PT1406895E - Formulações de lactonas e métodos para o seu uso - Google Patents

Formulações de lactonas e métodos para o seu uso Download PDF

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Publication number
PT1406895E
PT1406895E PT02734779T PT02734779T PT1406895E PT 1406895 E PT1406895 E PT 1406895E PT 02734779 T PT02734779 T PT 02734779T PT 02734779 T PT02734779 T PT 02734779T PT 1406895 E PT1406895 E PT 1406895E
Authority
PT
Portugal
Prior art keywords
lactone
formulations
lactone formulations
Prior art date
Application number
PT02734779T
Other languages
English (en)
Inventor
David Terrero
Original Assignee
Magnachem Int Lab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Magnachem Int Lab Inc filed Critical Magnachem Int Lab Inc
Publication of PT1406895E publication Critical patent/PT1406895E/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/58—One oxygen atom, e.g. butenolide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/93—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
PT02734779T 2001-06-13 2002-06-12 Formulações de lactonas e métodos para o seu uso PT1406895E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US29787501P 2001-06-13 2001-06-13

Publications (1)

Publication Number Publication Date
PT1406895E true PT1406895E (pt) 2008-11-04

Family

ID=23148076

Family Applications (1)

Application Number Title Priority Date Filing Date
PT02734779T PT1406895E (pt) 2001-06-13 2002-06-12 Formulações de lactonas e métodos para o seu uso

Country Status (21)

Country Link
US (3) US6900242B2 (pt)
EP (1) EP1406895B1 (pt)
JP (1) JP2005500289A (pt)
KR (1) KR20040030676A (pt)
AR (1) AR036056A1 (pt)
AT (1) ATE406367T1 (pt)
AU (1) AU2002306150B2 (pt)
BR (1) BR0210432A (pt)
CA (1) CA2450660C (pt)
CO (1) CO5550429A2 (pt)
CY (1) CY1108590T1 (pt)
DE (1) DE60228576D1 (pt)
DK (1) DK1406895T3 (pt)
ES (1) ES2315365T3 (pt)
IL (3) IL159296A0 (pt)
MX (1) MXPA03011554A (pt)
PT (1) PT1406895E (pt)
RS (1) RS52139B (pt)
UY (1) UY27334A1 (pt)
WO (1) WO2002100854A1 (pt)
ZA (1) ZA200400208B (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2450660C (en) * 2001-06-13 2011-08-16 Magnachem International Laboratories, Inc. Lactone formulations and method of use
US8188145B2 (en) 2002-06-12 2012-05-29 Magnachem International Laboratories, Inc. Synthetic lactone formulations and method of use
CN1720242A (zh) 2002-11-05 2006-01-11 马格纳化学国际实验室公司 合成的内酯制剂及其使用方法
US20050045197A1 (en) * 2003-08-28 2005-03-03 Gelder Steven K. Multiple drug delivery system & method
JP2012507010A (ja) * 2008-10-24 2012-03-22 マグナケム インターナショナル ラボラトリーズ， インコーポレイテッド Ｒａｄ９と選択的に相互作用する化合物をスクリーニングするための方法
CN103099901B (zh) * 2013-01-26 2014-07-30 张红 一种治疗子宫内膜移位症的中药灌肠剂
KR101988479B1 (ko) * 2017-10-11 2019-09-24 (주)휴럼 리트세노라이드를 유효성분으로 하는 헬리코박터 파이로리 균주로부터 유래되는 위장질환 예방 및 치료용 약학 조성물

