (ru) |
CZ (1) | CZ292947B6 (ru) |
DE (1) | DE69207429T2 (ru) |
DK (1) | DK0619806T3 (ru) |
ES (1) | ES2081636T3 (ru) |
FI (1) | FI107049B (ru) |
GR (1) | GR3018679T3 (ru) |
HU (1) | HUT70514A (ru) |
NO (1) | NO300970B1 (ru) |
PL (1) | PL173659B1 (ru) |
RU (1) | RU2081112C1 (ru) |
WO (1) | WO1993011110A1 (ru) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1994003445A1 (en) * | 1992-08-04 | 1994-02-17 | Pfizer Inc. | 3-benzylamino-2-phenyl-piperidine derivatives as substance p receptor antagonists |
EP0700384B1 (en) * | 1993-05-28 | 1997-07-16 | Pfizer Inc. | Process for preparing and resolving 2-phenyl-3-aminopiperidine |
GB9317987D0 (en) * | 1993-08-26 | 1993-10-13 | Glaxo Group Ltd | Chemical compounds |
TW340842B (en) * | 1995-08-24 | 1998-09-21 | Pfizer | Substituted benzylaminopiperidine compounds |
DE69623580T2 (de) | 1995-12-21 | 2003-01-09 | Pfizer | 3-((5-Substituierte Benzyl)Amino)-2-Phenylpiperidine als Substance-P-Antagonisten |
US6194599B1 (en) | 1997-04-08 | 2001-02-27 | Catalytica, Inc. | Process for preparing biaryl compounds |
US5922898A (en) * | 1997-04-08 | 1999-07-13 | Catalytica Pharmaceuticals, Inc. | Process for preparing biaryl compounds |
NZ329807A (en) * | 1997-04-23 | 2000-07-28 | Pfizer | NK-1 receptor antagonists and P receptor antagonists 2-Diarylmethyl-3-amino-1-azabicyclo[2.2.2]octane derivatives and amino substituted N-containing rings as agents for treating irritable bowel syndrome |
US6214846B1 (en) | 1997-06-27 | 2001-04-10 | Merck Sharp & Dohme Limited | Substituted 3-(benzylamino)piperidine derivatives and their use as therapeutic agents |
DE19824470A1 (de) * | 1998-05-30 | 1999-12-02 | Boehringer Ingelheim Pharma | Neue Neurokininantagonisten, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen |
EP1035115B1 (en) | 1999-02-24 | 2004-09-29 | F. Hoffmann-La Roche Ag | 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists |
RS49964B (sr) * | 1999-05-17 | 2008-09-29 | Pfizer Products Inc., | Postupak za dobijanje 2-fenil-3-aminopiridina,njegovih supstituisanih fenil derivata, i njegovih soli |
US6962999B2 (en) * | 2001-07-25 | 2005-11-08 | Pharmacore, Inc. | Process for preparing unsymmetrical biaryls and alkylated aromatic compounds from arylnitriles |
US6911544B2 (en) * | 2002-10-23 | 2005-06-28 | Pfizer Inc. | Process for the preparation of (S,S)-cis-2-phenyl-3-aminopiperidine |
US7105467B2 (en) * | 2003-07-08 | 2006-09-12 | Pharmacore, Inc. | Nickel catalyzed cross-coupling reactions between organomagnesium compounds and anisole derivatives |
TWI280239B (en) | 2003-07-15 | 2007-05-01 | Hoffmann La Roche | Process for preparation of pyridine derivatives |
US7105707B2 (en) * | 2003-12-17 | 2006-09-12 | Pharmacore, Inc. | Process for preparing alkynyl-substituted aromatic and heterocyclic compounds |
CN101267808A (zh) | 2005-09-23 | 2008-09-17 | 弗·哈夫曼-拉罗切有限公司 | 新型制剂 |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3560510A (en) * | 1969-03-05 | 1971-02-02 | Aldrich Chem Co Inc | 2-benzhydrylquinuclidines |
CA1160229A (en) * | 1979-03-13 | 1984-01-10 | Pieter T. Haken | Pyridyliminomethylbenzene derivatives |
GB2056974B (en) * | 1979-07-19 | 1984-02-29 | Shell Int Research | Heterocyclic acylamino compounds having fungicidal herbicidal and plant-growth regulating properties |
