PT95652A - Processo para a preparacao de derivados de amino-piridinil-amino-fenois e de composicoes farmaceuticas que os contem - Google Patents
Processo para a preparacao de derivados de amino-piridinil-amino-fenois e de composicoes farmaceuticas que os contem Download PDFInfo
- Publication number
- PT95652A PT95652A PT95652A PT9565290A PT95652A PT 95652 A PT95652 A PT 95652A PT 95652 A PT95652 A PT 95652A PT 9565290 A PT9565290 A PT 9565290A PT 95652 A PT95652 A PT 95652A
- Authority
- PT
- Portugal
- Prior art keywords
- compound
- formula
- amino
- hydrogen
- lower alkyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/36—Radicals substituted by singly-bound nitrogen atoms
- C07D213/42—Radicals substituted by singly-bound nitrogen atoms having hetero atoms attached to the substituent nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Pyridine Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/425,713 US4959378A (en) | 1989-10-24 | 1989-10-24 | Aminopyridinylaminophenol compounds useful as topical antiinflammatory agents for the treatment of skin disorders |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT95652A true PT95652A (pt) | 1991-09-13 |
Family
ID=23687726
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT95652A PT95652A (pt) | 1989-10-24 | 1990-10-23 | Processo para a preparacao de derivados de amino-piridinil-amino-fenois e de composicoes farmaceuticas que os contem |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4959378A (ref) |
| EP (1) | EP0424848A3 (ref) |
| JP (1) | JPH03151364A (ref) |
| KR (1) | KR910007881A (ref) |
| AU (1) | AU6485790A (ref) |
| CA (1) | CA2028285A1 (ref) |
| FI (1) | FI905192A7 (ref) |
| IE (1) | IE903809A1 (ref) |
| IL (1) | IL96082A0 (ref) |
| NO (1) | NO904576L (ref) |
| PT (1) | PT95652A (ref) |
| ZA (1) | ZA908459B (ref) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1990009985A1 (en) * | 1989-02-23 | 1990-09-07 | Otsuka Pharmaceutical Factory, Inc. | p-AMINOPHENOL DERIVATIVE AND PRODUCTION AND APPLICATION THEREOF |
| US4959378A (en) * | 1989-10-24 | 1990-09-25 | Hoechst-Roussel Pharmaceuticals Inc. | Aminopyridinylaminophenol compounds useful as topical antiinflammatory agents for the treatment of skin disorders |
| US6022884A (en) * | 1997-11-07 | 2000-02-08 | Amgen Inc. | Substituted pyridine compounds and methods of use |
| US6455554B1 (en) | 1999-06-07 | 2002-09-24 | Targacept, Inc. | Oxopyridinyl pharmaceutical compositions and methods for use |
| JP4202250B2 (ja) | 2001-07-25 | 2008-12-24 | バイオマリン ファーマシューティカル インコーポレイテッド | 血液脳関門輸送を調節するための組成物および方法 |
| MX2007004781A (es) * | 2004-10-20 | 2007-05-11 | Applied Research Systems | Derivados de 3-arilamino piridina. |
| EP2671507A3 (en) | 2005-04-28 | 2014-02-19 | Proteus Digital Health, Inc. | Pharma-informatics system |
| MX2009002893A (es) | 2006-09-18 | 2009-07-10 | Raptor Pharmaceutical Inc | Tratamiento de trastornos hepaticos mediante la administracion de conjugados de la proteina asociada al receptor (rap). |
| CA2752373C (en) | 2009-02-20 | 2017-10-10 | To-Bbb Holding B.V. | Glutathione-based drug delivery system |
