RO74431A - Procedeu pentru prepararea unor derivati ai kanamicinei 1-n-substituite - Google Patents

Procedeu pentru prepararea unor derivati ai kanamicinei 1-n-substituite

Info

Publication number
RO74431A
RO74431A RO7790001A RO9000177A RO74431A RO 74431 A RO74431 A RO 74431A RO 7790001 A RO7790001 A RO 7790001A RO 9000177 A RO9000177 A RO 9000177A RO 74431 A RO74431 A RO 74431A
Authority
RO
Romania
Prior art keywords
kanamicin
derivatives
substituted
preparation
substituted kanamicin
Prior art date
Application number
RO7790001A
Other languages
English (en)
French (fr)
Romanian (ro)
Inventor
William A Million
Kenneth Richardson
Original Assignee
Pfizer Corp,Pa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp,Pa filed Critical Pfizer Corp,Pa
Publication of RO74431A publication Critical patent/RO74431A/ro

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
RO7790001A 1976-04-14 1977-04-12 Procedeu pentru prepararea unor derivati ai kanamicinei 1-n-substituite RO74431A (ro)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB15421/76A GB1530201A (en) 1976-04-14 1976-04-14 Process for the preparation of aminoglycoside antibiotics and intermediates therefor

Publications (1)

Publication Number Publication Date
RO74431A true RO74431A (ro) 1981-08-30

Family

ID=10058845

Family Applications (2)

Application Number Title Priority Date Filing Date
RO7790001A RO74431A (ro) 1976-04-14 1977-04-12 Procedeu pentru prepararea unor derivati ai kanamicinei 1-n-substituite
RO77101733A RO79969A (ro) 1976-04-14 1977-04-12 Procedeu pentru prepararea unor derivati ai kanamicinei

Family Applications After (1)

Application Number Title Priority Date Filing Date
RO77101733A RO79969A (ro) 1976-04-14 1977-04-12 Procedeu pentru prepararea unor derivati ai kanamicinei

Country Status (28)

Country Link
JP (2) JPS52139044A (de)
AR (1) AR219074A1 (de)
AT (1) AT356267B (de)
AU (1) AU497416B2 (de)
BE (1) BE853564A (de)
BG (2) BG28072A4 (de)
CA (1) CA1083568A (de)
CH (1) CH622528A5 (de)
CS (1) CS202570B2 (de)
DD (2) DD130661A5 (de)
DE (1) DE2716533C3 (de)
DK (1) DK164277A (de)
EG (1) EG12909A (de)
ES (1) ES457793A1 (de)
FI (1) FI771144A (de)
FR (1) FR2348223A1 (de)
GB (1) GB1530201A (de)
GR (1) GR68936B (de)
IE (1) IE45030B1 (de)
IL (1) IL51775A (de)
LU (1) LU77108A1 (de)
NL (1) NL7703567A (de)
NZ (1) NZ183733A (de)
PH (1) PH14029A (de)
PL (2) PL112867B1 (de)
PT (1) PT66422B (de)
RO (2) RO74431A (de)
ZA (1) ZA771944B (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2924659A1 (de) * 1979-06-19 1981-01-22 Bayer Ag Pseudotrisaccharide, ihre herstellung und verwendung als arzneimittel
JPH0414628Y2 (de) * 1984-12-13 1992-04-02
JPS61191642U (de) * 1985-05-20 1986-11-28
IT1225484B (it) * 1987-11-27 1990-11-14 Pierrel Spa Procedimento di sintesi dell'amikacina
CN101481397B (zh) * 2009-01-23 2012-10-31 北京大学 一种新的卡那霉素a衍生物及其制备方法和用途
RU2591188C2 (ru) 2010-11-08 2016-07-10 Альбирео Аб Ингибиторы ibat для лечения заболеваний печени
CA2952406A1 (en) 2014-06-25 2015-12-30 Ea Pharma Co., Ltd. Solid formulation and method for preventing or reducing coloration thereof
CA2952405A1 (en) 2014-06-25 2015-12-30 Ea Pharma Co., Ltd. Solid formulation and method for stabilizing the same
EP3012252A1 (de) 2014-10-24 2016-04-27 Ferring BV Kristalline Form von elobixibat
US10441605B2 (en) 2016-02-09 2019-10-15 Albireo Ab Oral cholestyramine formulation and use thereof
US10441604B2 (en) 2016-02-09 2019-10-15 Albireo Ab Cholestyramine pellets and methods for preparation thereof
US10786529B2 (en) 2016-02-09 2020-09-29 Albireo Ab Oral cholestyramine formulation and use thereof
US11007142B2 (en) 2018-08-09 2021-05-18 Albireo Ab Oral cholestyramine formulation and use thereof
US10722457B2 (en) 2018-08-09 2020-07-28 Albireo Ab Oral cholestyramine formulation and use thereof

Also Published As

Publication number Publication date
EG12909A (en) 1979-12-31
ES457793A1 (es) 1978-08-01
RO79969A (ro) 1983-02-01
BG28072A4 (en) 1980-02-25
JPS5549587B2 (de) 1980-12-12
GB1530201A (en) 1978-10-25
JPS5421326B2 (de) 1979-07-30
DE2716533A1 (de) 1977-11-03
PH14029A (en) 1980-12-12
DE2716533B2 (de) 1981-04-30
AT356267B (de) 1980-04-25
NZ183733A (en) 1979-12-11
DD135496A5 (de) 1979-05-09
PL197372A1 (pl) 1979-06-18
DD130661A5 (de) 1978-04-19
IE45030L (en) 1977-10-14
ZA771944B (en) 1978-03-29
BE853564A (fr) 1977-10-13
IL51775A0 (en) 1977-05-31
PT66422B (en) 1978-09-18
IE45030B1 (en) 1982-06-02
NL7703567A (nl) 1977-10-18
LU77108A1 (de) 1979-01-18
DE2716533C3 (de) 1982-05-13
FR2348223A1 (fr) 1977-11-10
CH622528A5 (en) 1981-04-15
AU497416B2 (en) 1978-12-14
DK164277A (da) 1977-10-15
IL51775A (en) 1980-07-31
FI771144A (de) 1977-10-15
AU2372177A (en) 1978-10-05
PL112867B1 (en) 1980-11-29
JPS52139044A (en) 1977-11-19
PT66422A (en) 1977-05-01
GR68936B (de) 1982-03-29
CS202570B2 (en) 1981-01-30
RO79969B (ro) 1983-01-30
BG27759A3 (en) 1979-12-12
JPS535141A (en) 1978-01-18
CA1083568A (en) 1980-08-12
AR219074A1 (es) 1980-07-31
ATA261477A (de) 1979-09-15

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