PT820284E - Derivados de ureido biologicamente activos uteis no tratamento de esclerose multipla - Google Patents

Derivados de ureido biologicamente activos uteis no tratamento de esclerose multipla Download PDF

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Publication number
PT820284E
PT820284E PT97904356T PT97904356T PT820284E PT 820284 E PT820284 E PT 820284E PT 97904356 T PT97904356 T PT 97904356T PT 97904356 T PT97904356 T PT 97904356T PT 820284 E PT820284 E PT 820284E
Authority
PT
Portugal
Prior art keywords
methyl
bis
carbonyl
sulfonic acid
imino
Prior art date
Application number
PT97904356T
Other languages
English (en)
Portuguese (pt)
Inventor
Nicola Mongelli
Rachele Alzani
Elena Cozzi
Andrea Lombardi Borgia
Massimo Temponi
Francesco Colotta
Original Assignee
Pharmacia & Upjohn Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Spa filed Critical Pharmacia & Upjohn Spa
Publication of PT820284E publication Critical patent/PT820284E/pt

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
PT97904356T 1996-02-09 1997-01-24 Derivados de ureido biologicamente activos uteis no tratamento de esclerose multipla PT820284E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9602721.4A GB9602721D0 (en) 1996-02-09 1996-02-09 Biologically active ureido derivatives useful in the treatment of multiple sclerosis

Publications (1)

Publication Number Publication Date
PT820284E true PT820284E (pt) 2000-07-31

Family

ID=10788461

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97904356T PT820284E (pt) 1996-02-09 1997-01-24 Derivados de ureido biologicamente activos uteis no tratamento de esclerose multipla

Country Status (22)

Country Link
US (1) US5859046A (ko)
EP (1) EP0820284B1 (ko)
JP (1) JPH11504041A (ko)
KR (1) KR19980703718A (ko)
AR (1) AR005724A1 (ko)
AT (1) ATE189388T1 (ko)
AU (1) AU1720097A (ko)
BR (1) BR9702075A (ko)
CA (1) CA2217008A1 (ko)
DE (1) DE69701243T2 (ko)
DK (1) DK0820284T3 (ko)
EA (1) EA000166B1 (ko)
ES (1) ES2144844T3 (ko)
GB (1) GB9602721D0 (ko)
GR (1) GR3033332T3 (ko)
HU (1) HUP9900796A2 (ko)
IL (1) IL121808A0 (ko)
NO (1) NO974651L (ko)
PL (1) PL322717A1 (ko)
PT (1) PT820284E (ko)
WO (1) WO1997028796A1 (ko)
ZA (1) ZA97902B (ko)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999027939A1 (en) * 1997-12-04 1999-06-10 The Government Of The United States Of America, Represented By The Secretary, Department Of Health And Human Services Ureido derivatives of poly-4-amino-2-carboxy-1-methyl pyrrole compounds for inhibition of inflammation
GB9727524D0 (en) 1997-12-31 1998-02-25 Pharmacia & Upjohn Spa Synergistic antitumor composition containing a biologically active ureido compound
US6348464B1 (en) 1999-11-12 2002-02-19 Guilford Pharmaceuticals, Inc. Pyrrolecarbonylimino derivatives as naaladase inhibitors
DK1599461T3 (da) 2003-03-03 2009-08-17 Eisai Corp North America Thiolactoner som NAALADase-inhibitorer
EP3381897A1 (en) 2017-03-27 2018-10-03 Leadiant Biosciences SA Derivatives of the disodium 2,2'-{carbonylbis[imino-3,1-phenylenecarbonylimino(1-methyl-1h-pyrrole-4,2-diyl)carbonylimino]}dinaphthalene-1,5-disulfonate salt and related compounds as heparanase inhibitors for the treatment of cancer

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9304589D0 (en) * 1993-03-05 1993-04-21 Erba Carlo Spa Biologically active ureido derivatives useful as antimetastic agents
GB9307948D0 (en) * 1993-04-16 1993-06-02 Erba Carlo Spa Biologically active ureido derivatives useful in the treatment of lentivirus-induced disease

Also Published As

Publication number Publication date
EA000166B1 (ru) 1998-10-29
ZA97902B (en) 1997-08-01
EP0820284A1 (en) 1998-01-28
WO1997028796A1 (en) 1997-08-14
IL121808A0 (en) 1998-02-22
MX9707673A (es) 1997-11-29
DK0820284T3 (da) 2000-07-24
GR3033332T3 (en) 2000-09-29
ATE189388T1 (de) 2000-02-15
JPH11504041A (ja) 1999-04-06
PL322717A1 (en) 1998-02-16
AU1720097A (en) 1997-08-28
KR19980703718A (ko) 1998-12-05
DE69701243D1 (de) 2000-03-09
EP0820284B1 (en) 2000-02-02
DE69701243T2 (de) 2000-09-07
US5859046A (en) 1999-01-12
BR9702075A (pt) 1998-06-09
AR005724A1 (es) 1999-07-14
CA2217008A1 (en) 1997-08-14
ES2144844T3 (es) 2000-06-16
NO974651D0 (no) 1997-10-08
EA199700302A1 (ru) 1998-04-30
NO974651L (no) 1997-12-02
GB9602721D0 (en) 1996-04-10
HUP9900796A2 (hu) 1999-07-28

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