PL370029A1 - Pochodne 2-amino-4-heteroaryloaminopirymidyny do stosowania w leczeniu raka - Google Patents

Pochodne 2-amino-4-heteroaryloaminopirymidyny do stosowania w leczeniu raka

Info

Publication number
PL370029A1
PL370029A1 PL02370029A PL37002902A PL370029A1 PL 370029 A1 PL370029 A1 PL 370029A1 PL 02370029 A PL02370029 A PL 02370029A PL 37002902 A PL37002902 A PL 37002902A PL 370029 A1 PL370029 A1 PL 370029A1
Authority
PL
Poland
Prior art keywords
heteroarylaminopyrimidine
cancer
derivatives
amino
treatment
Prior art date
Application number
PL02370029A
Other languages
English (en)
Inventor
John L. Buchanan
Stuart Chaffee
Jean-Christophe Harmange
Perry M. Novak
Xiaotian Zhu
Original Assignee
Amgen Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Amgen Inc. filed Critical Amgen Inc.
Publication of PL370029A1 publication Critical patent/PL370029A1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL02370029A 2001-08-22 2002-08-22 Pochodne 2-amino-4-heteroaryloaminopirymidyny do stosowania w leczeniu raka PL370029A1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31428501P 2001-08-22 2001-08-22
US10/225,819 US7115617B2 (en) 2001-08-22 2002-08-21 Amino-substituted pyrimidinyl derivatives and methods of use

Publications (1)

Publication Number Publication Date
PL370029A1 true PL370029A1 (pl) 2005-05-16

Family

ID=26919947

Family Applications (1)

Application Number Title Priority Date Filing Date
PL02370029A PL370029A1 (pl) 2001-08-22 2002-08-22 Pochodne 2-amino-4-heteroaryloaminopirymidyny do stosowania w leczeniu raka

Country Status (8)

Country Link
US (1) US7115617B2 (pl)
EP (1) EP1418916A1 (pl)
JP (1) JP2005501860A (pl)
AU (1) AU2002329826C1 (pl)
CA (1) CA2458011A1 (pl)
MX (1) MXPA04001622A (pl)
PL (1) PL370029A1 (pl)
WO (1) WO2003018022A1 (pl)

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Also Published As

Publication number Publication date
EP1418916A1 (en) 2004-05-19
WO2003018022A8 (en) 2003-10-02
AU2002329826B2 (en) 2005-06-09
MXPA04001622A (es) 2004-07-08
AU2002329826C1 (en) 2005-11-17
CA2458011A1 (en) 2003-03-06
JP2005501860A (ja) 2005-01-20
US7115617B2 (en) 2006-10-03
WO2003018022A1 (en) 2003-03-06
US20030125346A1 (en) 2003-07-03

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