RU2317293C9 - N-замещенные амиды индолил-3-глиоксиловой кислоты противоопухолевого действия, лекарственное средство на их основе, способ их получения и способ лечения опухолевых заболеваний - Google Patents
N-замещенные амиды индолил-3-глиоксиловой кислоты противоопухолевого действия, лекарственное средство на их основе, способ их получения и способ лечения опухолевых заболеваний Download PDFInfo
- Publication number
- RU2317293C9 RU2317293C9 RU2006105708/04A RU2006105708A RU2317293C9 RU 2317293 C9 RU2317293 C9 RU 2317293C9 RU 2006105708/04 A RU2006105708/04 A RU 2006105708/04A RU 2006105708 A RU2006105708 A RU 2006105708A RU 2317293 C9 RU2317293 C9 RU 2317293C9
- Authority
- RU
- Russia
- Prior art keywords
- substituted
- alkyl
- indol
- chlorobenzyl
- quinolin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10334040.8 | 2003-07-25 | ||
| DE10334040A DE10334040A1 (de) | 2003-07-25 | 2003-07-25 | Neue N-substituierte Indolyl-3-glyoxylsäureamide, deren Verwendung als Arzneimittel und Verfahren zu deren Herstellung |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| RU2006105708A RU2006105708A (ru) | 2006-06-27 |
| RU2317293C2 RU2317293C2 (ru) | 2008-02-20 |
| RU2317293C9 true RU2317293C9 (ru) | 2008-05-10 |
Family
ID=34129467
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2006105708/04A RU2317293C9 (ru) | 2003-07-25 | 2004-07-09 | N-замещенные амиды индолил-3-глиоксиловой кислоты противоопухолевого действия, лекарственное средство на их основе, способ их получения и способ лечения опухолевых заболеваний |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP1651600A2 (de) |
| JP (1) | JP2007503376A (de) |
| KR (1) | KR20060037398A (de) |
| CN (1) | CN1839129A (de) |
| AR (1) | AR045928A1 (de) |
| AU (1) | AU2004263238A1 (de) |
| BR (1) | BRPI0412898A (de) |
| CA (1) | CA2533433A1 (de) |
| DE (1) | DE10334040A1 (de) |
| IL (1) | IL173335A0 (de) |
| MX (1) | MXPA06000995A (de) |
| NO (1) | NO20060697L (de) |
| RS (1) | RS20060049A (de) |
| RU (1) | RU2317293C9 (de) |
| TW (1) | TW200524863A (de) |
| UA (1) | UA83498C2 (de) |
| WO (1) | WO2005014542A2 (de) |
| ZA (1) | ZA200601300B (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2008019357A2 (en) | 2006-08-07 | 2008-02-14 | Ironwood Pharmaceuticals, Inc. | Indole compounds |
| AR084433A1 (es) | 2010-12-22 | 2013-05-15 | Ironwood Pharmaceuticals Inc | Inhibidores de la faah y composiciones farmaceuticas que los contienen |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2460347A1 (en) * | 2001-09-13 | 2003-03-20 | Synta Pharmaceuticals Corp. | 3-glyoxlylamideindoles for treating cancer |
-
2003
- 2003-07-25 DE DE10334040A patent/DE10334040A1/de not_active Withdrawn
-
2004
- 2004-07-09 JP JP2006521430A patent/JP2007503376A/ja not_active Withdrawn
- 2004-07-09 EP EP04740854A patent/EP1651600A2/de not_active Withdrawn
- 2004-07-09 KR KR1020067001636A patent/KR20060037398A/ko not_active Application Discontinuation
- 2004-07-09 WO PCT/EP2004/007573 patent/WO2005014542A2/de active Application Filing
- 2004-07-09 MX MXPA06000995A patent/MXPA06000995A/es unknown
- 2004-07-09 RU RU2006105708/04A patent/RU2317293C9/ru not_active IP Right Cessation
- 2004-07-09 CA CA002533433A patent/CA2533433A1/en not_active Abandoned
- 2004-07-09 CN CNA2004800240832A patent/CN1839129A/zh active Pending
- 2004-07-09 AU AU2004263238A patent/AU2004263238A1/en not_active Abandoned
- 2004-07-09 RS YUP-2006/0049A patent/RS20060049A/sr unknown
- 2004-07-09 BR BRPI0412898-2A patent/BRPI0412898A/pt not_active IP Right Cessation
- 2004-07-19 TW TW093121509A patent/TW200524863A/zh unknown
- 2004-07-23 AR ARP040102632A patent/AR045928A1/es not_active Application Discontinuation
- 2004-09-07 UA UAA200601216A patent/UA83498C2/uk unknown
-
2006
- 2006-01-24 IL IL173335A patent/IL173335A0/en unknown
- 2006-02-13 ZA ZA200601300A patent/ZA200601300B/xx unknown
- 2006-02-14 NO NO20060697A patent/NO20060697L/no not_active Application Discontinuation
Non-Patent Citations (1)
| Title |
|---|
| Li WT et al., Synthesis and biological evaluation of N-heterocyclic indolyl glyoxylamides as orally active anticancer agents. Journal of Medicinal Chemistry, 2003, 46(9), p.1706-15. * |
Also Published As
| Publication number | Publication date |
|---|---|
| TW200524863A (en) | 2005-08-01 |
| JP2007503376A (ja) | 2007-02-22 |
| IL173335A0 (en) | 2006-06-11 |
| WO2005014542A2 (de) | 2005-02-17 |
| EP1651600A2 (de) | 2006-05-03 |
| DE10334040A1 (de) | 2005-03-10 |
| WO2005014542A3 (de) | 2006-10-19 |
| MXPA06000995A (es) | 2006-04-11 |
| RU2317293C2 (ru) | 2008-02-20 |
| KR20060037398A (ko) | 2006-05-03 |
| CA2533433A1 (en) | 2005-02-17 |
| RS20060049A (en) | 2008-08-07 |
| BRPI0412898A (pt) | 2006-10-03 |
| CN1839129A (zh) | 2006-09-27 |
| AU2004263238A1 (en) | 2005-02-17 |
| ZA200601300B (en) | 2007-03-28 |
| NO20060697L (no) | 2006-02-14 |
| UA83498C2 (uk) | 2008-07-25 |
| AR045928A1 (es) | 2005-11-16 |
| RU2006105708A (ru) | 2006-06-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TH4A | Reissue of patent specification | ||
| MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20100710 |