MXPA06010097A - Inhibidores de dipeptidil peptidasa-iv. - Google Patents

Inhibidores de dipeptidil peptidasa-iv.

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Publication number
MXPA06010097A
MXPA06010097A MXPA06010097A MXPA06010097A MXPA06010097A MX PA06010097 A MXPA06010097 A MX PA06010097A MX PA06010097 A MXPA06010097 A MX PA06010097A MX PA06010097 A MXPA06010097 A MX PA06010097A MX PA06010097 A MXPA06010097 A MX PA06010097A
Authority
MX
Mexico
Prior art keywords
dpp
inhibitors
compounds
relates
r3nh2
Prior art date
Application number
MXPA06010097A
Other languages
English (en)
Inventor
Achim Feurer
Paul John Edwards
Silvia Cerezo-Galvez
Victor Giulio Matassa
Sonja Nordhoff
Claudia Rosenbaum
Stephan Bulat
Original Assignee
Santhera Pharmaceuticals Ch
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Santhera Pharmaceuticals Ch filed Critical Santhera Pharmaceuticals Ch
Publication of MXPA06010097A publication Critical patent/MXPA06010097A/es

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/40—Acylated substituent nitrogen atom
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Abstract

La invencion se refiere a compuestos de la formula (I) Z-C(R1R2)-C(R3NH2)-C(R4R5)-X-N(R6R7) (I), en donde Z, R1-7 y X tienen significados como se citan en la descripcion y en las reivindicaciones; dichos compuestos son utiles como inhibidores DPP-IV; la invencion tambien se refiere a la preparacion de dichos compuestos asi como la produccion y uso de los mismos como medicamento.
MXPA06010097A 2004-03-05 2005-02-25 Inhibidores de dipeptidil peptidasa-iv. MXPA06010097A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04005347A EP1593671A1 (en) 2004-03-05 2004-03-05 DPP-IV inhibitors
PCT/EP2005/002010 WO2005095343A1 (en) 2004-03-05 2005-02-25 Dpp-iv inhibitors

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EP (2) EP1593671A1 (es)
JP (1) JP2007526267A (es)
KR (1) KR20070007816A (es)
CN (1) CN1980892A (es)
AU (1) AU2005229330B2 (es)
CA (1) CA2558446A1 (es)
MX (1) MXPA06010097A (es)
NO (1) NO20064032L (es)
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WO (1) WO2005095343A1 (es)

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CN116157389A (zh) 2020-08-03 2023-05-23 阿尔比里奥公司 苯并硫杂(二)氮杂环庚三烯化合物及其作为胆汁酸调节剂的用途
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CN116583504A (zh) 2020-12-04 2023-08-11 阿尔比里奥公司 苯并硫杂(二)氮杂环庚三烯化合物及其作为胆汁酸调节剂的用途

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WO2005095343A1 (en) 2005-10-13
EP1593671A1 (en) 2005-11-09
RU2006131597A (ru) 2008-04-10
AU2005229330B2 (en) 2008-12-18
US20070197522A1 (en) 2007-08-23
JP2007526267A (ja) 2007-09-13
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KR20070007816A (ko) 2007-01-16
RU2345067C2 (ru) 2009-01-27
CA2558446A1 (en) 2005-10-13

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