RS56498B1 - Heterociklična jedinjenja, medikamenti koji sadrže navedena jedinjenja, njihova primena i postupci za njihovo dobijanje - Google Patents

Heterociklična jedinjenja, medikamenti koji sadrže navedena jedinjenja, njihova primena i postupci za njihovo dobijanje

Info

Publication number
RS56498B1
RS56498B1 RS20171069A RSP20171069A RS56498B1 RS 56498 B1 RS56498 B1 RS 56498B1 RS 20171069 A RS20171069 A RS 20171069A RS P20171069 A RSP20171069 A RS P20171069A RS 56498 B1 RS56498 B1 RS 56498B1
Authority
RS
Serbia
Prior art keywords
tube
grooves
opening
ring
needle
Prior art date
Application number
RS20171069A
Other languages
English (en)
Serbian (sr)
Inventor
Armin Heckel
Sara Frattini
Dieter Hamprecht
Joerg Kley
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of RS56498B1 publication Critical patent/RS56498B1/sr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Virology (AREA)
  • Immunology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Infusion, Injection, And Reservoir Apparatuses (AREA)
RS20171069A 2011-11-02 2012-10-29 Heterociklična jedinjenja, medikamenti koji sadrže navedena jedinjenja, njihova primena i postupci za njihovo dobijanje RS56498B1 (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11187553 2011-11-02
EP12777930.4A EP2773633B1 (en) 2011-11-02 2012-10-29 Heterocyclic compounds, medicaments containing said compounds, use thereof and processes for the preparation thereof
PCT/EP2012/071352 WO2013064450A1 (en) 2011-11-02 2012-10-29 Heterocyclic compounds, medicaments containing said compounds, use thereof and processes for the preparation thereof

Publications (1)

Publication Number Publication Date
RS56498B1 true RS56498B1 (sr) 2018-01-31

Family

ID=47073464

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20171069A RS56498B1 (sr) 2011-11-02 2012-10-29 Heterociklična jedinjenja, medikamenti koji sadrže navedena jedinjenja, njihova primena i postupci za njihovo dobijanje

Country Status (34)

Country Link
US (4) US8759349B2 (cg-RX-API-DMAC7.html)
EP (1) EP2773633B1 (cg-RX-API-DMAC7.html)
JP (1) JP6091513B2 (cg-RX-API-DMAC7.html)
KR (1) KR102006612B1 (cg-RX-API-DMAC7.html)
CN (2) CN106279110B (cg-RX-API-DMAC7.html)
AP (1) AP2014007670A0 (cg-RX-API-DMAC7.html)
AU (1) AU2012331274B2 (cg-RX-API-DMAC7.html)
BR (1) BR112014010583A2 (cg-RX-API-DMAC7.html)
CA (1) CA2854217C (cg-RX-API-DMAC7.html)
CL (1) CL2014001047A1 (cg-RX-API-DMAC7.html)
CO (1) CO6940429A2 (cg-RX-API-DMAC7.html)
CY (1) CY1120974T1 (cg-RX-API-DMAC7.html)
DK (1) DK2773633T3 (cg-RX-API-DMAC7.html)
EA (1) EA025158B9 (cg-RX-API-DMAC7.html)
EC (1) ECSP14001929A (cg-RX-API-DMAC7.html)
ES (1) ES2645744T3 (cg-RX-API-DMAC7.html)
GE (1) GEP20186880B (cg-RX-API-DMAC7.html)
HR (1) HRP20171614T1 (cg-RX-API-DMAC7.html)
HU (1) HUE034929T2 (cg-RX-API-DMAC7.html)
IL (1) IL232035A (cg-RX-API-DMAC7.html)
LT (1) LT2773633T (cg-RX-API-DMAC7.html)
ME (1) ME02905B (cg-RX-API-DMAC7.html)
MX (1) MX348522B (cg-RX-API-DMAC7.html)
NO (1) NO2773633T3 (cg-RX-API-DMAC7.html)
PE (1) PE20141607A1 (cg-RX-API-DMAC7.html)
PH (1) PH12014500970B1 (cg-RX-API-DMAC7.html)
PL (1) PL2773633T3 (cg-RX-API-DMAC7.html)
PT (1) PT2773633T (cg-RX-API-DMAC7.html)
RS (1) RS56498B1 (cg-RX-API-DMAC7.html)
SG (1) SG11201401907TA (cg-RX-API-DMAC7.html)
SI (1) SI2773633T1 (cg-RX-API-DMAC7.html)
TN (1) TN2014000180A1 (cg-RX-API-DMAC7.html)
UA (1) UA115868C2 (cg-RX-API-DMAC7.html)
WO (1) WO2013064450A1 (cg-RX-API-DMAC7.html)

