RU2472497C2 - Титрование тапентадола - Google Patents
Титрование тапентадола Download PDFInfo
- Publication number
- RU2472497C2 RU2472497C2 RU2009142940/15A RU2009142940A RU2472497C2 RU 2472497 C2 RU2472497 C2 RU 2472497C2 RU 2009142940/15 A RU2009142940/15 A RU 2009142940/15A RU 2009142940 A RU2009142940 A RU 2009142940A RU 2472497 C2 RU2472497 C2 RU 2472497C2
- Authority
- RU
- Russia
- Prior art keywords
- dose
- administration
- tapentadol
- period
- day
- Prior art date
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07008218.5 | 2007-04-23 | ||
| EP07008218A EP1985292A1 (en) | 2007-04-23 | 2007-04-23 | Titration of tapentadol |
| PCT/EP2008/003178 WO2008128740A1 (en) | 2007-04-23 | 2008-04-21 | Titration of tapentadol |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2009142940A RU2009142940A (ru) | 2011-05-27 |
| RU2472497C2 true RU2472497C2 (ru) | 2013-01-20 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2009142940/15A RU2472497C2 (ru) | 2007-04-23 | 2008-04-21 | Титрование тапентадола |
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|---|---|
| US (4) | US20090012180A1 (enExample) |
| EP (5) | EP1985292A1 (enExample) |
| JP (4) | JP5933176B2 (enExample) |
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| EP1985292A1 (en) * | 2007-04-23 | 2008-10-29 | Grünenthal GmbH | Titration of tapentadol |
| JP6216489B2 (ja) * | 2008-10-30 | 2017-10-18 | グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング | 新規の、効力のあるタペンタドール剤形 |
| US8870876B2 (en) * | 2009-02-13 | 2014-10-28 | Tarsus Medical Inc. | Methods and devices for treating hallux valgus |
| US8277459B2 (en) | 2009-09-25 | 2012-10-02 | Tarsus Medical Inc. | Methods and devices for treating a structural bone and joint deformity |
| US8652141B2 (en) | 2010-01-21 | 2014-02-18 | Tarsus Medical Inc. | Methods and devices for treating hallux valgus |
| US20130116333A1 (en) * | 2010-05-05 | 2013-05-09 | Ratiopharm Gmbh | Solid tapentadol in non-crystalline form |
| US8696719B2 (en) | 2010-06-03 | 2014-04-15 | Tarsus Medical Inc. | Methods and devices for treating hallux valgus |
| HRP20161166T1 (hr) * | 2010-06-30 | 2016-11-04 | Grünenthal GmbH | Tapentadol za uporabu u liječenju sindroma iritabilnog crijeva |
| EP3650439B1 (en) * | 2010-07-23 | 2021-02-24 | Grünenthal GmbH | Salts or co-crystals of 3-(3-dimethylamino-1-ethyl-2-methyl-propyl)-phenol |
| CN101948397A (zh) * | 2010-09-07 | 2011-01-19 | 天津泰普药品科技发展有限公司 | 镇痛药他喷他多重要中间体的制备方法 |
| RS54711B1 (sr) * | 2011-03-04 | 2016-08-31 | Grünenthal GmbH | Parenteralno davanje tapentadola |
| SI3287123T1 (sl) | 2011-03-04 | 2020-07-31 | Gruenenthal Gmbh | Vodna farmacevtska formulacija tapentadola za peroralno uporabo |
| KR101911362B1 (ko) | 2011-03-04 | 2018-10-25 | 그뤼넨탈 게엠베하 | 타펜타돌을 함유하는 반고체 수성 약제학적 조성물 |
| PL2694050T3 (pl) * | 2011-04-05 | 2020-03-31 | Grünenthal GmbH | Tapentadol do stosowania w leczeniu bólu związanego z nerwobólami nerwu trójdzielnego |
| US20120309841A1 (en) * | 2011-04-05 | 2012-12-06 | Gruenenthal Gmbh | Method of Inhibiting Chronification of Pain |
| RS60152B1 (sr) | 2011-04-29 | 2020-05-29 | Gruenenthal Gmbh | Tapentadol za sprečavanje i lečenje depresije i anksioznosti |
| WO2014152296A1 (en) * | 2013-03-15 | 2014-09-25 | Mallinckrodt Llc | Abuse deterrent solid dosage form for immediate release with functional score |
| EP2845625A1 (en) * | 2013-09-04 | 2015-03-11 | Grünenthal GmbH | Tapentadol for use in the treatment of fibromyalgia and chronic fatigue syndrome |
| PT3479823T (pt) | 2015-03-27 | 2020-09-29 | Gruenenthal Gmbh | Formulação estável para administração parentérica de tapentadol |
| JP6853791B2 (ja) * | 2015-05-26 | 2021-03-31 | テクノファージ， インベスティガサン エ デセンボルビメント エム ビオテクノロジア，エスエー | パーキンソン病及び関連する障害の治療における使用のための組成物 |
| WO2017148595A1 (en) * | 2016-02-29 | 2017-09-08 | Grünenthal GmbH | Titration of cebranopadol |
| EP3515412B1 (en) | 2016-09-23 | 2025-04-23 | Grünenthal GmbH | Stable formulation for parenteral administration of tapentadol |
| AU2021237693A1 (en) | 2020-03-16 | 2022-09-08 | Grünenthal GmbH | Scored tablet |
| WO2022194941A1 (en) * | 2021-03-17 | 2022-09-22 | Actelion Pharmaceuticals Ltd | Pharmaceutical dosage system |
| US20240238221A1 (en) * | 2021-05-07 | 2024-07-18 | Grünenthal GmbH | Tapentadol for treating neuropathic pain in covid-19 patients |
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| RU2150465C1 (ru) * | 1994-07-23 | 2000-06-10 | Грюненталь Гмбх | 1-фенил-3-диметиламино-пропановые соединения, способ их получения (варианты) и болеутоляющее лекарственное средство |
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| DE102007019417A1 (de) | 2007-04-23 | 2008-11-13 | Grünenthal GmbH | Tapentadol zur Schmerzbehandlung bei Arthrose |
| EP1985292A1 (en) * | 2007-04-23 | 2008-10-29 | Grünenthal GmbH | Titration of tapentadol |
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2007
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2008
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