RO63003A - Procede pour la preparation des n-(heteroarylmethyl)-deltaen hauf-desoxynomorphines et des norcodeines - Google Patents

Procede pour la preparation des n-(heteroarylmethyl)-deltaen hauf-desoxynomorphines et des norcodeines

Info

Publication number
RO63003A
RO63003A RO7300076068A RO7606873A RO63003A RO 63003 A RO63003 A RO 63003A RO 7300076068 A RO7300076068 A RO 7300076068A RO 7606873 A RO7606873 A RO 7606873A RO 63003 A RO63003 A RO 63003A
Authority
RO
Romania
Prior art keywords
norcodeins
desoxynomorphines
deltaen
hauf
heteroarylmethyl
Prior art date
Application number
RO7300076068A
Other languages
English (en)
French (fr)
Romanian (ro)
Inventor
Gerhard Walther
Herbert Merz
Adolf Langbein
Klaus Stockhaus
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of RO63003A publication Critical patent/RO63003A/ro

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Emergency Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Networks Using Active Elements (AREA)
RO7300076068A 1972-09-14 1973-09-13 Procede pour la preparation des n-(heteroarylmethyl)-deltaen hauf-desoxynomorphines et des norcodeines RO63003A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2245141A DE2245141A1 (de) 1972-09-14 1972-09-14 Neue n-(heteroarylmethyl)-desoxynormorphine und -norcodeine, deren saeureadditionssalze, verfahren zu deren herstellung sowie deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
RO63003A true RO63003A (fr) 1978-05-15

Family

ID=5856355

Family Applications (2)

Application Number Title Priority Date Filing Date
RO7300076068A RO63003A (fr) 1972-09-14 1973-09-13 Procede pour la preparation des n-(heteroarylmethyl)-deltaen hauf-desoxynomorphines et des norcodeines
RO7382817A RO70193A (ro) 1972-09-14 1973-09-13 Procedeu pentru prepararea n-(heteroaril-metil)-delta 7-dezoxinormorfine si-norcodiene

Family Applications After (1)

Application Number Title Priority Date Filing Date
RO7382817A RO70193A (ro) 1972-09-14 1973-09-13 Procedeu pentru prepararea n-(heteroaril-metil)-delta 7-dezoxinormorfine si-norcodiene

Country Status (24)

Country Link
US (1) US3928359A (US06371994-20020416-C00029.png)
JP (1) JPS4966700A (US06371994-20020416-C00029.png)
AT (1) AT326281B (US06371994-20020416-C00029.png)
BE (1) BE804836A (US06371994-20020416-C00029.png)
BG (7) BG21228A3 (US06371994-20020416-C00029.png)
CH (7) CH605958A5 (US06371994-20020416-C00029.png)
CS (8) CS168679B2 (US06371994-20020416-C00029.png)
DD (1) DD109384A5 (US06371994-20020416-C00029.png)
DE (1) DE2245141A1 (US06371994-20020416-C00029.png)
ES (8) ES418563A1 (US06371994-20020416-C00029.png)
FI (1) FI55512C (US06371994-20020416-C00029.png)
FR (1) FR2199982B1 (US06371994-20020416-C00029.png)
GB (1) GB1449222A (US06371994-20020416-C00029.png)
HU (1) HU166367B (US06371994-20020416-C00029.png)
IE (1) IE38320B1 (US06371994-20020416-C00029.png)
IL (1) IL43216A (US06371994-20020416-C00029.png)
NL (1) NL7312621A (US06371994-20020416-C00029.png)
NO (1) NO139482C (US06371994-20020416-C00029.png)
PL (8) PL91807B1 (US06371994-20020416-C00029.png)
RO (2) RO63003A (US06371994-20020416-C00029.png)
SE (1) SE413510B (US06371994-20020416-C00029.png)
SU (8) SU498911A3 (US06371994-20020416-C00029.png)
YU (2) YU243973A (US06371994-20020416-C00029.png)
ZA (1) ZA737289B (US06371994-20020416-C00029.png)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4236008A (en) * 1978-09-19 1980-11-25 E. I. Du Pont De Nemours And Company Fluorination of precursors for fluorine analogs of hydrocodone and oxycodone
US4241065A (en) * 1979-07-02 1980-12-23 E. I. Du Pont De Nemours And Company Fluoro analogs of hydrocodone and oxycodone useful as analgesics, narcotic antagonists or both
JP2002501923A (ja) 1998-01-29 2002-01-22 モナシュ ユニバーシティ 治療用化合物

