PT93782A - Processo para a preparacao de derivados de isotiazol-piridona azetidinil-substituidos e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados de isotiazol-piridona azetidinil-substituidos e de composicoes farmaceuticas que os contem Download PDF

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Publication number
PT93782A
PT93782A PT93782A PT9378290A PT93782A PT 93782 A PT93782 A PT 93782A PT 93782 A PT93782 A PT 93782A PT 9378290 A PT9378290 A PT 9378290A PT 93782 A PT93782 A PT 93782A
Authority
PT
Portugal
Prior art keywords
quot
cyclopropyl
dione
azetidinyl
quinoline
Prior art date
Application number
PT93782A
Other languages
English (en)
Portuguese (pt)
Inventor
Jordi Frigola-Constansa
Juan Pares-Corominas
Augusto Colombo-Pinol
Original Assignee
Esteve Labor Dr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr
Publication of PT93782A publication Critical patent/PT93782A/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT93782A 1989-04-18 1990-04-17 Processo para a preparacao de derivados de isotiazol-piridona azetidinil-substituidos e de composicoes farmaceuticas que os contem PT93782A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8905129A FR2645862B1 (fr) 1989-04-18 1989-04-18 Derives d'isothiazolo-pyrydone azetidinyl substitues, leur preparation et leur application en tant que medicaments

Publications (1)

Publication Number Publication Date
PT93782A true PT93782A (pt) 1990-11-20

Family

ID=9380854

Family Applications (1)

Application Number Title Priority Date Filing Date
PT93782A PT93782A (pt) 1989-04-18 1990-04-17 Processo para a preparacao de derivados de isotiazol-piridona azetidinil-substituidos e de composicoes farmaceuticas que os contem

Country Status (15)

Country Link
US (1) US5087621A (xx)
EP (1) EP0394120A1 (xx)
JP (1) JPH0730088B2 (xx)
KR (1) KR940006636B1 (xx)
AU (1) AU629630B2 (xx)
CA (1) CA2014673A1 (xx)
DD (1) DD298402A5 (xx)
ES (1) ES2021515A6 (xx)
FR (1) FR2645862B1 (xx)
HU (1) HU204056B (xx)
NO (1) NO901690L (xx)
PT (1) PT93782A (xx)
RU (1) RU2041226C1 (xx)
YU (1) YU70390A (xx)
ZA (1) ZA902866B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2676445B1 (fr) * 1991-05-16 1995-02-03 Esteve Labor Dr Derives de pyridone amino acide azetidinyl substitues, leur preparation et leur application en tant que medicaments.
US5556861A (en) * 1991-10-01 1996-09-17 Laboratoire Roger Bellon 1,8 benzonaphthyridine derivatives and antimicrobial compositions
US5885983A (en) * 1996-05-10 1999-03-23 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
WO2000063168A1 (en) * 1999-04-16 2000-10-26 Coelacanth Chemical Corporation Synthesis of azetidine derivatives
WO2006118605A2 (en) * 2004-11-11 2006-11-09 Achillion Pharmaceuticals, Inc. 8a, 9-dihydro-4a-h-isothiazolo[5,4-b] quinoline-3, 4-diones and related compounds as anti-infective agents
WO2006074317A1 (en) * 2005-01-05 2006-07-13 Achillion Pharmaceuticals, Inc. 1-thia-2,4a-diaza-cyclopenta[b]naphthalene-3,4-diones and related compounds as anti-infective agents
US7199128B2 (en) * 2005-02-02 2007-04-03 Achillion Pharmaceuticals, Inc. 8-N-substituted-2H-isothiazolo[5,4-b]quinolizine-3,4-diones and related compounds as antiinfective agents
EP1913004B1 (en) 2005-07-27 2010-09-22 Achillion Pharmaceuticals, Inc. 8-methoxy-9h-isothiazolo[5,4-b]quinoline-3,4-diones and related compounds as anti-infective agents
EA201101451A1 (ru) * 2009-04-03 2012-03-30 Ачиллион Фармасьютикалз, Инк. Гидрокситиенохинолоны и родственные соединения как противоинфекционные средства

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4767762A (en) * 1985-12-23 1988-08-30 Abbott Laboratories Tricyclic quinoline and naphthyride antibacterials
US4687770A (en) * 1985-12-23 1987-08-18 Abbott Laboratories Isoxazolo-pyrido-benzoxazine and isothiazolo-pyrido-benzoxazine derivatives
DE3701665A1 (de) * 1987-01-19 1988-07-28 Schering Ag Polymer-komplexe, verfahren zu deren herstellung und diese enthaltende pharmazeutische mittel
IL89351A0 (en) * 1988-03-14 1989-09-10 Lundbeck & Co As H 4,5,6,7-tetrahydroisothiazolo(4,5-c)pyridines,process for their preparation and pharmaceutical compositions containing them
JPH0265092A (ja) * 1988-08-29 1990-03-05 Nec Corp 薄膜el素子の製造方法

Also Published As

Publication number Publication date
FR2645862A1 (fr) 1990-10-19
RU2041226C1 (ru) 1995-08-09
FR2645862B1 (fr) 1991-07-12
DD298402A5 (de) 1992-02-20
ES2021515A6 (es) 1991-11-01
NO901690D0 (no) 1990-04-17
US5087621A (en) 1992-02-11
NO901690L (no) 1990-10-19
YU70390A (en) 1992-05-28
HU204056B (en) 1991-11-28
KR900016227A (ko) 1990-11-13
HU902460D0 (en) 1990-08-28
AU629630B2 (en) 1992-10-08
EP0394120A1 (fr) 1990-10-24
HUT54377A (en) 1991-02-28
JPH02292289A (ja) 1990-12-03
ZA902866B (en) 1991-02-27
JPH0730088B2 (ja) 1995-04-05
CA2014673A1 (fr) 1990-10-18
AU5360890A (en) 1990-10-25
KR940006636B1 (ko) 1994-07-23

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Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19960201