RU2520735C2 - Гидроксилированный пиримидил циклопентан в качестве ингибитора протеинкиназы (акт) - Google Patents
Гидроксилированный пиримидил циклопентан в качестве ингибитора протеинкиназы (акт) Download PDFInfo
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- RU2520735C2 RU2520735C2 RU2010132912/04A RU2010132912A RU2520735C2 RU 2520735 C2 RU2520735 C2 RU 2520735C2 RU 2010132912/04 A RU2010132912/04 A RU 2010132912/04A RU 2010132912 A RU2010132912 A RU 2010132912A RU 2520735 C2 RU2520735 C2 RU 2520735C2
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| PCT/US2009/030602 WO2009089453A1 (en) | 2008-01-09 | 2009-01-09 | Hydroxylated pyrimidyl cyclopentane as akt protein kinase inhibitor |
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Families Citing this family (9)
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| US9409886B2 (en) | 2007-07-05 | 2016-08-09 | Array Biopharma Inc. | Pyrimidyl cyclopentanes as AKT protein kinase inhibitors |
| SG185274A1 (en) * | 2007-07-05 | 2012-11-29 | Array Biopharma Inc | Pyrimidyl cyclopentanes as akt protein kinase inhibitors |
| US8846683B2 (en) | 2007-07-05 | 2014-09-30 | Array Biopharma, Inc. | Pyrimidyl cyclopentanes as Akt protein kinase inhibitors |
| EP2242755B1 (en) | 2008-01-08 | 2012-09-12 | Array Biopharma, Inc. | Pyrrolopyridines as kinase inhibitors |
| WO2009089462A1 (en) | 2008-01-09 | 2009-07-16 | Array Biopharma Inc. | 5h-cyclopenta[d]pyrimidines as akt protein kinase inhibitors |
| ES2392014T3 (es) | 2008-01-09 | 2012-12-03 | Array Biopharma, Inc. | Pirazolopiridinas como inhibidores de la cinasa |
| BR112014028573B1 (pt) | 2012-05-17 | 2021-11-16 | Genentech, Inc | Processo de fabricação de compostos de ciclopentapirimidina hidroxilada |
| PL3068770T3 (pl) | 2013-11-15 | 2020-04-30 | F. Hoffmann-La Roche Ag | Sposoby przygotowania związków pirymidynylocyklopentanu |
| WO2017156350A1 (en) | 2016-03-09 | 2017-09-14 | K-Gen, Inc. | Methods of cancer treatment |
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| WO2008006040A1 (en) * | 2006-07-06 | 2008-01-10 | Array Biopharma Inc. | Hydroxylated and methoxylated cyclopenta [d] pyrimidines as akt protein kinase inhibitors |
| RU2010103811A (ru) * | 2007-07-05 | 2011-08-10 | Эррэй Биофарма Инк. (Us) | Пиримидилциклопентаны в качестве ингибиторов akt-протеинкиназы |
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2009
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- 2010-07-26 CO CO10090857A patent/CO6280510A2/es active IP Right Grant
- 2010-08-09 EC EC2010010392A patent/ECSP10010392A/es unknown
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| EP2240455A1 (en) | 2010-10-20 |
| CO6280510A2 (es) | 2011-05-20 |
| KR101624752B1 (ko) | 2016-05-26 |
| JP2011509306A (ja) | 2011-03-24 |
| CN101932565B (zh) | 2013-06-12 |
| AU2009204019A1 (en) | 2009-07-16 |
| HK1149269A1 (en) | 2011-09-30 |
| ECSP10010392A (es) | 2010-09-30 |
| BRPI0907372A2 (pt) | 2015-07-14 |
| KR20100103865A (ko) | 2010-09-28 |
| ES2401685T3 (es) | 2013-04-23 |
| WO2009089453A9 (en) | 2009-11-05 |
| EP2240455B1 (en) | 2012-12-26 |
| CR11591A (es) | 2010-11-30 |
| UA100544C2 (ru) | 2013-01-10 |
| MX2010007546A (es) | 2010-09-30 |
| IL206607A0 (en) | 2010-12-30 |
| JP5539225B2 (ja) | 2014-07-02 |
| AU2009204019B2 (en) | 2014-02-20 |
| US20100292244A1 (en) | 2010-11-18 |
| RU2010132912A (ru) | 2012-02-20 |
| MA32343B1 (fr) | 2011-06-01 |
| WO2009089453A1 (en) | 2009-07-16 |
| US8853216B2 (en) | 2014-10-07 |
| CN101932565A (zh) | 2010-12-29 |
| NZ586720A (en) | 2012-11-30 |
| ES2401685T8 (es) | 2014-11-06 |
| CA2711692A1 (en) | 2009-07-16 |
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