RS20070369A - Conversion of 2-pyrazolines to pyrazoles using bromine - Google Patents
Conversion of 2-pyrazolines to pyrazoles using bromineInfo
- Publication number
- RS20070369A RS20070369A RSP-2007/0369A RSP20070369A RS20070369A RS 20070369 A RS20070369 A RS 20070369A RS P20070369 A RSP20070369 A RS P20070369A RS 20070369 A RS20070369 A RS 20070369A
- Authority
- RS
- Serbia
- Prior art keywords
- formula
- bromine
- pyrazolines
- pyrazoles
- conversion
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Chemical Treatment Of Metals (AREA)
- Enzymes And Modification Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
Ovaj pronalazak se odnosi na postupak izrade jedinjenja sa Formulom 1 gde su: L, R1, R2 i X, kao što su izloženi u opisu, koji obuhvata dovođenje u kontakt 2-pirazolina Formule 2 sa bromom na temperaturi od najmanje oko 80°C (Formula 1) (Formula 2). Ovaj pronalazak, takođe, izlaže izradu jedinjenja sa Formulom 3 gde su: X, Z, R5, R6, R7, R8a, R8b i n, kao što su definisani u opisu, upotrebom jedinjenja sa Formulom la, gde je R10, kao što je definisan u opisu, a koje je pripremljeno pomoću gore pomenutog postupka za izradu jedinjenja sa Formulom 1. (Formula 3) (Formula 4).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US66341005P | 2005-03-18 | 2005-03-18 | |
PCT/US2006/009617 WO2006102025A1 (en) | 2005-03-18 | 2006-03-14 | Conversion of 2-pyrazolines to pyrazoles using bromine |
Publications (1)
Publication Number | Publication Date |
---|---|
RS20070369A true RS20070369A (en) | 2009-01-22 |
Family
ID=36592996
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RS20120261A RS52344B (sr) | 2005-03-18 | 2006-03-14 | Konverzija 2-pirazolina u pirazole upotrebom broma |
RSP-2007/0369A RS20070369A (en) | 2005-03-18 | 2006-03-14 | Conversion of 2-pyrazolines to pyrazoles using bromine |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
RS20120261A RS52344B (sr) | 2005-03-18 | 2006-03-14 | Konverzija 2-pirazolina u pirazole upotrebom broma |
Country Status (20)
Country | Link |
---|---|
US (1) | US7951953B2 (sr) |
EP (1) | EP1858878B1 (sr) |
JP (1) | JP5086987B2 (sr) |
KR (1) | KR101337159B1 (sr) |
CN (1) | CN101142207B (sr) |
AT (1) | ATE555103T1 (sr) |
AU (1) | AU2006227484B2 (sr) |
BR (1) | BRPI0609844B1 (sr) |
CA (1) | CA2601870C (sr) |
DK (1) | DK1858878T3 (sr) |
ES (1) | ES2385496T3 (sr) |
IL (1) | IL185329A (sr) |
MX (1) | MX2007011162A (sr) |
PL (1) | PL1858878T3 (sr) |
RS (2) | RS52344B (sr) |
RU (1) | RU2410381C2 (sr) |
TW (1) | TWI371449B (sr) |
UA (1) | UA93869C2 (sr) |
WO (1) | WO2006102025A1 (sr) |
ZA (1) | ZA200707470B (sr) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1924575A1 (en) * | 2005-08-24 | 2008-05-28 | E.I.Du pont de nemours and company | Anthranilamides for controlling invertebrate pests |
CN101550130B (zh) * | 2008-04-01 | 2012-11-07 | 中国中化股份有限公司 | 一种制备3-卤代-1-(3-氯-2-吡啶基)-1h-吡唑-5-甲酰卤的方法 |
CN101863874B (zh) * | 2009-04-14 | 2013-11-06 | 中国中化股份有限公司 | 一种吡唑亚胺类化合物及其应用 |
JP5972868B2 (ja) | 2010-06-15 | 2016-08-17 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH | アントラニル酸ジアミド誘導体 |
TW202128643A (zh) * | 2019-11-11 | 2021-08-01 | 美商富曼西公司 | 用於製備3—溴—1—(3—氯吡啶—2—基)—1h—吡唑—5—羧酸乙酯的方法 |
TW202140436A (zh) * | 2020-01-08 | 2021-11-01 | 美商富曼西公司 | 用於製備3-溴-1-(3-氯吡啶-2-基)-1h-吡唑-5-羧酸乙酯的方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI371450B (en) | 2001-08-13 | 2012-09-01 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-carboxylates,their preparation and use |
TWI325302B (en) | 2001-08-13 | 2010-06-01 | Du Pont | Benzoxazinone compounds |
TWI343376B (en) | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
-
2006
- 2006-03-14 RS RS20120261A patent/RS52344B/sr unknown
- 2006-03-14 BR BRPI0609844-4A patent/BRPI0609844B1/pt active IP Right Grant
- 2006-03-14 CN CN2006800087738A patent/CN101142207B/zh active Active
- 2006-03-14 AU AU2006227484A patent/AU2006227484B2/en active Active
- 2006-03-14 RS RSP-2007/0369A patent/RS20070369A/sr unknown
- 2006-03-14 CA CA2601870A patent/CA2601870C/en not_active Expired - Fee Related
- 2006-03-14 ZA ZA200707470A patent/ZA200707470B/xx unknown
- 2006-03-14 EP EP06738651A patent/EP1858878B1/en active Active
- 2006-03-14 KR KR1020077023792A patent/KR101337159B1/ko active IP Right Grant
