PT1562604E - Compostos de prostaglandina para o tratamento de obesidade - Google Patents
Compostos de prostaglandina para o tratamento de obesidade Download PDFInfo
- Publication number
- PT1562604E PT1562604E PT03758747T PT03758747T PT1562604E PT 1562604 E PT1562604 E PT 1562604E PT 03758747 T PT03758747 T PT 03758747T PT 03758747 T PT03758747 T PT 03758747T PT 1562604 E PT1562604 E PT 1562604E
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- Prior art keywords
- compound
- prostaglandin
- obesity
- treatment
- keto
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/557—Eicosanoids, e.g. leukotrienes or prostaglandins
- A61K31/5575—Eicosanoids, e.g. leukotrienes or prostaglandins having a cyclopentane, e.g. prostaglandin E2, prostaglandin F2-alpha
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
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- Pharmacology & Pharmacy (AREA)
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- General Chemical & Material Sciences (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| WO2007111806A2 (en) * | 2006-03-23 | 2007-10-04 | Massachusetts Eye And Ear Infirmary | Cyclopentane heptanoic acid compounds for reducing body fat |
| CA2824317C (en) * | 2011-01-19 | 2014-12-16 | Terakine Therapeutics, Inc. | Uses of certain f-series prostaglandin analogs for treating diabetes and dyslipidemia |
| US8426471B1 (en) | 2011-12-19 | 2013-04-23 | Topokine Therapeutics, Inc. | Methods and compositions for reducing body fat and adipocytes |
| SG11201600237YA (en) | 2012-11-21 | 2016-02-26 | Topokine Therapeutics Inc | Methods and compositions for locally increasing body fat |
| WO2014159679A1 (en) | 2013-03-12 | 2014-10-02 | The United States Of America, As Represented By The Secretary, Department Of Health & Human Services | Methods for using lubiprostone to absorb fluid from the subretinal space |
| AU2014250937A1 (en) | 2013-04-12 | 2015-10-22 | Allergan, Inc. | Sustained release of bimatoprost, bimatoprost analogs, prostamides and prostaglandins for fat reduction |
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| US9820993B2 (en) | 2013-05-15 | 2017-11-21 | Topokine Therapeutics, Inc. | Methods and compositions for topical delivery of prostaglandins to subcutaneous fat |
| WO2015200425A1 (en) | 2014-06-27 | 2015-12-30 | Topokine Therapeutics, Inc. | Topical dosage regimen |
| US11452703B2 (en) | 2020-05-21 | 2022-09-27 | Peregrine Ophthalmic PTE LTD. | Methods and compositions for reducing adipocyte numbers |
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| JP2000157260A (ja) * | 1998-11-26 | 2000-06-13 | Toyobo Co Ltd | 初代前駆脂肪細胞の分化誘導方法及びその分化用培地 |
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| BR0209863A (pt) | 2001-05-18 | 2004-06-08 | Sucampo Ag | Composição catártica |
| JP4786866B2 (ja) | 2001-08-31 | 2011-10-05 | スキャンポ・アーゲー | クロライドチャンネルオープナーとしてのプロスタグランジンアナログ |
| AR037524A1 (es) | 2001-11-14 | 2004-11-17 | Sucampo Ag | Unidad de dosificacion que comprende un analogo de prostaglandina para el tratamiento de la constipacion |
| US7732487B2 (en) | 2001-11-19 | 2010-06-08 | Sucampo Ag | Method for treating a disease or condition responsive to opening of C1C-2 channel |
| JP4889219B2 (ja) | 2002-12-27 | 2012-03-07 | スキャンポ・アーゲー | 腹部不快感の処置のためのプロスタグランジン誘導体 |
| DE602004030245D1 (de) | 2003-07-03 | 2011-01-05 | Sucampo Ag | Pharmazeutische magensaftresistent überzogene zusammensetzung enthaltend prostaglandin-analoga als chloridkanalöffner |
| TWI387454B (zh) | 2004-09-02 | 2013-03-01 | 蘇坎波公司 | 治療胃腸道疾病之方法及組成物 |
| US20060281818A1 (en) | 2005-03-21 | 2006-12-14 | Sucampo Ag, North Carolina State University | Method for treating mucosal disorders |
| KR101466980B1 (ko) | 2005-04-12 | 2014-12-01 | 수캄포 아게 | 위장 장애 치료를 위한 프로스타글란딘 화합물과 양성자펌프 억제제의 병용 |
-
2003
- 2003-10-22 ES ES03758747T patent/ES2379652T3/es not_active Expired - Lifetime
- 2003-10-22 EP EP03758747A patent/EP1562604B1/en not_active Expired - Lifetime
- 2003-10-22 PT PT03758747T patent/PT1562604E/pt unknown
- 2003-10-22 US US10/531,874 patent/US8114911B2/en not_active Expired - Fee Related
- 2003-10-22 WO PCT/JP2003/013453 patent/WO2004037268A1/en not_active Ceased
- 2003-10-22 NZ NZ539582A patent/NZ539582A/en not_active IP Right Cessation
- 2003-10-22 CA CA2502439A patent/CA2502439C/en not_active Expired - Fee Related
- 2003-10-22 AT AT03758747T patent/ATE539756T1/de active
- 2003-10-22 AU AU2003274735A patent/AU2003274735B2/en not_active Ceased
- 2003-10-22 JP JP2004546433A patent/JP4705782B2/ja not_active Expired - Fee Related
- 2003-10-22 DK DK03758747.4T patent/DK1562604T3/da active
Also Published As
| Publication number | Publication date |
|---|---|
| AU2003274735B2 (en) | 2008-12-04 |
| EP1562604B1 (en) | 2012-01-04 |
| ES2379652T3 (es) | 2012-04-30 |
| DK1562604T3 (da) | 2012-04-02 |
| CA2502439A1 (en) | 2004-05-06 |
| CA2502439C (en) | 2011-11-22 |
| JP2006506381A (ja) | 2006-02-23 |
| US8114911B2 (en) | 2012-02-14 |
| US20050261373A1 (en) | 2005-11-24 |
| WO2004037268A1 (en) | 2004-05-06 |
| NZ539582A (en) | 2007-07-27 |
| EP1562604A1 (en) | 2005-08-17 |
| JP4705782B2 (ja) | 2011-06-22 |
| ATE539756T1 (de) | 2012-01-15 |
| AU2003274735A1 (en) | 2004-05-13 |
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