RS62317B1 - Trpv4 antagonisti - Google Patents

Trpv4 antagonisti

Info

Publication number
RS62317B1
RS62317B1 RS20211119A RSP20211119A RS62317B1 RS 62317 B1 RS62317 B1 RS 62317B1 RS 20211119 A RS20211119 A RS 20211119A RS P20211119 A RSP20211119 A RS P20211119A RS 62317 B1 RS62317 B1 RS 62317B1
Authority
RS
Serbia
Prior art keywords
sulfonyl
hydroxy
pyrrolidin
hydroxymethyl
oxy
Prior art date
Application number
RS20211119A
Other languages
English (en)
Serbian (sr)
Inventor
Edward J Brnardic
Carl A Brooks
Brian Griffin Lawhorn
Guosen Ye
Linda S Barton
Brian W Budzik
Jay M Matthews
John Jeffrey Mcatee
Jaclyn R Patterson
Joseph E Pero
Robert Sanchez
Matthew Robert Sender
Lamont Roscoe Terrell
David J Behm
James V Thomas
Original Assignee
Glaxosmithkline Ip No 2 Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Ip No 2 Ltd filed Critical Glaxosmithkline Ip No 2 Ltd
Publication of RS62317B1 publication Critical patent/RS62317B1/sr

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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