RS52128B - Postupak za proizvodnju [fenilsulfanilfenil] piperidina - Google Patents

Postupak za proizvodnju [fenilsulfanilfenil] piperidina

Info

Publication number
RS52128B
RS52128B RS20120063A RSP20120063A RS52128B RS 52128 B RS52128 B RS 52128B RS 20120063 A RS20120063 A RS 20120063A RS P20120063 A RSP20120063 A RS P20120063A RS 52128 B RS52128 B RS 52128B
Authority
RS
Serbia
Prior art keywords
compound
alkyl
formula
acid
hydrogen
Prior art date
Application number
RS20120063A
Other languages
English (en)
Serbian (sr)
Inventor
Michael Harold Rock
Sebastian Brandes
Original Assignee
H. Lundbeck A/S
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by H. Lundbeck A/S filed Critical H. Lundbeck A/S
Publication of RS52128B publication Critical patent/RS52128B/sr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/52Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
RS20120063A 2008-03-03 2009-03-02 Postupak za proizvodnju [fenilsulfanilfenil] piperidina RS52128B (sr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US3309308P 2008-03-03 2008-03-03
DKPA200800314 2008-03-03
PCT/EP2009/052440 WO2009109541A1 (en) 2008-03-03 2009-03-02 Process for the manufacture of [phenylsulfanylphenyl]piperidines

Publications (1)

Publication Number Publication Date
RS52128B true RS52128B (sr) 2012-08-31

Family

ID=40547924

Family Applications (1)

Application Number Title Priority Date Filing Date
RS20120063A RS52128B (sr) 2008-03-03 2009-03-02 Postupak za proizvodnju [fenilsulfanilfenil] piperidina

Country Status (28)

Country Link
US (1) US8362255B2 (enExample)
EP (1) EP2260024B1 (enExample)
JP (1) JP5564439B2 (enExample)
KR (1) KR20100122914A (enExample)
CN (1) CN101959859B (enExample)
AR (1) AR070737A1 (enExample)
AT (1) ATE539055T1 (enExample)
AU (1) AU2009221170B2 (enExample)
BR (1) BRPI0908166A2 (enExample)
CA (1) CA2715579A1 (enExample)
CL (1) CL2009000490A1 (enExample)
CO (1) CO6290758A2 (enExample)
CY (1) CY1113887T1 (enExample)
DK (1) DK2260024T3 (enExample)
EA (1) EA017855B1 (enExample)
ES (1) ES2377862T3 (enExample)
HR (1) HRP20120118T1 (enExample)
IL (1) IL207471A (enExample)
MX (1) MX2010008729A (enExample)
NZ (1) NZ587593A (enExample)
PL (1) PL2260024T3 (enExample)
PT (1) PT2260024E (enExample)
RS (1) RS52128B (enExample)
SI (1) SI2260024T1 (enExample)
TW (1) TW200940505A (enExample)
UA (1) UA98698C2 (enExample)
WO (1) WO2009109541A1 (enExample)
ZA (1) ZA201006135B (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2007260356B2 (en) * 2006-06-16 2013-01-24 H. Lundbeck A/S Crystalline forms of 4- [2- (4-methylphenylsulfanyl) -phenyl] piperidine with combined serotonin and norepinephrine reuptake inhibition for the treatment of neuropathic pain
JP2012163850A (ja) * 2011-02-08 2012-08-30 Nippon Sheet Glass Co Ltd 正立等倍レンズアレイプレート、光走査ユニット、画像読取装置および画像書込装置
KR20150013548A (ko) 2012-05-21 2015-02-05 노파르티스 아게 키나제 억제제로서의 신규 고리-치환된 n-피리디닐 아미드
CN104710345B (zh) * 2013-12-17 2017-09-05 江苏恩华药业股份有限公司 用于制备4‑(2‑(4‑甲基苯基硫基))苯基哌啶的化合物、其制备方法及应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2324087A (en) * 1997-04-10 1998-10-14 Merck & Co Inc Preparation of (S)-3-Carbethoxy-3-benzylpiperidine
AU1805701A (en) 1999-12-20 2001-07-03 Eli Lilly And Company A process for preparing trans-2,4-disubstituted piperidines
UA81749C2 (uk) * 2001-10-04 2008-02-11 Х. Луннбек А/С Фенілпіперазинові похідні як інгібітори зворотного захоплення серотоніну
UA81300C2 (en) * 2003-04-04 2007-12-25 Lundbeck & Co As H Derivates of 4-(2-fenilsulfanilfenil)-1,2,3,6-tetrahydropiridin as retarding agents of serotonin recapture
CA2521258C (en) * 2003-04-04 2009-12-01 H. Lundbeck A/S 4-(2-phenylsulfanyl-phenyl)-piperidine derivatives as serotonin reuptake inhibitors
AU2007260356B2 (en) * 2006-06-16 2013-01-24 H. Lundbeck A/S Crystalline forms of 4- [2- (4-methylphenylsulfanyl) -phenyl] piperidine with combined serotonin and norepinephrine reuptake inhibition for the treatment of neuropathic pain

Also Published As

Publication number Publication date
AU2009221170B2 (en) 2013-08-22
IL207471A0 (en) 2010-12-30
HRP20120118T1 (hr) 2012-03-31
AR070737A1 (es) 2010-04-28
US20110054178A1 (en) 2011-03-03
WO2009109541A1 (en) 2009-09-11
JP5564439B2 (ja) 2014-07-30
HK1153458A1 (en) 2012-03-30
US8362255B2 (en) 2013-01-29
CN101959859A (zh) 2011-01-26
AU2009221170A1 (en) 2009-09-11
DK2260024T3 (da) 2012-02-27
CN101959859B (zh) 2013-08-14
NZ587593A (en) 2012-03-30
ES2377862T3 (es) 2012-04-02
CA2715579A1 (en) 2009-09-11
ATE539055T1 (de) 2012-01-15
BRPI0908166A2 (pt) 2015-08-11
MX2010008729A (es) 2010-09-24
EP2260024A1 (en) 2010-12-15
CL2009000490A1 (es) 2010-04-16
TW200940505A (en) 2009-10-01
EP2260024B1 (en) 2011-12-28
JP2011513358A (ja) 2011-04-28
ZA201006135B (en) 2011-10-26
EA201071025A1 (ru) 2011-02-28
KR20100122914A (ko) 2010-11-23
CY1113887T1 (el) 2016-07-27
UA98698C2 (en) 2012-06-11
CO6290758A2 (es) 2011-06-20
PL2260024T3 (pl) 2012-04-30
IL207471A (en) 2014-06-30
EA017855B1 (ru) 2013-03-29
PT2260024E (pt) 2012-03-06
SI2260024T1 (sl) 2012-04-30

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