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2107989A1 (de) * 1971-02-19 1972-09-07 Boehringer Sohn Ingelheim N-(Furyl-methy])-morphinane, deren Säureadditionssalze sowie Verfahren zu deren Herstellung

Also Published As

Publication number Publication date
NO139482B (no) 1978-12-11
SU506299A3 (ru) 1976-03-05
BG21225A3 (US06371994-20020416-C00029.png) 1976-03-20
JPS4966700A (US06371994-20020416-C00029.png) 1974-06-27
GB1449222A (en) 1976-09-15
PL91807B1 (US06371994-20020416-C00029.png) 1977-03-31
ES430200A1 (es) 1976-10-16
CH590287A5 (US06371994-20020416-C00029.png) 1977-07-29
HU166367B (US06371994-20020416-C00029.png) 1975-03-28
ES430201A1 (es) 1976-10-16
IE38320L (en) 1974-03-14
BG21224A3 (US06371994-20020416-C00029.png) 1976-03-20
YU243973A (en) 1982-05-31
BE804836A (fr) 1974-03-13
FR2199982A1 (US06371994-20020416-C00029.png) 1974-04-19
PL87721B1 (US06371994-20020416-C00029.png) 1976-07-31
PL90720B1 (US06371994-20020416-C00029.png) 1977-01-31
IL43216A (en) 1976-07-30
BG21230A3 (US06371994-20020416-C00029.png) 1976-03-20
IL43216A0 (en) 1973-11-28
ES430202A1 (es) 1976-10-16
PL91836B1 (US06371994-20020416-C00029.png) 1977-03-31
BG21227A3 (US06371994-20020416-C00029.png) 1976-03-20
ES430197A1 (es) 1976-10-16
AU6030173A (en) 1975-03-13
PL91809B1 (US06371994-20020416-C00029.png) 1977-03-31
SU509239A3 (ru) 1976-03-30
BG21229A3 (US06371994-20020416-C00029.png) 1976-03-20
BG21228A3 (US06371994-20020416-C00029.png) 1976-03-20
CH591491A5 (US06371994-20020416-C00029.png) 1977-09-30
DE2245141A1 (de) 1974-03-21
NO139482C (no) 1979-03-21
SU498911A3 (ru) 1976-01-05
SU503523A3 (ru) 1976-02-15
CS168674B2 (US06371994-20020416-C00029.png) 1976-06-29
CH589088A5 (US06371994-20020416-C00029.png) 1977-06-30
CS168680B2 (US06371994-20020416-C00029.png) 1976-06-29
CH589089A5 (US06371994-20020416-C00029.png) 1977-06-30
CH605958A5 (US06371994-20020416-C00029.png) 1978-10-13
CH589090A5 (US06371994-20020416-C00029.png) 1977-06-30
RO70193A (ro) 1981-04-30
CH591490A5 (US06371994-20020416-C00029.png) 1977-09-30
SU505366A3 (ru) 1976-02-28
YU254879A (en) 1983-01-21
ES430199A1 (es) 1976-10-16
ES430203A1 (es) 1976-10-16
AT326281B (de) 1975-12-10
SE413510B (sv) 1980-06-02
CS168679B2 (US06371994-20020416-C00029.png) 1976-06-29
ES418563A1 (es) 1976-05-01
CS168678B2 (US06371994-20020416-C00029.png) 1976-06-29
ZA737289B (en) 1975-05-28
CS168676B2 (US06371994-20020416-C00029.png) 1976-06-29
PL91808B1 (US06371994-20020416-C00029.png) 1977-03-31
FR2199982B1 (US06371994-20020416-C00029.png) 1977-01-28
CS168677B2 (US06371994-20020416-C00029.png) 1976-06-29
IE38320B1 (en) 1978-02-15
SU503524A3 (ru) 1976-02-15
CS168673B2 (US06371994-20020416-C00029.png) 1976-06-29
SU520049A3 (ru) 1976-06-30
NL7312621A (US06371994-20020416-C00029.png) 1974-03-18
CS168675B2 (US06371994-20020416-C00029.png) 1976-06-29
DD109384A5 (US06371994-20020416-C00029.png) 1974-11-05
FI55512C (fi) 1979-08-10
BG21412A3 (US06371994-20020416-C00029.png) 1976-05-20
PL91837B1 (US06371994-20020416-C00029.png) 1977-03-31
US3928359A (en) 1975-12-23
PL91829B1 (US06371994-20020416-C00029.png) 1977-03-31
ATA761673A (de) 1975-02-15
ES430198A1 (es) 1976-10-16
SU528878A3 (ru) 1976-09-15
FI55512B (fi) 1979-04-30

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