PT1389089E - Processo e composição para solubilizar um composto biologicamente activo com uma baixa solubilidade em água - Google Patents

Processo e composição para solubilizar um composto biologicamente activo com uma baixa solubilidade em água Download PDF

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Publication number
PT1389089E
PT1389089E PT02737899T PT02737899T PT1389089E PT 1389089 E PT1389089 E PT 1389089E PT 02737899 T PT02737899 T PT 02737899T PT 02737899 T PT02737899 T PT 02737899T PT 1389089 E PT1389089 E PT 1389089E
Authority
PT
Portugal
Prior art keywords
biologically active
lipid particles
container
lipophilic
solubilising
Prior art date
Application number
PT02737899T
Other languages
English (en)
Portuguese (pt)
Inventor
Peter Van Hoogevest
Steve Leigh
Mathew Louis Steven Leigh
Henricus Tiemessen
Original Assignee
Phares Pharm Res Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Phares Pharm Res Nv filed Critical Phares Pharm Res Nv
Publication of PT1389089E publication Critical patent/PT1389089E/pt

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/127—Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • A61K9/1277—Preparation processes; Proliposomes
    • A61K9/1278—Post-loading, e.g. by ion or pH gradient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
PT02737899T 2001-03-27 2002-03-26 Processo e composição para solubilizar um composto biologicamente activo com uma baixa solubilidade em água PT1389089E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP01302841 2001-03-27

Publications (1)

Publication Number Publication Date
PT1389089E true PT1389089E (pt) 2009-11-30

Family

ID=8181836

Family Applications (1)

Application Number Title Priority Date Filing Date
PT02737899T PT1389089E (pt) 2001-03-27 2002-03-26 Processo e composição para solubilizar um composto biologicamente activo com uma baixa solubilidade em água

Country Status (11)

Country Link
US (2) US20040115255A1 (enExample)
EP (1) EP1389089B1 (enExample)
JP (3) JP2004524368A (enExample)
AT (1) ATE440593T1 (enExample)
AU (1) AU2002312777B2 (enExample)
CA (1) CA2442539C (enExample)
DE (1) DE60233484D1 (enExample)
DK (1) DK1389089T3 (enExample)
ES (1) ES2332584T3 (enExample)
PT (1) PT1389089E (enExample)
WO (1) WO2002080883A2 (enExample)

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Also Published As

Publication number Publication date
CA2442539C (en) 2011-11-08
US20040115255A1 (en) 2004-06-17
CA2442539A1 (en) 2002-10-17
JP2004524368A (ja) 2004-08-12
DK1389089T3 (da) 2009-12-21
US20080131499A1 (en) 2008-06-05
EP1389089A2 (en) 2004-02-18
ATE440593T1 (de) 2009-09-15
WO2002080883A2 (en) 2002-10-17
WO2002080883A3 (en) 2003-12-11
DE60233484D1 (de) 2009-10-08
JP2012207042A (ja) 2012-10-25
EP1389089B1 (en) 2009-08-26
ES2332584T3 (es) 2010-02-09
AU2002312777B2 (en) 2007-07-05
AU2002312777A2 (en) 2002-10-21
JP2010013461A (ja) 2010-01-21

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