| IL255113B (en) | 2009-05-06 | 2022-09-01 | Laboratory Skin Care Inc | Dermal delivery compositions comprising active agent-calcium phosphate particle complexes and methods of using the same |
| US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB750925A (en) * | 1953-10-26 | 1956-06-20 | Wellcome Found | Improvements in and relating to pyridine derivatives and the manufacture thereof |
| US3118884A (en) * | 1959-10-19 | 1964-01-21 | Schering Corp | Derivatives of 3-azaphenothiazine and 3-azaphenoxazine |
| DE1795499A1 (de) * | 1964-08-29 | 1972-02-10 | Degussa | Neue substituierte Diaminopyridine |
| DE1795544A1 (de) * | 1964-08-29 | 1973-02-15 | Degussa | Verfahren zur herstellung von phenylamino-pyridinen |
| DE1568426A1 (de) * | 1966-11-16 | 1970-04-02 | Degussa | Verfahren zur Herstellung von neuen N-aromatisch substituierten Saeureamiden |
| FR8363M (ref) * | 1967-02-01 | 1971-02-15 | ||
| US3495969A (en) * | 1967-09-25 | 1970-02-17 | Mobil Oil Corp | Substituted nitropyridines as herbicides |
| US3576616A (en) * | 1969-05-15 | 1971-04-27 | Monsanto Co | Herbicidal compositions and methods |
| US3721676A (en) * | 1969-11-12 | 1973-03-20 | Merck & Co Inc | Certain 3-amino-2(1h)pyridones |
| GB2073736B (en) * | 1979-10-03 | 1984-02-01 | Ici Ltd | Process for preparing pyridinyloxyphenoxy compounds and derivatives thereof |
| IE56702B1 (en) * | 1982-12-01 | 1991-11-06 | Usv Pharma Corp | Antiinflammatory antiallergic compounds |
| US4959378A (en) * | 1989-10-24 | 1990-09-25 | Hoechst-Roussel Pharmaceuticals Inc. | Aminopyridinylaminophenol compounds useful as topical antiinflammatory agents for the treatment of skin disorders |
-
1989
- 1989-10-24 US US07/425,713 patent/US4959378A/en not_active Expired - Lifetime
-
1990
- 1990-10-22 EP EP19900120237 patent/EP0424848A3/en not_active Withdrawn
- 1990-10-22 FI FI905192A patent/FI905192A7/fi not_active Application Discontinuation
- 1990-10-22 KR KR1019900016854A patent/KR910007881A/ko not_active Withdrawn
- 1990-10-22 IL IL96082A patent/IL96082A0/xx unknown
- 1990-10-23 CA CA002028285A patent/CA2028285A1/en not_active Abandoned
- 1990-10-23 ZA ZA908459A patent/ZA908459B/xx unknown
- 1990-10-23 JP JP2283579A patent/JPH03151364A/ja active Pending
- 1990-10-23 IE IE380990A patent/IE903809A1/en unknown
- 1990-10-23 NO NO90904576A patent/NO904576L/no unknown
- 1990-10-23 PT PT95652A patent/PT95652A/pt not_active Application Discontinuation
- 1990-10-23 AU AU64857/90A patent/AU6485790A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| IE903809A1 (en) | 1991-04-24 |
| US4959378B1 (ref) | 1993-08-10 |
| IL96082A0 (en) | 1991-07-18 |
| NO904576D0 (no) | 1990-10-23 |
| CA2028285A1 (en) | 1991-04-25 |
| FI905192A7 (fi) | 1991-04-25 |
| ZA908459B (en) | 1991-08-28 |
| JPH03151364A (ja) | 1991-06-27 |
| EP0424848A3 (en) | 1991-10-02 |
| US4959378A (en) | 1990-09-25 |
| FI905192A0 (fi) | 1990-10-22 |
| EP0424848A2 (en) | 1991-05-02 |
| AU6485790A (en) | 1991-05-02 |
| KR910007881A (ko) | 1991-05-30 |
| NO904576L (no) | 1991-04-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB1A | Laying open of patent application |
Effective date: 19910402 |
|
| FC3A | Refusal |
Effective date: 19961015 |