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US2624732A (en) * 1950-05-10 1953-01-06 Burroughs Wellcome Co Preparation of 5-benzyl-2,4-diaminopyrimidines
US3203953A (en) * 1963-01-18 1965-08-31 Ciba Geigy Corp Lactone obtained from helenium sp. and derivatives thereof
US3210377A (en) * 1963-06-05 1965-10-05 Olin Mathieson Gamma lactones
US4001425A (en) * 1974-04-17 1977-01-04 E. I. Du Pont De Nemours And Company Methods of treating hypertension and pharmaceutical compositions comprising 1-tertiary-alkyl-3-(substituted furyl)ureas as antihypertensive agents
JPS5111173B2 (pt) * 1974-04-25 1976-04-09
JPS51125722A (en) 1975-01-13 1976-11-02 Sumitomo Chem Co Ltd Germicides for industry and their preparation
JPS597713B2 (ja) 1977-12-19 1984-02-20 三井東圧化学株式会社 新規γ↓−ブチロラクトン誘導体とその製造法
JPS56128776A (en) 1980-03-14 1981-10-08 Otsuka Pharmaceut Factory Inc Alpha-methylene gamma-butyrolactone derivative
JPS58199413A (ja) 1982-05-13 1983-11-19 Pioneer Electronic Corp デイジタル変調信号の読取装置
JPS6058973A (ja) * 1983-09-13 1985-04-05 Mitsubishi Yuka Yakuhin Kk γ−プチロラクトン誘導体及びそれを有効成分とする免疫調節剤
JPS6226221A (ja) 1985-07-29 1987-02-04 Japan Tobacco Inc 抗変異原性剤
JP2524760B2 (ja) 1987-07-10 1996-08-14 テイカ株式会社 新規抗生物質
JPH01163175A (ja) 1987-12-21 1989-06-27 Ss Pharmaceut Co Ltd フラン−２−オン誘導体
US5242945A (en) * 1991-04-12 1993-09-07 American Home Products Corporation Tetronic and thiotetronic acid derivatives as phospholipase a2 inhibitors
US5250735A (en) * 1992-04-03 1993-10-05 University Of Pittsburgh 2-(N-substituted-aminoalkyl)-5-(E)-alkylidene cyclopentanones, 2-(N-substituted-aminoalkyl)-5-(E)-arylalkylidene cyclopentanones, and derivatives thereof
EP0720607A1 (en) * 1993-09-17 1996-07-10 PHARMACIA & UPJOHN COMPANY Substituted tetronic acids useful for treating hiv and other retroviruses
US5595756A (en) * 1993-12-22 1997-01-21 Inex Pharmaceuticals Corporation Liposomal compositions for enhanced retention of bioactive agents
DE69522589T2 (de) * 1994-06-07 2002-04-18 Teijin Ltd Vitamin D3-Derivate und ein Verfahren zu ihrer Herstellung
AUPN191295A0 (en) 1995-03-23 1995-04-27 Unisearch Limited Microbiocide or microbial regulator
US5962460A (en) * 1995-06-27 1999-10-05 National Science Council (Taiwan) Antineoplastic α-methylene-γ-butyrolactones
US5646164A (en) * 1995-11-14 1997-07-08 National Science Council α-methylene-γ-butyrolactones: new inhibitors of platelet aggregation
DK0869784T3 (da) 1995-11-17 2006-01-16 Univ Johns Hopkins Hæmning af fedtsyresyntase som middel til formindskelse af adipocytmængden
US6222048B1 (en) * 1995-12-18 2001-04-24 Merck Frosst Canada & Co. Diaryl-2-(5H)-furanones as Cox-2 inhibitors
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CA2450660C (en) * 2001-06-13 2011-08-16 Magnachem International Laboratories, Inc. Lactone formulations and method of use
US6686724B2 (en) * 2002-05-21 2004-02-03 Ford Motor Company Method of and apparatus for controlling charging and/or discharging of a battery for a hybrid electric vehicle
US8188145B2 (en) * 2002-06-12 2012-05-29 Magnachem International Laboratories, Inc. Synthetic lactone formulations and method of use
CN1720242A (zh) * 2002-11-05 2006-01-11 马格纳化学国际实验室公司 合成的内酯制剂及其使用方法

Also Published As

Publication number Publication date
CA2450660C (en) 2011-08-16
US20110092588A1 (en) 2011-04-21
EP1406895B1 (en) 2008-08-27
UY27334A1 (es) 2003-02-28
IL159296A0 (en) 2004-06-01
CA2450660A1 (en) 2002-12-19
BR0210432A (pt) 2004-08-03
ES2315365T3 (es) 2009-04-01
CY1108590T1 (el) 2014-04-09
CO5550429A2 (es) 2005-08-31
EP1406895A1 (en) 2004-04-14
AU2002306150B2 (en) 2008-02-14
DK1406895T3 (da) 2008-12-01
US20030069393A1 (en) 2003-04-10
KR20040030676A (ko) 2004-04-09
RS98603A (en) 2006-12-15
IL159296A (en) 2011-06-30
US20050209316A1 (en) 2005-09-22
WO2002100854A1 (en) 2002-12-19
ZA200400208B (en) 2005-06-29
ATE406367T1 (de) 2008-09-15
EP1406895A4 (en) 2004-11-17
US8536348B2 (en) 2013-09-17
RS52139B (en) 2012-08-31
IL211958A0 (en) 2011-06-30
US6900242B2 (en) 2005-05-31
JP2005500289A (ja) 2005-01-06
DE60228576D1 (de) 2008-10-09
AR036056A1 (es) 2004-08-04
MXPA03011554A (es) 2004-10-28

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