PL3221331T3 - Steroidy, 6-alkilo-7-hydroksy-4-en-3-ony jako związki pośrednie do wytwarzania steroidowych modulatorów fxr - Google Patents

Steroidy, 6-alkilo-7-hydroksy-4-en-3-ony jako związki pośrednie do wytwarzania steroidowych modulatorów fxr

Info

Publication number
PL3221331T3
PL3221331T3 PL15800909T PL15800909T PL3221331T3 PL 3221331 T3 PL3221331 T3 PL 3221331T3 PL 15800909 T PL15800909 T PL 15800909T PL 15800909 T PL15800909 T PL 15800909T PL 3221331 T3 PL3221331 T3 PL 3221331T3
Authority
PL
Poland
Prior art keywords
steroids
intermediates
hydroxy
alkyl
production
Prior art date
Application number
PL15800909T
Other languages
English (en)
Polish (pl)
Inventor
Alexander Weymouth-Wilson
Zofia KOMSTA
James Boydell
Carl OTTER
Laura WALLIS
Rhys BATCHELOR
Original Assignee
NZP UK Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB1420594.2A external-priority patent/GB201420594D0/en
Priority claimed from GBGB1420593.4A external-priority patent/GB201420593D0/en
Priority claimed from GBGB1505670.8A external-priority patent/GB201505670D0/en
Application filed by NZP UK Limited filed Critical NZP UK Limited
Publication of PL3221331T3 publication Critical patent/PL3221331T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C07J9/005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PL15800909T 2014-11-19 2015-11-19 Steroidy, 6-alkilo-7-hydroksy-4-en-3-ony jako związki pośrednie do wytwarzania steroidowych modulatorów fxr PL3221331T3 (pl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB1420594.2A GB201420594D0 (en) 2014-11-19 2014-11-19 Compounds
GBGB1420593.4A GB201420593D0 (en) 2014-11-19 2014-11-19 Compounds
GBGB1505670.8A GB201505670D0 (en) 2015-04-01 2015-04-01 Compounds
EP15800909.2A EP3221331B1 (en) 2014-11-19 2015-11-19 6-alkyl-7-hydroxy-4-en-3-one steroids as intermediates for the production of steroidal fxr modulators
PCT/GB2015/053516 WO2016079517A1 (en) 2014-11-19 2015-11-19 6-alkyl-7-hydroxy-4-en-3-one steroids as intermediates for the production of steroidal fxr modulators

Publications (1)

Publication Number Publication Date
PL3221331T3 true PL3221331T3 (pl) 2020-03-31

Family

ID=54704019

Family Applications (1)

Application Number Title Priority Date Filing Date
PL15800909T PL3221331T3 (pl) 2014-11-19 2015-11-19 Steroidy, 6-alkilo-7-hydroksy-4-en-3-ony jako związki pośrednie do wytwarzania steroidowych modulatorów fxr

Country Status (15)

Country Link
US (1) US10301350B2 (enExample)
EP (1) EP3221331B1 (enExample)
JP (1) JP6700274B2 (enExample)
KR (1) KR102526631B1 (enExample)
CN (1) CN107207559B (enExample)
BR (1) BR112017010319B1 (enExample)
CA (1) CA2968309A1 (enExample)
DK (1) DK3221331T3 (enExample)
EA (1) EA033427B1 (enExample)
ES (1) ES2759725T3 (enExample)
MX (1) MX375863B (enExample)
PL (1) PL3221331T3 (enExample)
PT (1) PT3221331T (enExample)
TW (1) TWI690536B (enExample)
WO (1) WO2016079517A1 (enExample)

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GB201608777D0 (en) * 2016-05-18 2016-06-29 Dextra Lab Ltd Compounds
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Also Published As

Publication number Publication date
DK3221331T3 (da) 2019-12-02
NZ731924A (en) 2020-12-18
KR20170086604A (ko) 2017-07-26
JP2017534670A (ja) 2017-11-24
US20170327528A1 (en) 2017-11-16
WO2016079517A1 (en) 2016-05-26
EP3221331B1 (en) 2019-09-18
EP3221331A1 (en) 2017-09-27
MX375863B (es) 2025-03-07
MX2017006563A (es) 2018-01-26
US10301350B2 (en) 2019-05-28
JP6700274B2 (ja) 2020-05-27
EA033427B1 (ru) 2019-10-31
HK1246801A1 (en) 2018-09-14
BR112017010319A2 (pt) 2017-12-26
CA2968309A1 (en) 2016-05-26
PT3221331T (pt) 2019-12-23
CN107207559B (zh) 2019-10-25
CN107207559A (zh) 2017-09-26
EA201790884A8 (ru) 2019-07-31
BR112017010319B1 (pt) 2023-04-11
EA201790884A1 (ru) 2017-11-30
ES2759725T3 (es) 2020-05-12
KR102526631B1 (ko) 2023-04-27
TW201632537A (zh) 2016-09-16
TWI690536B (zh) 2020-04-11

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