PL4065582T3 - Polimorficzne pochodne karbazolu i ich zastosowania - Google Patents

Polimorficzne pochodne karbazolu i ich zastosowania

Info

Publication number
PL4065582T3
PL4065582T3 PL20828454.7T PL20828454T PL4065582T3 PL 4065582 T3 PL4065582 T3 PL 4065582T3 PL 20828454 T PL20828454 T PL 20828454T PL 4065582 T3 PL4065582 T3 PL 4065582T3
Authority
PL
Poland
Prior art keywords
polymorphous
applications
carbazole derivatives
carbazole
derivatives
Prior art date
Application number
PL20828454.7T
Other languages
English (en)
Inventor
Alfredo C. Castro
Iii James Martin Nolan
Sarah Jean BETHUNE
Corinne Marie FOLBERTH
Original Assignee
Ikena Oncology, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ikena Oncology, Inc. filed Critical Ikena Oncology, Inc.
Publication of PL4065582T3 publication Critical patent/PL4065582T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PL20828454.7T 2019-11-26 2020-11-25 Polimorficzne pochodne karbazolu i ich zastosowania PL4065582T3 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962940481P 2019-11-26 2019-11-26
PCT/US2020/062197 WO2021108528A1 (en) 2019-11-26 2020-11-25 Polymorphic carbazole derivatives and uses thereof

Publications (1)

Publication Number Publication Date
PL4065582T3 true PL4065582T3 (pl) 2025-08-18

Family

ID=73856339

Family Applications (1)

Application Number Title Priority Date Filing Date
PL20828454.7T PL4065582T3 (pl) 2019-11-26 2020-11-25 Polimorficzne pochodne karbazolu i ich zastosowania

Country Status (14)

Country Link
US (3) US11591339B2 (pl)
EP (2) EP4065582B1 (pl)
JP (2) JP2023502531A (pl)
KR (1) KR20220125231A (pl)
CN (1) CN115279764A (pl)
AU (1) AU2020394424A1 (pl)
CA (1) CA3159317A1 (pl)
ES (1) ES3028099T3 (pl)
FI (1) FI4065582T3 (pl)
IL (1) IL293326A (pl)
MX (1) MX2022006308A (pl)
PL (1) PL4065582T3 (pl)
PT (1) PT4065582T (pl)
WO (1) WO2021108528A1 (pl)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI778050B (zh) 2017-04-21 2022-09-21 美商醫肯納腫瘤學公司 吲哚ahr抑制劑及其用途
PL4065582T3 (pl) 2019-11-26 2025-08-18 Ikena Oncology, Inc. Polimorficzne pochodne karbazolu i ich zastosowania
US12570638B2 (en) 2020-05-20 2026-03-10 Sail Biomedicines, Inc. Fused imidazole derivatives as AHR antagonists

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PL4065582T3 (pl) 2019-11-26 2025-08-18 Ikena Oncology, Inc. Polimorficzne pochodne karbazolu i ich zastosowania
IL293325A (en) 2019-11-26 2022-07-01 Ikena Oncology Inc Ahr inhibitors and uses thereof
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Also Published As

Publication number Publication date
ES3028099T3 (en) 2025-06-18
EP4529955A3 (en) 2025-07-16
EP4065582B1 (en) 2025-02-19
US20250276975A1 (en) 2025-09-04
JP2025113368A (ja) 2025-08-01
CN115279764A (zh) 2022-11-01
MX2022006308A (es) 2022-06-22
JP2023502531A (ja) 2023-01-24
WO2021108528A1 (en) 2021-06-03
EP4529955A2 (en) 2025-04-02
AU2020394424A1 (en) 2022-06-16
KR20220125231A (ko) 2022-09-14
US20210253579A1 (en) 2021-08-19
US12162884B2 (en) 2024-12-10
IL293326A (en) 2022-07-01
PT4065582T (pt) 2025-05-22
CA3159317A1 (en) 2021-06-03
FI4065582T3 (fi) 2025-05-25
EP4065582A1 (en) 2022-10-05
US20230286990A1 (en) 2023-09-14
US11591339B2 (en) 2023-02-28

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