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HUE032813T2 (en) 2005-12-28 2017-11-28 Vertex Pharma Solid forms of N- [2,4-bis (1,1-dimethyl ethyl) -5-hydroxyphenyl] -1,4-dihydro-4-oxoquinoline-3-carboxamide
PL2773633T3 (pl) * 2011-11-02 2018-01-31 Boehringer Ingelheim Int Związki heterocykliczne, leki zawierające wymienione związki, ich zastosowanie i procesy ich wytwarzania
KR20160054460A (ko) * 2013-07-02 2016-05-16 더 캘리포니아 인스티튜트 포 바이오메디칼 리써치 낭성 섬유증의 치료를 위한 화합물
WO2015003958A1 (en) * 2013-07-08 2015-01-15 Boehringer Ingelheim International Gmbh Amiloride-type compounds as inhibitors in epithelial sodium channels for the treatment of diseases of the lungs and airways
EP3204358B1 (en) 2014-10-07 2018-09-19 Vertex Pharmaceuticals Incorporated Co-crystals of modulators of cystic fibrosis transmembrane conductance regulator
SG11201703284XA (en) 2014-10-24 2017-06-29 Ono Pharmaceutical Co Kcnq2-5 channel activator
HK1246718A1 (zh) * 2015-01-07 2018-09-14 斯克利普斯研究所 用於治疗囊性纤维化的化合物
GB201610854D0 (en) 2016-06-21 2016-08-03 Entpr Therapeutics Ltd Compounds
GB201619694D0 (en) 2016-11-22 2017-01-04 Entpr Therapeutics Ltd Compounds
GB201717051D0 (en) 2017-10-17 2017-11-29 Enterprise Therapeutics Ltd Compounds
GB201808093D0 (en) 2018-05-18 2018-07-04 Enterprise Therapeutics Ltd Compounds
AU2021341508A1 (en) 2020-09-10 2023-05-25 Precirix N.V. Antibody fragment against fap
CN112107580A (zh) * 2020-09-29 2020-12-22 北京鑫开元医药科技有限公司 一种脾酪氨酸激酶抑制剂的制剂组合物及其制备方法
WO2023203135A1 (en) 2022-04-22 2023-10-26 Precirix N.V. Improved radiolabelled antibody
IL318992A (en) 2022-05-02 2025-04-01 Precirix N V Cancer treatment through advance directives
WO2024243025A1 (en) * 2023-05-19 2024-11-28 Ikena Oncology, Inc. Naphthyl-substituted pyrido[4,3-d]pyrimidines and related compounds and their use in treating medical conditions

