PT1029852E - Processo para obtencao de enantiomeros de cis-olirtina - Google Patents

Processo para obtencao de enantiomeros de cis-olirtina

Info

Publication number
PT1029852E
PT1029852E PT98935042T PT98935042T PT1029852E PT 1029852 E PT1029852 E PT 1029852E PT 98935042 T PT98935042 T PT 98935042T PT 98935042 T PT98935042 T PT 98935042T PT 1029852 E PT1029852 E PT 1029852E
Authority
PT
Portugal
Prior art keywords
olirtine
enantiomers
enantiomer
cis
order
Prior art date
Application number
PT98935042T
Other languages
English (en)
Portuguese (pt)
Inventor
Antoni Torrens-Jover
Jordi Frigola-Constansa
Original Assignee
Esteve Labor Dr
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Esteve Labor Dr filed Critical Esteve Labor Dr
Publication of PT1029852E publication Critical patent/PT1029852E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PT98935042T 1997-08-04 1998-07-31 Processo para obtencao de enantiomeros de cis-olirtina PT1029852E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES009701728A ES2130083B1 (es) 1997-08-04 1997-08-04 Procedimiento para la obtencion de los enantiomeros de cizolirtina.
PCT/ES1998/000223 WO1999007684A1 (es) 1997-08-04 1998-07-31 Procedimiento para la obtencion de los enantiomeros de cizolirtina

Publications (1)

Publication Number Publication Date
PT1029852E true PT1029852E (pt) 2003-03-31

Family

ID=8300306

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98935042T PT1029852E (pt) 1997-08-04 1998-07-31 Processo para obtencao de enantiomeros de cis-olirtina

Country Status (12)

Country Link
US (1) US6118009A (ja)
EP (1) EP1029852B1 (ja)
JP (1) JP2001512718A (ja)
AT (1) ATE227272T1 (ja)
AU (1) AU8442698A (ja)
CA (1) CA2299447C (ja)
DE (1) DE69809282T2 (ja)
DK (1) DK1029852T3 (ja)
ES (2) ES2130083B1 (ja)
NO (1) NO314499B1 (ja)
PT (1) PT1029852E (ja)
WO (1) WO1999007684A1 (ja)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040142929A1 (en) * 2001-07-06 2004-07-22 Ramon Merce-Vidal Derivatives of aryl (or heteroaryl) azolylcarbinoles for the treatment of urinary incontinence
TW200533657A (en) * 2004-02-17 2005-10-16 Esteve Labor Dr Substituted pyrazoline compounds, their preparation and use as medicaments
JP2007531785A (ja) * 2004-04-05 2007-11-08 ラボラトリオス・デル・デエレ・エステベ・エセ・ア 活性物質組合せ物
EP1584335A3 (en) * 2004-04-05 2006-02-22 Laboratorios Del Dr. Esteve, S.A. Active substance combination comprising a carbinol composition and an opioid
ES2244326B1 (es) * 2004-04-05 2007-02-16 Laboratorios Del Dr. Esteve, S.A. Combinacion de substancias activas.
US20060040924A1 (en) * 2004-06-22 2006-02-23 Laboratorios Dr. Esteve S.A. Derivatives of aryl (or heteroaryl) azolylcarbinols for the treatment of renal colic
WO2006063861A1 (en) * 2004-12-17 2006-06-22 Laboratorios Del Dr. Esteve, S.A. Process for obtaining cizolirtine and its enantiomers
EP1671968A1 (en) * 2004-12-17 2006-06-21 Laboratorios Del Dr. Esteve, S.A. Process for obtaining enantiomers of thienylazolylalcoxyethanamines
EP1671953A1 (en) * 2004-12-17 2006-06-21 Laboratorios Del Dr. Esteve, S.A. Process for obtaining cizolirtine and its enantiomers
EP1743892A1 (en) * 2005-07-15 2007-01-17 Laboratorios del Dr. Esteve S.A. Substituted pyrazoline compounds, their preparation and use as medicaments
EP1743890A1 (en) * 2005-07-15 2007-01-17 Laboratorios Del Dr. Esteve, S.A. 4,5-Dihydro-1H-pyrazole derivatives, their preparation and use as medicaments
US7897589B2 (en) * 2005-07-15 2011-03-01 Laboratorios Del Dr. Esteve, S.A. Substituted pyrazoline compounds, their preparation and use as medicaments
EP1757587A1 (en) * 2005-07-15 2007-02-28 Laboratorios Del Dr. Esteve, S.A. Substituted pyrazoline compounds, their preparation and use as medicaments
EP1820502A1 (en) 2006-02-10 2007-08-22 Laboratorios Del Dr. Esteve, S.A. Active substance combination comprising azolylcarbinol compounds
EP2151234A1 (en) * 2008-07-28 2010-02-10 Laboratorios Del. Dr. Esteve, S.A. Pharmaceutical formulation comprising a CB1-receptor compound in a solid solution and/or solid dispersion
US20100291151A1 (en) * 2009-04-21 2010-11-18 Auspex Pharmaceuticals, Inc. 1-methylpyrazole modulators of substance p, calcitonin gene-related peptide, adrenergic receptor, and/or 5-ht receptor
DE102010056283A1 (de) 2010-12-24 2012-06-28 Volkswagen Ag Wärmeübertragungssystem
CN108558695A (zh) * 2018-05-15 2018-09-21 浙江华贝药业有限责任公司 2,2,2-三氟-n-[(1s,4s)-4-羟基四氢萘-1-基]-乙酰胺制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4943635A (en) * 1987-08-27 1990-07-24 President & Fellows Of Harvard College Enantioselective reduction of ketones
EP0640089B1 (en) * 1992-05-14 1996-12-27 Pfizer Inc. Enantioselective oxazaborolidine catalysts
US5442118A (en) * 1994-04-22 1995-08-15 Sepracor, Inc. Asymmetric synthesis of (R)- and (S)-arylethanolamines from iminoketones

Also Published As

Publication number Publication date
DE69809282T2 (de) 2003-09-11
ES2130083A1 (es) 1999-06-16
ES2187044T3 (es) 2003-05-16
WO1999007684A1 (es) 1999-02-18
JP2001512718A (ja) 2001-08-28
CA2299447A1 (en) 1999-02-18
NO314499B1 (no) 2003-03-31
NO20000560L (no) 2000-03-29
US6118009A (en) 2000-09-12
EP1029852A1 (en) 2000-08-23
NO20000560D0 (no) 2000-02-03
ES2130083B1 (es) 2000-01-16
AU8442698A (en) 1999-03-01
ATE227272T1 (de) 2002-11-15
DK1029852T3 (da) 2003-02-24
EP1029852B1 (en) 2002-11-06
DE69809282D1 (de) 2002-12-12
CA2299447C (en) 2007-05-29

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