HK1247916A1 - 新型5-ht2拮抗劑 - Google Patents
新型5-ht2拮抗劑Info
- Publication number
- HK1247916A1 HK1247916A1 HK18107294.8A HK18107294A HK1247916A1 HK 1247916 A1 HK1247916 A1 HK 1247916A1 HK 18107294 A HK18107294 A HK 18107294A HK 1247916 A1 HK1247916 A1 HK 1247916A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- antagonists
- novel
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrane Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Indole Compounds (AREA)
- Quinoline Compounds (AREA)
- Furan Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP15173111.4A EP3109237A1 (en) | 2015-06-22 | 2015-06-22 | Novel 5-ht2 antagonists |
| PCT/EP2016/064446 WO2016207231A1 (en) | 2015-06-22 | 2016-06-22 | Novel 5-ht2 antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK1247916A1 true HK1247916A1 (zh) | 2018-10-05 |
Family
ID=53496439
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK18107294.8A HK1247916A1 (zh) | 2015-06-22 | 2018-06-04 | 新型5-ht2拮抗劑 |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US10544103B2 (zh) |
| EP (2) | EP3109237A1 (zh) |
| JP (1) | JP6718886B2 (zh) |
| KR (1) | KR102610630B1 (zh) |
| CN (1) | CN107787321B (zh) |
| AU (1) | AU2016282325B2 (zh) |
| CA (1) | CA2988033C (zh) |
| CY (1) | CY1123880T1 (zh) |
| DK (1) | DK3310762T3 (zh) |
| ES (1) | ES2819499T3 (zh) |
| HK (1) | HK1247916A1 (zh) |
| HR (1) | HRP20201485T1 (zh) |
| HU (1) | HUE050667T2 (zh) |
| IL (1) | IL256496B (zh) |
| LT (1) | LT3310762T (zh) |
| MX (1) | MX2017016939A (zh) |
| PL (1) | PL3310762T3 (zh) |
| PT (1) | PT3310762T (zh) |
| RS (1) | RS61266B1 (zh) |
| RU (1) | RU2706229C2 (zh) |
| SI (1) | SI3310762T1 (zh) |
| WO (1) | WO2016207231A1 (zh) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3753924A1 (en) | 2019-06-18 | 2020-12-23 | AnaMar AB | New tricyclic 5-ht2 antagonists |
| WO2021042038A1 (en) * | 2019-08-29 | 2021-03-04 | University Of Cincinnati | Treatment of pain by targeting nr4a1 |
| AU2023250955A1 (en) * | 2022-04-07 | 2024-10-17 | Corbus Pharmaceuticals, Inc. | Cannabinoid receptor 1 antagonists/inverse agonists and uses thereof |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US641992A (en) * | 1898-03-31 | 1900-01-23 | Guillaume Arnaud Nussbaum | Steam-generator. |
| GB1223491A (en) * | 1967-10-13 | 1971-02-24 | American Home Prod | Guanidines |
| US4107326A (en) | 1977-05-06 | 1978-08-15 | American Cyanamid Company | Novel benzylideneaminoguanidines |
| DZ3335A1 (fr) | 2000-03-23 | 2001-09-27 | Solvay Pharm Bv | Derives de 4,5-dihydro-1h-pyrazole ayant une activite antagoniste de cb1 |
| CA2532316A1 (en) | 2003-07-15 | 2005-01-27 | Bayer Healthcare Ag | Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases |
| DE102004061750A1 (de) | 2004-12-22 | 2006-07-06 | Bayer Healthcare Ag | Heteroaryl-substituierte Pyrazoline |
| DE102005014089A1 (de) | 2005-03-22 | 2006-09-28 | Schering Ag | Tetrahydronaphthalinderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer |
| JP5157892B2 (ja) * | 2006-02-20 | 2013-03-06 | アステラス製薬株式会社 | アミド誘導体またはその塩 |
| CN101431994A (zh) | 2006-04-27 | 2009-05-13 | 索尔瓦药物有限公司 | CBx大麻素受体调节剂作为钾通道调节剂的用途 |
| EP1882475A1 (en) * | 2006-07-26 | 2008-01-30 | Novartis AG | Method of treating disorders mediated by the fibroblast growth factor receptor |
| AR062907A1 (es) | 2006-09-22 | 2008-12-17 | Solvay Pharm Bv | Derivados de sulfonilpirazol y sulfonilpirazolincarboxamidina como antagonistas de 5-ht6 |
| AR070898A1 (es) * | 2008-03-18 | 2010-05-12 | Solvay Pharm Bv | Derivados de arilsulfonil pirazolin carboxamidina como antagonistas de 5-ht6 |
| EP2470270A1 (en) * | 2009-07-31 | 2012-07-04 | AnaMar AB | Compounds for treatment of inflammation |
| WO2012008528A1 (ja) * | 2010-07-15 | 2012-01-19 | 大日本住友製薬株式会社 | ピラゾール化合物 |
| CA2837524C (en) | 2011-07-01 | 2019-08-20 | Merck Patent Gmbh | Dihydropyrazoles |
-
2015
- 2015-06-22 EP EP15173111.4A patent/EP3109237A1/en not_active Withdrawn
-
2016
- 2016-06-22 PT PT167318716T patent/PT3310762T/pt unknown
- 2016-06-22 LT LTEP16731871.6T patent/LT3310762T/lt unknown
- 2016-06-22 WO PCT/EP2016/064446 patent/WO2016207231A1/en active Application Filing
- 2016-06-22 AU AU2016282325A patent/AU2016282325B2/en active Active
- 2016-06-22 DK DK16731871.6T patent/DK3310762T3/da active
- 2016-06-22 PL PL16731871T patent/PL3310762T3/pl unknown
- 2016-06-22 ES ES16731871T patent/ES2819499T3/es active Active
- 2016-06-22 JP JP2017561762A patent/JP6718886B2/ja active Active
- 2016-06-22 RS RS20201293A patent/RS61266B1/sr unknown
- 2016-06-22 SI SI201630908T patent/SI3310762T1/sl unknown
- 2016-06-22 US US15/737,125 patent/US10544103B2/en active Active
- 2016-06-22 RU RU2017140648A patent/RU2706229C2/ru active
- 2016-06-22 CN CN201680036640.5A patent/CN107787321B/zh active Active
- 2016-06-22 MX MX2017016939A patent/MX2017016939A/es unknown
- 2016-06-22 HU HUE16731871A patent/HUE050667T2/hu unknown
- 2016-06-22 KR KR1020187001184A patent/KR102610630B1/ko active IP Right Grant
- 2016-06-22 EP EP16731871.6A patent/EP3310762B1/en active Active
- 2016-06-22 CA CA2988033A patent/CA2988033C/en active Active
-
2017
- 2017-12-21 IL IL256496A patent/IL256496B/en active IP Right Grant
-
2018
- 2018-06-04 HK HK18107294.8A patent/HK1247916A1/zh unknown
-
2020
- 2020-09-17 HR HRP20201485TT patent/HRP20201485T1/hr unknown
- 2020-10-06 CY CY20201100935T patent/CY1123880T1/el unknown
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