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NL6812003A (cg-RX-API-DMAC7.html) 1967-09-07 1969-03-11
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AU774865B2 (en) 1999-07-19 2004-07-08 University Of North Carolina At Chapel Hill, The Conjugates of sodium channel blockers and methods of using the same
WO2001052902A1 (en) 2000-01-24 2001-07-26 Isis Pharmaceuticals, Inc. Antisense modulation of inducible nitric oxide synthase expression
WO2006023573A2 (en) 2004-08-18 2006-03-02 Johnson Michael R Aliphatic amide & ester pyrazinoylguanidine sodium channel blockers
GB0526244D0 (en) * 2005-12-22 2006-02-01 Novartis Ag Organic compounds
WO2008013557A1 (en) * 2006-07-24 2008-01-31 International Stem Cell Corporation Synthetic cornea from retinal stem cells
ATE499363T1 (de) * 2007-05-07 2011-03-15 Novartis Ag Organische verbindungen
NZ585789A (en) 2007-12-10 2012-03-30 Novartis Ag Pyrazine-2-carboxamide derivatives to treat diseases mediated by blockade of the epithelial sodium channel
EP2285785B1 (en) * 2008-05-13 2012-09-05 Novartis AG 3,5-diamino-6-chloro-pyrazine-2-carboxylic acid derivatives and their use as epithelial sodium channel blockers for the treatment of arway diseases
MX2010013675A (es) 2008-06-10 2011-02-15 Novartis Ag Derivados de pirazina como bloqueadores del canal de sodio epitelial.
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PL2773633T3 (pl) * 2011-11-02 2018-01-31 Boehringer Ingelheim Int Związki heterocykliczne, leki zawierające wymienione związki, ich zastosowanie i procesy ich wytwarzania

Also Published As

Publication number Publication date
IL232035A0 (en) 2014-05-28
EA025158B9 (ru) 2018-03-30
MX2014005166A (es) 2014-05-28
HUE034929T2 (en) 2018-03-28
KR20140085498A (ko) 2014-07-07
JP2014534222A (ja) 2014-12-18
PH12014500970B1 (en) 2017-10-06
CA2854217A1 (en) 2013-05-10
AP2014007670A0 (en) 2014-05-31
US20180194747A1 (en) 2018-07-12
SG11201401907TA (en) 2014-05-29
JP6091513B2 (ja) 2017-03-08
GEP20186880B (en) 2018-07-25
DK2773633T3 (da) 2017-11-13
US20150336933A1 (en) 2015-11-26
EP2773633A1 (en) 2014-09-10
ME02905B (me) 2018-10-20
PT2773633T (pt) 2017-11-14
KR102006612B1 (ko) 2019-08-02
UA115868C2 (uk) 2018-01-10
PH12014500970A1 (en) 2014-06-09
MX348522B (es) 2017-06-16
SI2773633T1 (sl) 2017-11-30
TN2014000180A1 (en) 2015-09-30
ECSP14001929A (es) 2015-11-30
AU2012331274A1 (en) 2014-04-03
IL232035A (en) 2017-05-29
EP2773633B1 (en) 2017-08-02
US20130109697A1 (en) 2013-05-02
BR112014010583A2 (pt) 2020-04-22
NZ622469A (en) 2016-08-26
PL2773633T3 (pl) 2018-01-31
ES2645744T3 (es) 2017-12-07
LT2773633T (lt) 2017-11-10
CL2014001047A1 (es) 2014-11-07
NO2773633T3 (cg-RX-API-DMAC7.html) 2017-12-30
US20140228374A1 (en) 2014-08-14
CN106279110B (zh) 2019-12-10
CN104024244A (zh) 2014-09-03
EA201400521A1 (ru) 2014-09-30
CY1120974T1 (el) 2019-12-11
AU2012331274B2 (en) 2017-06-08
HK1196819A1 (zh) 2014-12-24
US9920035B2 (en) 2018-03-20
PE20141607A1 (es) 2014-11-23
CN104024244B (zh) 2016-09-14
CN106279110A (zh) 2017-01-04
EA025158B1 (ru) 2016-11-30
CA2854217C (en) 2019-12-31
WO2013064450A1 (en) 2013-05-10
CO6940429A2 (es) 2014-05-09
HRP20171614T1 (hr) 2017-12-01
US8759349B2 (en) 2014-06-24

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