- 2006-03-14 US US11/885,325 patent/US7951953B2/en active Active
- 2006-03-14 AT AT06738651T patent/ATE555103T1/de active
- 2006-03-14 MX MX2007011162A patent/MX2007011162A/es active IP Right Grant
- 2006-03-14 PL PL06738651T patent/PL1858878T3/pl unknown
- 2006-03-14 UA UAA200709764A patent/UA93869C2/ru unknown
- 2006-03-14 JP JP2008502077A patent/JP5086987B2/ja active Active
- 2006-03-14 DK DK06738651.6T patent/DK1858878T3/da active
- 2006-03-14 TW TW095108602A patent/TWI371449B/zh active
- 2006-03-14 ES ES06738651T patent/ES2385496T3/es active Active
- 2006-03-14 RU RU2007138552/04A patent/RU2410381C2/ru active
- 2006-03-14 WO PCT/US2006/009617 patent/WO2006102025A1/en active Application Filing
-
2007
- 2007-08-16 IL IL185329A patent/IL185329A/en active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
AU2006227484A1 (en) | 2006-09-28 |
CN101142207B (zh) | 2011-10-05 |
KR20070112292A (ko) | 2007-11-22 |
UA93869C2 (en) | 2011-03-25 |
JP5086987B2 (ja) | 2012-11-28 |
MX2007011162A (es) | 2007-10-17 |
DK1858878T3 (da) | 2012-08-06 |
EP1858878B1 (en) | 2012-04-25 |
BRPI0609844B1 (pt) | 2015-06-30 |
TWI371449B (en) | 2012-09-01 |
RS52344B (sr) | 2012-12-31 |
RU2410381C2 (ru) | 2011-01-27 |
ZA200707470B (en) | 2008-12-31 |
ATE555103T1 (de) | 2012-05-15 |
US20080177078A1 (en) | 2008-07-24 |
RU2007138552A (ru) | 2009-04-27 |
ES2385496T3 (es) | 2012-07-25 |
US7951953B2 (en) | 2011-05-31 |
WO2006102025A1 (en) | 2006-09-28 |
CN101142207A (zh) | 2008-03-12 |
IL185329A (en) | 2013-04-30 |
CA2601870A1 (en) | 2006-09-28 |
PL1858878T3 (pl) | 2012-09-28 |
EP1858878A1 (en) | 2007-11-28 |
CA2601870C (en) | 2013-06-11 |
IL185329A0 (en) | 2008-02-09 |
AU2006227484B2 (en) | 2011-08-11 |
BRPI0609844A2 (pt) | 2010-05-04 |
TW200700407A (en) | 2007-01-01 |
JP2008533169A (ja) | 2008-08-21 |
KR101337159B1 (ko) | 2013-12-05 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IL176547A0 (en) | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives having cb1-antagonistic activity | |
MXPA06010097A (es) | Inhibidores de dipeptidil peptidasa-iv. | |
IL185329A0 (en) | Conversion of 2-pyrazolines to pyrazoles using bromine | |
SG165380A1 (en) | Process for the production of amides | |
MX2009008858A (es) | Derivado de pirazolcarbonitrilo que contiene fluor y el metodo para producirlo y derivado del acido pirazolcarboxilico que contiene fluor obtenido utilizando el derivado de pirazolcarbonitrilo que contiene fluor y el método para producirlo. | |
NO20080738L (no) | Fremgangsmater for neurobeskyttelse | |
UA101835C2 (uk) | Спосіб отримання похідних 1-(2-галогенбіфеніл-4-іл)-циклопропанкарбонової кислоти | |
TW200612959A (en) | Method for preparing hydroxamic acids | |
IL185545A0 (en) | Method of preparation of pure 4-pyrrolidinophenylbenzyl ether derivatives as maob inhibitors | |
TW200619201A (en) | Process for the preparation of pyrazoles | |
TW200602331A (en) | Process for preparing thiazole compound | |
TW200700419A (en) | 5,6-dialkyl-7-aminoazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds | |
TW200740763A (en) | A method for preparing 5-hydroxy-1-alkyl pyrazole derivatives | |
MX2009013336A (es) | Sintesis de 3-aminopirazoles sustituidos. | |
WO2009008287A1 (ja) | 4-(トリクロロメチルチオ)アニリン類およびその製造方法、ならびに4-(トリフルオロメチルチオ)アニリン類の製造方法 | |
TW200700370A (en) | Producing method of haloalkylether compounds | |
TW200640856A (en) | Method for preparing enantiomerically pure 4-pyrrolidinophenylbenzylether derivatives | |
TW200730481A (en) | Process for preparing haloalkyl(thio)vinimidinium salts and 4-(haloalkyl(thio))-pyrazoles and their conversion to crop protection compositions | |
TW200631926A (en) | Process for the production of nitrobenzoles | |
MY145132A (en) | Conversion of 2-pyrazolines to pyrazoles using bromine | |
AU2001284755A1 (en) | Process for the preparation of alkyllithium compounds | |
UA84594C2 (en) | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists | |
TW200724523A (en) | The manufacturing method of prostaglandin F derivatives and the novel intermediates thereof | |
TH59387B (th) | อนุพันธ์ n-ไตรอะโซลอิลเมทธิล-พิเพอราซิน เป็น นิวโรไคนิน-รีเซปเตอร์แอนทาโกนิสท์ | |
DK1572615T3 (da) | Fremgangsmåde til syntese af peptider indeholdende en 4-hydroxyprolin-substruktur |