HUE056059T2 - TRPV4 antagonisták - Google Patents

TRPV4 antagonisták

Info

Publication number
HUE056059T2
HUE056059T2 HUE17784400A HUE17784400A HUE056059T2 HU E056059 T2 HUE056059 T2 HU E056059T2 HU E17784400 A HUE17784400 A HU E17784400A HU E17784400 A HUE17784400 A HU E17784400A HU E056059 T2 HUE056059 T2 HU E056059T2
Authority
HU
Hungary
Prior art keywords
trpv4 antagonists
trpv4
antagonists
Prior art date
Application number
HUE17784400A
Other languages
English (en)
Inventor
Edward J Brnardic
Carl A Brooks
Brian Griffin Lawhorn
Guosen Ye
Linda S Barton
Brian W Budzik
Jay M Matthews
John Jeffrey Mcatee
Jaclyn R Patterson
Joseph E Pero
Robert Sanchez
Matthew Robert Sender
Lamont Roscoe Terrell
David J Behm
James V Thomas
Original Assignee
Glaxosmithkline Ip No 2 Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxosmithkline Ip No 2 Ltd filed Critical Glaxosmithkline Ip No 2 Ltd
Publication of HUE056059T2 publication Critical patent/HUE056059T2/hu

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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