IL51775A - Process and novel intermediates for the preparation of 1-n-substituted kanamycin derivatives - Google Patents

Process and novel intermediates for the preparation of 1-n-substituted kanamycin derivatives

Info

Publication number
IL51775A
IL51775A IL51775A IL5177577A IL51775A IL 51775 A IL51775 A IL 51775A IL 51775 A IL51775 A IL 51775A IL 5177577 A IL5177577 A IL 5177577A IL 51775 A IL51775 A IL 51775A
Authority
IL
Israel
Prior art keywords
preparation
novel intermediates
kanamycin derivatives
substituted
substituted kanamycin
Prior art date
Application number
IL51775A
Other languages
English (en)
Other versions
IL51775A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL51775A0 publication Critical patent/IL51775A0/xx
Publication of IL51775A publication Critical patent/IL51775A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL51775A 1976-04-14 1977-03-29 Process and novel intermediates for the preparation of 1-n-substituted kanamycin derivatives IL51775A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB15421/76A GB1530201A (en) 1976-04-14 1976-04-14 Process for the preparation of aminoglycoside antibiotics and intermediates therefor

Publications (2)

Publication Number Publication Date
IL51775A0 IL51775A0 (en) 1977-05-31
IL51775A true IL51775A (en) 1980-07-31

Family

ID=10058845

Family Applications (1)

Application Number Title Priority Date Filing Date
IL51775A IL51775A (en) 1976-04-14 1977-03-29 Process and novel intermediates for the preparation of 1-n-substituted kanamycin derivatives

Country Status (28)

Country Link
JP (2) JPS52139044A (de)
AR (1) AR219074A1 (de)
AT (1) AT356267B (de)
AU (1) AU497416B2 (de)
BE (1) BE853564A (de)
BG (2) BG27759A3 (de)
CA (1) CA1083568A (de)
CH (1) CH622528A5 (de)
CS (1) CS202570B2 (de)
DD (2) DD130661A5 (de)
DE (1) DE2716533C3 (de)
DK (1) DK164277A (de)
EG (1) EG12909A (de)
ES (1) ES457793A1 (de)
FI (1) FI771144A (de)
FR (1) FR2348223A1 (de)
GB (1) GB1530201A (de)
GR (1) GR68936B (de)
IE (1) IE45030B1 (de)
IL (1) IL51775A (de)
LU (1) LU77108A1 (de)
NL (1) NL7703567A (de)
NZ (1) NZ183733A (de)
PH (1) PH14029A (de)
PL (2) PL112867B1 (de)
PT (1) PT66422B (de)
RO (2) RO74431A (de)
ZA (1) ZA771944B (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2924659A1 (de) * 1979-06-19 1981-01-22 Bayer Ag Pseudotrisaccharide, ihre herstellung und verwendung als arzneimittel
JPH0414628Y2 (de) * 1984-12-13 1992-04-02
JPS61191642U (de) * 1985-05-20 1986-11-28
IT1225484B (it) * 1987-11-27 1990-11-14 Pierrel Spa Procedimento di sintesi dell'amikacina
CN101481397B (zh) * 2009-01-23 2012-10-31 北京大学 一种新的卡那霉素a衍生物及其制备方法和用途
RS60901B1 (sr) 2010-11-08 2020-11-30 Albireo Ab Ibat inhibitori za lečenje oboljenja jetre
CA2952405A1 (en) 2014-06-25 2015-12-30 Ea Pharma Co., Ltd. Solid formulation and method for stabilizing the same
CA2952406A1 (en) 2014-06-25 2015-12-30 Ea Pharma Co., Ltd. Solid formulation and method for preventing or reducing coloration thereof
EP3012252A1 (de) 2014-10-24 2016-04-27 Ferring BV Kristalline Form von elobixibat
US10786529B2 (en) 2016-02-09 2020-09-29 Albireo Ab Oral cholestyramine formulation and use thereof
US10441604B2 (en) 2016-02-09 2019-10-15 Albireo Ab Cholestyramine pellets and methods for preparation thereof
US10441605B2 (en) 2016-02-09 2019-10-15 Albireo Ab Oral cholestyramine formulation and use thereof
US11007142B2 (en) 2018-08-09 2021-05-18 Albireo Ab Oral cholestyramine formulation and use thereof
US10722457B2 (en) 2018-08-09 2020-07-28 Albireo Ab Oral cholestyramine formulation and use thereof

Also Published As

Publication number Publication date
ATA261477A (de) 1979-09-15
DD135496A5 (de) 1979-05-09
IE45030B1 (en) 1982-06-02
CH622528A5 (en) 1981-04-15
BG27759A3 (en) 1979-12-12
JPS5421326B2 (de) 1979-07-30
ZA771944B (en) 1978-03-29
IL51775A0 (en) 1977-05-31
JPS5549587B2 (de) 1980-12-12
PL197372A1 (pl) 1979-06-18
PT66422B (en) 1978-09-18
GB1530201A (en) 1978-10-25
BG28072A4 (en) 1980-02-25
PL112867B1 (en) 1980-11-29
EG12909A (en) 1979-12-31
PT66422A (en) 1977-05-01
JPS535141A (en) 1978-01-18
RO79969B (ro) 1983-01-30
RO74431A (ro) 1981-08-30
AU2372177A (en) 1978-10-05
BE853564A (fr) 1977-10-13
RO79969A (ro) 1983-02-01
AR219074A1 (es) 1980-07-31
GR68936B (de) 1982-03-29
DE2716533A1 (de) 1977-11-03
JPS52139044A (en) 1977-11-19
PH14029A (en) 1980-12-12
CS202570B2 (en) 1981-01-30
FR2348223A1 (fr) 1977-11-10
LU77108A1 (de) 1979-01-18
AT356267B (de) 1980-04-25
FI771144A (de) 1977-10-15
DE2716533B2 (de) 1981-04-30
NZ183733A (en) 1979-12-11
DK164277A (da) 1977-10-15
NL7703567A (nl) 1977-10-18
DD130661A5 (de) 1978-04-19
AU497416B2 (en) 1978-12-14
CA1083568A (en) 1980-08-12
DE2716533C3 (de) 1982-05-13
ES457793A1 (es) 1978-08-01
IE45030L (en) 1977-10-14

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