RU2276996C2 - Лечение повреждений головного мозга, спинного мозга и нервов - Google Patents

Лечение повреждений головного мозга, спинного мозга и нервов Download PDF

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RU2276996C2
RU2276996C2 RU2002121640/15A RU2002121640A RU2276996C2 RU 2276996 C2 RU2276996 C2 RU 2276996C2 RU 2002121640/15 A RU2002121640/15 A RU 2002121640/15A RU 2002121640 A RU2002121640 A RU 2002121640A RU 2276996 C2 RU2276996 C2 RU 2276996C2
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substance
receptor antagonist
brain
damage
composition according
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RU2002121640/15A
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Russian (ru)
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RU2002121640A (ru
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Роберт ВИНК (AU)
Роберт ВИНК
Алан Джон НИММОУ (AU)
Алан Джон НИММОУ
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Ф.Хоффманн-Ля Рош Аг
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00—Medicinal preparations containing inorganic active ingredients
    • A61K33/06—Aluminium, calcium or magnesium; Compounds thereof, e.g. clay
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/455—Nicotinic acids, e.g. niacin; Derivatives thereof, e.g. esters, amides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00—Medicinal preparations containing inorganic active ingredients
    • A61K33/14—Alkali metal chlorides; Alkaline earth metal chlorides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
RU2002121640/15A 2000-01-18 2001-01-18 Лечение повреждений головного мозга, спинного мозга и нервов RU2276996C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AUPQ5146A AUPQ514600A0 (en) 2000-01-18 2000-01-18 Brain injury treatment
AUPQ5146 2000-01-18

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RU2002121640A RU2002121640A (ru) 2004-03-27
RU2276996C2 true RU2276996C2 (ru) 2006-05-27

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US (5) US6841551B2 (enExample)
EP (1) EP1261335B1 (enExample)
JP (1) JP4794794B2 (enExample)
KR (1) KR100780119B1 (enExample)
CN (1) CN1261095C (enExample)
AU (2) AUPQ514600A0 (enExample)
BR (1) BR0107695A (enExample)
CA (1) CA2397723C (enExample)
CZ (1) CZ20022804A3 (enExample)
DE (1) DE60139244D1 (enExample)
HR (1) HRP20020593B1 (enExample)
HU (1) HUP0301920A3 (enExample)
IL (2) IL150548A0 (enExample)
MX (1) MXPA02007004A (enExample)
NO (1) NO329320B1 (enExample)
NZ (2) NZ519990A (enExample)
RU (1) RU2276996C2 (enExample)
WO (1) WO2001052844A1 (enExample)
YU (1) YU54702A (enExample)
ZA (1) ZA200205715B (enExample)

Cited By (1)

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Publication number Priority date Publication date Assignee Title
RU2749191C2 (ru) * 2011-03-14 2021-06-07 Н.В. Нютрисиа Способ лечения нейротравмы

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CN1261095C (zh) 2006-06-28
IL150548A0 (en) 2003-02-12
BR0107695A (pt) 2002-10-15
KR20020075784A (ko) 2002-10-05
CA2397723C (en) 2010-08-31
US10201568B2 (en) 2019-02-12
CN1426302A (zh) 2003-06-25
CZ20022804A3 (cs) 2002-11-13
MXPA02007004A (es) 2004-10-15
US20180071333A1 (en) 2018-03-15
EP1261335A4 (en) 2004-09-22
NZ534278A (en) 2005-08-26
JP4794794B2 (ja) 2011-10-19
NO20023423D0 (no) 2002-07-17
WO2001052844A1 (en) 2001-07-26
AU782799B2 (en) 2005-09-01
US6841551B2 (en) 2005-01-11
EP1261335A1 (en) 2002-12-04
US20030109417A1 (en) 2003-06-12
ZA200205715B (en) 2003-10-17
KR100780119B1 (ko) 2007-11-27
EP1261335B1 (en) 2009-07-15
PL358251A1 (en) 2004-08-09
HRP20020593A2 (en) 2005-10-31
IL150548A (en) 2011-05-31
NZ519990A (en) 2004-10-29
AUPQ514600A0 (en) 2000-02-10
AU2656001A (en) 2001-07-31
CA2397723A1 (en) 2001-07-26
US20050107380A1 (en) 2005-05-19
HUP0301920A3 (en) 2010-03-29
NO20023423L (no) 2002-09-16
US20160030474A1 (en) 2016-02-04
US20090253698A1 (en) 2009-10-08
NO329320B1 (no) 2010-09-27
YU54702A (sh) 2006-01-16
JP2003520232A (ja) 2003-07-02
RU2002121640A (ru) 2004-03-27
HK1054872A1 (en) 2003-12-19
HUP0301920A2 (hu) 2003-09-29
US9186404B2 (en) 2015-11-17
HRP20020593B1 (hr) 2011-03-31
DE60139244D1 (de) 2009-08-27

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