PT1432408E - Composições farmacêuticas que compreendem dióxido de silício coloidal - Google Patents

Composições farmacêuticas que compreendem dióxido de silício coloidal Download PDF

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Publication number
PT1432408E
PT1432408E PT02774661T PT02774661T PT1432408E PT 1432408 E PT1432408 E PT 1432408E PT 02774661 T PT02774661 T PT 02774661T PT 02774661 T PT02774661 T PT 02774661T PT 1432408 E PT1432408 E PT 1432408E
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PT
Portugal
Prior art keywords
composition
tablet
rapamycin
weight
silicon dioxide
Prior art date
Application number
PT02774661T
Other languages
English (en)
Portuguese (pt)
Inventor
Barbara Haeberlin
Andrea Kramer
Silvia Heuerding
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9922916&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT1432408(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of PT1432408E publication Critical patent/PT1432408E/pt

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
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    • AHUMAN NECESSITIES
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    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
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    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
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    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurosurgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Communicable Diseases (AREA)
  • Zoology (AREA)
  • Transplantation (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
PT02774661T 2001-09-28 2002-09-27 Composições farmacêuticas que compreendem dióxido de silício coloidal PT1432408E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0123400.4A GB0123400D0 (en) 2001-09-28 2001-09-28 Organic compounds

Publications (1)

Publication Number Publication Date
PT1432408E true PT1432408E (pt) 2010-12-07

Family

ID=9922916

Family Applications (2)

Application Number Title Priority Date Filing Date
PT02774661T PT1432408E (pt) 2001-09-28 2002-09-27 Composições farmacêuticas que compreendem dióxido de silício coloidal
PT91778894T PT2193788E (pt) 2001-09-28 2002-09-27 Composições farmacêuticas compreendendo dióxido de silício coloidal

Family Applications After (1)

Application Number Title Priority Date Filing Date
PT91778894T PT2193788E (pt) 2001-09-28 2002-09-27 Composições farmacêuticas compreendendo dióxido de silício coloidal

Country Status (30)

Country Link
US (4) US20040254210A1 (enExample)
EP (2) EP1432408B8 (enExample)
JP (2) JP2005507897A (enExample)
KR (1) KR100626785B1 (enExample)
CN (3) CN1561201A (enExample)
AR (2) AR036643A1 (enExample)
AT (1) ATE485813T1 (enExample)
BR (2) BR0212922A (enExample)
CA (1) CA2458455C (enExample)
CO (1) CO5390072A1 (enExample)
CY (2) CY1111119T1 (enExample)
DE (1) DE60238131D1 (enExample)
DK (2) DK1432408T3 (enExample)
EC (1) ECSP024323A (enExample)
ES (2) ES2354687T3 (enExample)
GB (1) GB0123400D0 (enExample)
HU (1) HU229991B1 (enExample)
IL (2) IL160498A0 (enExample)
MX (1) MXPA04002814A (enExample)
MY (1) MY150060A (enExample)
NO (1) NO333892B1 (enExample)
NZ (2) NZ531599A (enExample)
PE (1) PE20030602A1 (enExample)
PL (1) PL209704B1 (enExample)
PT (2) PT1432408E (enExample)
RU (1) RU2322970C2 (enExample)
SI (1) SI1432408T1 (enExample)
TW (1) TWI242449B (enExample)
WO (1) WO2003028705A1 (enExample)
ZA (1) ZA200401300B (enExample)

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