AU497416B2 - Preparation of amino glcoside antibiotics and intermediates - Google Patents

Preparation of amino glcoside antibiotics and intermediates

Info

Publication number
AU497416B2
AU497416B2 AU23721/77A AU2372177A AU497416B2 AU 497416 B2 AU497416 B2 AU 497416B2 AU 23721/77 A AU23721/77 A AU 23721/77A AU 2372177 A AU2372177 A AU 2372177A AU 497416 B2 AU497416 B2 AU 497416B2
Authority
AU
Australia
Prior art keywords
glcoside
antibiotics
intermediates
amino
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
AU23721/77A
Other languages
English (en)
Other versions
AU2372177A (en
Inventor
Wa. Plews Rm. & Richardson K Million
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Corp
Original Assignee
Pfizer Corp
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp, Pfizer Inc filed Critical Pfizer Corp
Publication of AU2372177A publication Critical patent/AU2372177A/en
Application granted granted Critical
Publication of AU497416B2 publication Critical patent/AU497416B2/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU23721/77A 1976-04-14 1977-03-29 Preparation of amino glcoside antibiotics and intermediates Expired AU497416B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB15421/76A GB1530201A (en) 1976-04-14 1976-04-14 Process for the preparation of aminoglycoside antibiotics and intermediates therefor
GBGB15421/76 1976-04-14

Publications (2)

Publication Number Publication Date
AU2372177A AU2372177A (en) 1978-10-05
AU497416B2 true AU497416B2 (en) 1978-12-14

Family

ID=10058845

Family Applications (1)

Application Number Title Priority Date Filing Date
AU23721/77A Expired AU497416B2 (en) 1976-04-14 1977-03-29 Preparation of amino glcoside antibiotics and intermediates

Country Status (28)

Country Link
JP (2) JPS52139044A (es)
AR (1) AR219074A1 (es)
AT (1) AT356267B (es)
AU (1) AU497416B2 (es)
BE (1) BE853564A (es)
BG (2) BG27759A3 (es)
CA (1) CA1083568A (es)
CH (1) CH622528A5 (es)
CS (1) CS202570B2 (es)
DD (2) DD130661A5 (es)
DE (1) DE2716533C3 (es)
DK (1) DK164277A (es)
EG (1) EG12909A (es)
ES (1) ES457793A1 (es)
FI (1) FI771144A (es)
FR (1) FR2348223A1 (es)
GB (1) GB1530201A (es)
GR (1) GR68936B (es)
IE (1) IE45030B1 (es)
IL (1) IL51775A (es)
LU (1) LU77108A1 (es)
NL (1) NL7703567A (es)
NZ (1) NZ183733A (es)
PH (1) PH14029A (es)
PL (2) PL197372A1 (es)
PT (1) PT66422B (es)
RO (2) RO74431A (es)
ZA (1) ZA771944B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2924659A1 (de) * 1979-06-19 1981-01-22 Bayer Ag Pseudotrisaccharide, ihre herstellung und verwendung als arzneimittel
JPH0414628Y2 (es) * 1984-12-13 1992-04-02
JPS61191642U (es) * 1985-05-20 1986-11-28
IT1225484B (it) * 1987-11-27 1990-11-14 Pierrel Spa Procedimento di sintesi dell'amikacina
CN101481397B (zh) * 2009-01-23 2012-10-31 北京大学 一种新的卡那霉素a衍生物及其制备方法和用途
BR112013010157B1 (pt) 2010-11-08 2020-02-04 Albireo Ab iinibidores do ibat, seus usos, e composição e combinações farmacêuticas
JP6581082B2 (ja) 2014-06-25 2019-09-25 Ｅａファーマ株式会社 固形製剤及びその安定化方法
CN106659726A (zh) 2014-06-25 2017-05-10 Ea制药株式会社 固体制剂及其着色防止或着色减少方法
EP3012252A1 (en) 2014-10-24 2016-04-27 Ferring BV Crystal modifications of elobixibat
US10441605B2 (en) 2016-02-09 2019-10-15 Albireo Ab Oral cholestyramine formulation and use thereof
US10441604B2 (en) 2016-02-09 2019-10-15 Albireo Ab Cholestyramine pellets and methods for preparation thereof
US10786529B2 (en) 2016-02-09 2020-09-29 Albireo Ab Oral cholestyramine formulation and use thereof
US11007142B2 (en) 2018-08-09 2021-05-18 Albireo Ab Oral cholestyramine formulation and use thereof
US10722457B2 (en) 2018-08-09 2020-07-28 Albireo Ab Oral cholestyramine formulation and use thereof

Also Published As

Publication number Publication date
BG27759A3 (en) 1979-12-12
DE2716533A1 (de) 1977-11-03
GB1530201A (en) 1978-10-25
FR2348223A1 (fr) 1977-11-10
ES457793A1 (es) 1978-08-01
ATA261477A (de) 1979-09-15
AU2372177A (en) 1978-10-05
RO79969A (ro) 1983-02-01
ZA771944B (en) 1978-03-29
PT66422A (en) 1977-05-01
AT356267B (de) 1980-04-25
DE2716533B2 (de) 1981-04-30
IE45030B1 (en) 1982-06-02
DD135496A5 (de) 1979-05-09
JPS535141A (en) 1978-01-18
JPS52139044A (en) 1977-11-19
NL7703567A (nl) 1977-10-18
RO79969B (ro) 1983-01-30
NZ183733A (en) 1979-12-11
PL197372A1 (pl) 1979-06-18
BE853564A (fr) 1977-10-13
DD130661A5 (de) 1978-04-19
JPS5549587B2 (es) 1980-12-12
GR68936B (es) 1982-03-29
DK164277A (da) 1977-10-15
EG12909A (en) 1979-12-31
IL51775A (en) 1980-07-31
PL112867B1 (en) 1980-11-29
CS202570B2 (en) 1981-01-30
RO74431A (ro) 1981-08-30
FI771144A (es) 1977-10-15
DE2716533C3 (de) 1982-05-13
BG28072A4 (en) 1980-02-25
JPS5421326B2 (es) 1979-07-30
PH14029A (en) 1980-12-12
IL51775A0 (en) 1977-05-31
LU77108A1 (es) 1979-01-18
CA1083568A (en) 1980-08-12
AR219074A1 (es) 1980-07-31
PT66422B (en) 1978-09-18
CH622528A5 (en) 1981-04-15
IE45030L (en) 1977-10-14

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