CA1231710A (en) * | 1979-07-19 | 1988-01-19 | Haken Pieter Ten | Heterocyclic compounds having fungicidal, herbicidal and plant-growth regulating properties |
GB2067187B (en) * | 1979-12-07 | 1983-11-30 | Cosmos Enterprise | Process for the preparation of 1-(4-hydroxyphenyl)-2-(4-benzylpiperidino)-1-propanol and acid addition salts thereof |
EP0100158A3 (en) * | 1982-07-28 | 1985-03-27 | The Upjohn Company | (3-pyridinyl)heteroalkarylalkanols, alkanoic acids and esters |
US4552960A (en) * | 1983-06-20 | 1985-11-12 | Eli Lilly And Company | Fungicidal amines |
US4680283A (en) * | 1984-09-26 | 1987-07-14 | Merck & Co., Inc. | Analogs of substance P and eledoisin |
MX18467A (es) * | 1988-11-23 | 1993-07-01 | Pfizer | Agentes terapeuticos de quinuclidinas |
UA41251C2 (ru) * | 1990-01-04 | 2001-09-17 | Пфайзер, Інк. | Гидрированные азотсодержащие гетероциклические соединения, производные пиперидина, фармацевтическая композиция и способ угнетения активности вещества р в организме |
HU226529B1 (en) * | 1990-05-31 | 2009-03-30 | Pfizer | Process for preparing substituted piperidines |
US5138060A (en) * | 1991-01-03 | 1992-08-11 | Pfizer Inc. | Process and intermediates for preparing azabicyclo(2.2.2)octan-3-imines |
HUT65612A (en) * | 1991-01-10 | 1994-07-28 | Pfizer | Process n-alcyl-quinuclidinium salts of p-antagonistic activity |
CZ293955B6 (cs) * | 1991-03-26 | 2004-08-18 | Pfizeráinc | Postup přípravy substituovaných piperidinů |
DE69213451T2 (de) * | 1991-06-20 | 1997-01-09 | Pfizer | Fluoralkoxybenzylaminoderivate stickstoffhaltiger heterocyclen |
TW202432B (ru) * | 1991-06-21 | 1993-03-21 | Pfizer |
-
1991
- 1991-11-27 US US07/800,667 patent/US5364943A/en not_active Expired - Lifetime
-
1992
- 1992-11-24 CZ CZ19941300A patent/CZ292947B6/cs not_active IP Right Cessation
- 1992-11-24 BR BR9206823A patent/BR9206823A/pt not_active Application Discontinuation
- 1992-11-24 WO PCT/US1992/009929 patent/WO1993011110A1/en not_active Application Discontinuation
- 1992-11-24 RU RU9294027570A patent/RU2081112C1/ru not_active IP Right Cessation
- 1992-11-24 PL PL92303982A patent/PL173659B1/pl not_active IP Right Cessation
- 1992-11-24 ES ES92925298T patent/ES2081636T3/es not_active Expired - Lifetime
- 1992-11-24 AU AU31408/93A patent/AU670765B2/en not_active Ceased
- 1992-11-24 DK DK92925298.9T patent/DK0619806T3/da active
- 1992-11-24 DE DE69207429T patent/DE69207429T2/de not_active Expired - Fee Related
- 1992-11-24 AT AT92925298T patent/ATE132487T1/de not_active IP Right Cessation
- 1992-11-24 EP EP92925298A patent/EP0619806B1/en not_active Expired - Lifetime
- 1992-11-24 KR KR1019940701782A patent/KR0150254B1/ko not_active IP Right Cessation
- 1992-11-24 HU HU9401584A patent/HUT70514A/hu unknown
- 1992-11-24 CA CA002124083A patent/CA2124083C/en not_active Expired - Fee Related
- 1992-11-24 JP JP5510148A patent/JP2587903B2/ja not_active Expired - Fee Related
-
1994
- 1994-05-26 FI FI942457A patent/FI107049B/fi not_active IP Right Cessation
- 1994-05-26 NO NO941958A patent/NO300970B1/no unknown
- 1994-07-12 US US08/273,662 patent/US5663349A/en not_active Expired - Fee Related
-
1996
- 1996-01-17 GR GR960400080T patent/GR3018679T3/el unknown
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