RO74431A - PROCESS FOR THE PREPARATION OF 1-N-SUBSTITUTED KANAMICIN DERIVATIVES - Google Patents

PROCESS FOR THE PREPARATION OF 1-N-SUBSTITUTED KANAMICIN DERIVATIVES

Info

Publication number
RO74431A
RO74431A RO7790001A RO9000177A RO74431A RO 74431 A RO74431 A RO 74431A RO 7790001 A RO7790001 A RO 7790001A RO 9000177 A RO9000177 A RO 9000177A RO 74431 A RO74431 A RO 74431A
Authority
RO
Romania
Prior art keywords
kanamicin
derivatives
substituted
preparation
substituted kanamicin
Prior art date
Application number
RO7790001A
Other languages
French (fr)
Romanian (ro)
Inventor
William A Million
Kenneth Richardson
Original Assignee
Pfizer Corp,Pa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Corp,Pa filed Critical Pfizer Corp,Pa
Publication of RO74431A publication Critical patent/RO74431A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
RO7790001A 1976-04-14 1977-04-12 PROCESS FOR THE PREPARATION OF 1-N-SUBSTITUTED KANAMICIN DERIVATIVES RO74431A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB15421/76A GB1530201A (en) 1976-04-14 1976-04-14 Process for the preparation of aminoglycoside antibiotics and intermediates therefor

Publications (1)

Publication Number Publication Date
RO74431A true RO74431A (en) 1981-08-30

Family

ID=10058845

Family Applications (2)

Application Number Title Priority Date Filing Date
RO7790001A RO74431A (en) 1976-04-14 1977-04-12 PROCESS FOR THE PREPARATION OF 1-N-SUBSTITUTED KANAMICIN DERIVATIVES
RO77101733A RO79969A (en) 1976-04-14 1977-04-12 PROCESS FOR THE PREPARATION OF KANAMICINE DERIVATIVES

Family Applications After (1)

Application Number Title Priority Date Filing Date
RO77101733A RO79969A (en) 1976-04-14 1977-04-12 PROCESS FOR THE PREPARATION OF KANAMICINE DERIVATIVES

Country Status (28)

Country Link
JP (2) JPS52139044A (en)
AR (1) AR219074A1 (en)
AT (1) AT356267B (en)
AU (1) AU497416B2 (en)
BE (1) BE853564A (en)
BG (2) BG27759A3 (en)
CA (1) CA1083568A (en)
CH (1) CH622528A5 (en)
CS (1) CS202570B2 (en)
DD (2) DD130661A5 (en)
DE (1) DE2716533C3 (en)
DK (1) DK164277A (en)
EG (1) EG12909A (en)
ES (1) ES457793A1 (en)
FI (1) FI771144A (en)
FR (1) FR2348223A1 (en)
GB (1) GB1530201A (en)
GR (1) GR68936B (en)
IE (1) IE45030B1 (en)
IL (1) IL51775A (en)
LU (1) LU77108A1 (en)
NL (1) NL7703567A (en)
NZ (1) NZ183733A (en)
PH (1) PH14029A (en)
PL (2) PL112867B1 (en)
PT (1) PT66422B (en)
RO (2) RO74431A (en)
ZA (1) ZA771944B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2924659A1 (en) * 1979-06-19 1981-01-22 Bayer Ag PSEUDOTRISACCHARIDE, THEIR PRODUCTION AND USE AS A MEDICINAL PRODUCT
JPH0414628Y2 (en) * 1984-12-13 1992-04-02
JPS61191642U (en) * 1985-05-20 1986-11-28
IT1225484B (en) * 1987-11-27 1990-11-14 Pierrel Spa SYNTHESIS PROCEDURE OF AMIKACINA
CN101481397B (en) * 2009-01-23 2012-10-31 北京大学 Novel kanamycin A derivative, and preparation and use thereof
SG190029A1 (en) 2010-11-08 2013-06-28 Albireo Ab Ibat inhibitors for the treatment of liver diseases
CA2952405A1 (en) 2014-06-25 2015-12-30 Ea Pharma Co., Ltd. Solid formulation and method for stabilizing the same
WO2015199147A1 (en) 2014-06-25 2015-12-30 味の素株式会社 Solid preparation, and method for preventing or reducing discoloration thereof
EP3012252A1 (en) 2014-10-24 2016-04-27 Ferring BV Crystal modifications of elobixibat
US10441604B2 (en) 2016-02-09 2019-10-15 Albireo Ab Cholestyramine pellets and methods for preparation thereof
US10441605B2 (en) 2016-02-09 2019-10-15 Albireo Ab Oral cholestyramine formulation and use thereof
US10786529B2 (en) 2016-02-09 2020-09-29 Albireo Ab Oral cholestyramine formulation and use thereof
US10722457B2 (en) 2018-08-09 2020-07-28 Albireo Ab Oral cholestyramine formulation and use thereof
US11007142B2 (en) 2018-08-09 2021-05-18 Albireo Ab Oral cholestyramine formulation and use thereof

Also Published As

Publication number Publication date
GB1530201A (en) 1978-10-25
BG28072A4 (en) 1980-02-25
NL7703567A (en) 1977-10-18
PT66422A (en) 1977-05-01
DD135496A5 (en) 1979-05-09
NZ183733A (en) 1979-12-11
AR219074A1 (en) 1980-07-31
ATA261477A (en) 1979-09-15
PH14029A (en) 1980-12-12
DE2716533C3 (en) 1982-05-13
RO79969B (en) 1983-01-30
DK164277A (en) 1977-10-15
RO79969A (en) 1983-02-01
CH622528A5 (en) 1981-04-15
PT66422B (en) 1978-09-18
JPS535141A (en) 1978-01-18
CS202570B2 (en) 1981-01-30
GR68936B (en) 1982-03-29
JPS52139044A (en) 1977-11-19
DE2716533B2 (en) 1981-04-30
AU2372177A (en) 1978-10-05
PL197372A1 (en) 1979-06-18
JPS5421326B2 (en) 1979-07-30
IE45030B1 (en) 1982-06-02
FR2348223A1 (en) 1977-11-10
JPS5549587B2 (en) 1980-12-12
EG12909A (en) 1979-12-31
FI771144A (en) 1977-10-15
ES457793A1 (en) 1978-08-01
AT356267B (en) 1980-04-25
DD130661A5 (en) 1978-04-19
IL51775A (en) 1980-07-31
BG27759A3 (en) 1979-12-12
AU497416B2 (en) 1978-12-14
IE45030L (en) 1977-10-14
LU77108A1 (en) 1979-01-18
CA1083568A (en) 1980-08-12
BE853564A (en) 1977-10-13
ZA771944B (en) 1978-03-29
IL51775A0 (en) 1977-05-31
DE2716533A1 (en) 1977-11-03
PL112867B1 (en) 1980-11-29

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