RU2419608C2 - Новые соединения - Google Patents

Новые соединения Download PDF

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Publication number
RU2419608C2
RU2419608C2 RU2006141320/04A RU2006141320A RU2419608C2 RU 2419608 C2 RU2419608 C2 RU 2419608C2 RU 2006141320/04 A RU2006141320/04 A RU 2006141320/04A RU 2006141320 A RU2006141320 A RU 2006141320A RU 2419608 C2 RU2419608 C2 RU 2419608C2
Authority
RU
Russia
Prior art keywords
phenyl
acetamide
hydroxypropoxy
amino
piperidinyl
Prior art date
Application number
RU2006141320/04A
Other languages
English (en)
Russian (ru)
Other versions
RU2006141320A (ru
Inventor
Томас ЭРИКССОН (SE)
Томас Эрикссон
Томас КЛИНГСТЕДТ (SE)
Томас Клингстедт
Тесфаледет МУССИ (SE)
Тесфаледет МУССИ
Original Assignee
Астразенека Аб
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE0002331A external-priority patent/SE0002331D0/xx
Priority claimed from SE0004480A external-priority patent/SE0004480D0/xx
Application filed by Астразенека Аб filed Critical Астразенека Аб
Publication of RU2006141320A publication Critical patent/RU2006141320A/ru
Application granted granted Critical
Publication of RU2419608C2 publication Critical patent/RU2419608C2/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
RU2006141320/04A 2000-06-20 2001-06-14 Новые соединения RU2419608C2 (ru)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
SE0002331A SE0002331D0 (sv) 2000-06-20 2000-06-20 Novel compounds
SE0002331-7 2000-06-20
SE0004480-0 2000-12-05
SE0004480A SE0004480D0 (sv) 2000-12-05 2000-12-05 Novel compounds

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
RU2002132385/04A Division RU2298550C2 (ru) 2000-06-20 2001-06-14 Производные пиперидина, способы их получения и фармацевтическая композиция на их основе

Publications (2)

Publication Number Publication Date
RU2006141320A RU2006141320A (ru) 2008-06-10
RU2419608C2 true RU2419608C2 (ru) 2011-05-27

Family

ID=26655154

Family Applications (2)

Application Number Title Priority Date Filing Date
RU2002132385/04A RU2298550C2 (ru) 2000-06-20 2001-06-14 Производные пиперидина, способы их получения и фармацевтическая композиция на их основе
RU2006141320/04A RU2419608C2 (ru) 2000-06-20 2001-06-14 Новые соединения

Family Applications Before (1)

Application Number Title Priority Date Filing Date
RU2002132385/04A RU2298550C2 (ru) 2000-06-20 2001-06-14 Производные пиперидина, способы их получения и фармацевтическая композиция на их основе

Country Status (22)

Country Link
US (3) US6911458B2 (enExample)
EP (1) EP1299357A1 (enExample)
JP (1) JP4022142B2 (enExample)
KR (1) KR100799061B1 (enExample)
CN (1) CN1307157C (enExample)
AR (1) AR028948A1 (enExample)
AU (2) AU2001274763B2 (enExample)
BR (1) BR0111667A (enExample)
CA (1) CA2414095C (enExample)
CZ (1) CZ20024146A3 (enExample)
EE (1) EE05157B1 (enExample)
HU (1) HUP0301187A3 (enExample)
IL (2) IL153167A0 (enExample)
IS (1) IS6658A (enExample)
MX (1) MXPA02012425A (enExample)
MY (1) MY136520A (enExample)
NO (1) NO324698B1 (enExample)
NZ (1) NZ523047A (enExample)
PL (1) PL203936B1 (enExample)
RU (2) RU2298550C2 (enExample)
SK (1) SK17932002A3 (enExample)
WO (1) WO2001098273A1 (enExample)

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CN113767095A (zh) * 2019-05-01 2021-12-07 勃林格殷格翰国际有限公司 (r)-4-溴苯磺酸(2-甲基环氧乙烷-2-基)甲酯
EP4115885A1 (en) 2021-07-05 2023-01-11 Charité - Universitätsmedizin Berlin A pharmaceutical composition comprising bay 86-5277 and salts thereof for use in the treatment of viral infections and hyperinflammation
JP2025500826A (ja) 2021-12-14 2025-01-15 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 慢性腎疾患を処置するためのアルドステロンシンターゼ阻害薬

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