ES457793A1 - Procedimiento para preparar derivados 1-n-sustituidos de ca-namicina. - Google Patents

Procedimiento para preparar derivados 1-n-sustituidos de ca-namicina.

Info

Publication number
ES457793A1
ES457793A1 ES457793A ES457793A ES457793A1 ES 457793 A1 ES457793 A1 ES 457793A1 ES 457793 A ES457793 A ES 457793A ES 457793 A ES457793 A ES 457793A ES 457793 A1 ES457793 A1 ES 457793A1
Authority
ES
Spain
Prior art keywords
group
groups
formula
preparation
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES457793A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp
Original Assignee
Pfizer Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp filed Critical Pfizer Corp
Publication of ES457793A1 publication Critical patent/ES457793A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Procedimiento para preparar derivados 1-N-sustituidos de canamicina, de fórmula: ***1 (Ver fórmula 1) en la que R puede ser un grupo amino o hidroxilo y R1 puede ser un grupo alquilo inferior o un grupo alcanoilo alifático inferior, cualquiera de los cuales puede estar opcionalmente sustituido con grupos hidroxilo y/o amino.
ES457793A 1976-04-14 1977-04-14 Procedimiento para preparar derivados 1-n-sustituidos de ca-namicina. Expired ES457793A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB15421/76A GB1530201A (en) 1976-04-14 1976-04-14 Process for the preparation of aminoglycoside antibiotics and intermediates therefor

Publications (1)

Publication Number Publication Date
ES457793A1 true ES457793A1 (es) 1978-08-01

Family

ID=10058845

Family Applications (1)

Application Number Title Priority Date Filing Date
ES457793A Expired ES457793A1 (es) 1976-04-14 1977-04-14 Procedimiento para preparar derivados 1-n-sustituidos de ca-namicina.

Country Status (28)

Country Link
JP (2) JPS52139044A (es)
AR (1) AR219074A1 (es)
AT (1) AT356267B (es)
AU (1) AU497416B2 (es)
BE (1) BE853564A (es)
BG (2) BG27759A3 (es)
CA (1) CA1083568A (es)
CH (1) CH622528A5 (es)
CS (1) CS202570B2 (es)
DD (2) DD130661A5 (es)
DE (1) DE2716533C3 (es)
DK (1) DK164277A (es)
EG (1) EG12909A (es)
ES (1) ES457793A1 (es)
FI (1) FI771144A (es)
FR (1) FR2348223A1 (es)
GB (1) GB1530201A (es)
GR (1) GR68936B (es)
IE (1) IE45030B1 (es)
IL (1) IL51775A (es)
LU (1) LU77108A1 (es)
NL (1) NL7703567A (es)
NZ (1) NZ183733A (es)
PH (1) PH14029A (es)
PL (2) PL197372A1 (es)
PT (1) PT66422B (es)
RO (2) RO74431A (es)
ZA (1) ZA771944B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2924659A1 (de) * 1979-06-19 1981-01-22 Bayer Ag Pseudotrisaccharide, ihre herstellung und verwendung als arzneimittel
JPH0414628Y2 (es) * 1984-12-13 1992-04-02
JPS61191642U (es) * 1985-05-20 1986-11-28
IT1225484B (it) * 1987-11-27 1990-11-14 Pierrel Spa Procedimento di sintesi dell'amikacina
CN101481397B (zh) * 2009-01-23 2012-10-31 北京大学 一种新的卡那霉素a衍生物及其制备方法和用途
BR112013010157B1 (pt) 2010-11-08 2020-02-04 Albireo Ab iinibidores do ibat, seus usos, e composição e combinações farmacêuticas
JP6581082B2 (ja) 2014-06-25 2019-09-25 Ｅａファーマ株式会社 固形製剤及びその安定化方法
CN106659726A (zh) 2014-06-25 2017-05-10 Ea制药株式会社 固体制剂及其着色防止或着色减少方法
EP3012252A1 (en) 2014-10-24 2016-04-27 Ferring BV Crystal modifications of elobixibat
US10441605B2 (en) 2016-02-09 2019-10-15 Albireo Ab Oral cholestyramine formulation and use thereof
US10441604B2 (en) 2016-02-09 2019-10-15 Albireo Ab Cholestyramine pellets and methods for preparation thereof
US10786529B2 (en) 2016-02-09 2020-09-29 Albireo Ab Oral cholestyramine formulation and use thereof
US11007142B2 (en) 2018-08-09 2021-05-18 Albireo Ab Oral cholestyramine formulation and use thereof
US10722457B2 (en) 2018-08-09 2020-07-28 Albireo Ab Oral cholestyramine formulation and use thereof

Also Published As

Publication number Publication date
BG27759A3 (en) 1979-12-12
DE2716533A1 (de) 1977-11-03
GB1530201A (en) 1978-10-25
FR2348223A1 (fr) 1977-11-10
ATA261477A (de) 1979-09-15
AU497416B2 (en) 1978-12-14
AU2372177A (en) 1978-10-05
RO79969A (ro) 1983-02-01
ZA771944B (en) 1978-03-29
PT66422A (en) 1977-05-01
AT356267B (de) 1980-04-25
DE2716533B2 (de) 1981-04-30
IE45030B1 (en) 1982-06-02
DD135496A5 (de) 1979-05-09
JPS535141A (en) 1978-01-18
JPS52139044A (en) 1977-11-19
NL7703567A (nl) 1977-10-18
RO79969B (ro) 1983-01-30
NZ183733A (en) 1979-12-11
PL197372A1 (pl) 1979-06-18
BE853564A (fr) 1977-10-13
DD130661A5 (de) 1978-04-19
JPS5549587B2 (es) 1980-12-12
GR68936B (es) 1982-03-29
DK164277A (da) 1977-10-15
EG12909A (en) 1979-12-31
IL51775A (en) 1980-07-31
PL112867B1 (en) 1980-11-29
CS202570B2 (en) 1981-01-30
RO74431A (ro) 1981-08-30
FI771144A (es) 1977-10-15
DE2716533C3 (de) 1982-05-13
BG28072A4 (en) 1980-02-25
JPS5421326B2 (es) 1979-07-30
PH14029A (en) 1980-12-12
IL51775A0 (en) 1977-05-31
LU77108A1 (es) 1979-01-18
CA1083568A (en) 1980-08-12
AR219074A1 (es) 1980-07-31
PT66422B (en) 1978-09-18
CH622528A5 (en) 1981-04-15
IE45030L (en) 1977-10-14

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