PL2991976T3 - Synteza 3-(5-amino-2-metylo-4-oksochinazolin-3(4h)-ylo)piperydyno-2,6-dionu - Google Patents

Synteza 3-(5-amino-2-metylo-4-oksochinazolin-3(4h)-ylo)piperydyno-2,6-dionu

Info

Publication number
PL2991976T3
PL2991976T3 PL14728381T PL14728381T PL2991976T3 PL 2991976 T3 PL2991976 T3 PL 2991976T3 PL 14728381 T PL14728381 T PL 14728381T PL 14728381 T PL14728381 T PL 14728381T PL 2991976 T3 PL2991976 T3 PL 2991976T3
Authority
PL
Poland
Prior art keywords
oxoquinazolin
dione
piperidine
synthesis
amino
Prior art date
Application number
PL14728381T
Other languages
English (en)
Polish (pl)
Inventor
Alexander L Ruchelman
Benjamin M Cohen
Anusuya Choudhury
Matthew M Kreilein
William W Leong
Hon-Wah Man
Original Assignee
Celgene Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Celgene Corp filed Critical Celgene Corp
Publication of PL2991976T3 publication Critical patent/PL2991976T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PL14728381T 2013-05-01 2014-04-30 Synteza 3-(5-amino-2-metylo-4-oksochinazolin-3(4h)-ylo)piperydyno-2,6-dionu PL2991976T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361818254P 2013-05-01 2013-05-01
PCT/US2014/036083 WO2014179416A1 (en) 2013-05-01 2014-04-30 Synthesis of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4h)-yl) piperidine-2,6-dione
EP14728381.6A EP2991976B1 (en) 2013-05-01 2014-04-30 Synthesis of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4h)-yl) piperidine-2,6-dione

Publications (1)

Publication Number Publication Date
PL2991976T3 true PL2991976T3 (pl) 2018-01-31

Family

ID=50885008

Family Applications (1)

Application Number Title Priority Date Filing Date
PL14728381T PL2991976T3 (pl) 2013-05-01 2014-04-30 Synteza 3-(5-amino-2-metylo-4-oksochinazolin-3(4h)-ylo)piperydyno-2,6-dionu

Country Status (26)

Country Link
US (3) US9067912B2 (enExample)
EP (2) EP3199532A1 (enExample)
JP (2) JP6490055B2 (enExample)
KR (1) KR20160003228A (enExample)
CN (2) CN105377831B (enExample)
AR (1) AR096165A1 (enExample)
AU (2) AU2014260011A1 (enExample)
CA (1) CA2910971A1 (enExample)
CY (1) CY1119525T1 (enExample)
DK (1) DK2991976T3 (enExample)
ES (1) ES2645944T3 (enExample)
HR (1) HRP20171535T1 (enExample)
HU (1) HUE034770T2 (enExample)
LT (1) LT2991976T (enExample)
MX (1) MX363652B (enExample)
NZ (1) NZ628322A (enExample)
PH (1) PH12015502477A1 (enExample)
PL (1) PL2991976T3 (enExample)
PT (1) PT2991976T (enExample)
RS (1) RS56565B1 (enExample)
RU (1) RU2015151359A (enExample)
SG (1) SG11201508836XA (enExample)
SI (1) SI2991976T1 (enExample)
SM (1) SMT201700513T1 (enExample)
TW (1) TW201536766A (enExample)
WO (1) WO2014179416A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RS52349B (sr) 2006-09-26 2012-12-31 Celgene Corporation 5-supstituisani derivati hinazolinona kao antitumorski agensi
CA2829570C (en) 2011-03-11 2019-05-07 Celgene Corporation Solid forms of 3-(5-amino-2-methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses
EP2892887B1 (en) 2012-09-04 2020-07-15 Celgene Corporation Isotopologues of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4h)-yl) piperidine-2-6-dione and methods of preparation thereof
US10973822B2 (en) 2015-07-02 2021-04-13 Celgene Corporation Combination therapy for treatment of hematological cancers and solid tumors
CN106083622B (zh) * 2016-06-16 2018-06-19 常州齐晖药业有限公司 一种甲苯咪唑中间体3,4-二氨基二苯甲酮的制备方法
US20180258064A1 (en) * 2017-03-07 2018-09-13 Celgene Corporation Solid forms of 3-(5-amino-2-methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses
CN113101295A (zh) * 2020-03-20 2021-07-13 上海疆云医疗健康科技有限公司 二苯乙烯类似物在治疗糖尿病肾脏疾病中的用途
KR20240055046A (ko) * 2021-09-02 2024-04-26 신톤 비.브이. 오시머티닙을 제조하는 방법

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2032538A2 (en) * 2006-06-08 2009-03-11 Array Biopharma, Inc. Quinoline compounds and methods of use
RS52349B (sr) * 2006-09-26 2012-12-31 Celgene Corporation 5-supstituisani derivati hinazolinona kao antitumorski agensi
RU2017120977A (ru) * 2011-03-11 2018-11-15 Селджин Корпорейшн Способ лечения рака с использованием 3-(5-амино-2-метил-4-оксо-4h-хиназолин-3-ил)пиперидин-2,6-диона
CA2829570C (en) * 2011-03-11 2019-05-07 Celgene Corporation Solid forms of 3-(5-amino-2-methyl-4-oxo-4h-quinazolin-3-yl)-piperidine-2,6-dione, and their pharmaceutical compositions and uses
EP2892887B1 (en) * 2012-09-04 2020-07-15 Celgene Corporation Isotopologues of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4h)-yl) piperidine-2-6-dione and methods of preparation thereof
EP2943201B2 (en) * 2013-01-14 2020-07-29 Deuterx, LLC 3-(5-substituted-4-oxoquinazolin-3(4h)-yl)-3-deutero-piperidine-2,6-dione derivatives

Also Published As

Publication number Publication date
RS56565B1 (sr) 2018-02-28
NZ628322A (en) 2017-06-30
CN107935994A (zh) 2018-04-20
US9303014B2 (en) 2016-04-05
CN105377831B (zh) 2018-02-02
KR20160003228A (ko) 2016-01-08
JP6490055B2 (ja) 2019-03-27
RU2015151359A (ru) 2017-06-06
MX2015015073A (es) 2016-03-03
EP2991976A1 (en) 2016-03-09
SI2991976T1 (sl) 2017-11-30
LT2991976T (lt) 2017-10-25
CA2910971A1 (en) 2014-11-06
CN105377831A (zh) 2016-03-02
JP2019069958A (ja) 2019-05-09
SMT201700513T1 (it) 2018-01-11
US20150274694A1 (en) 2015-10-01
US9067912B2 (en) 2015-06-30
US9266858B2 (en) 2016-02-23
PH12015502477A1 (en) 2016-02-22
MX363652B (es) 2019-03-28
AR096165A1 (es) 2015-12-09
ES2645944T3 (es) 2017-12-11
WO2014179416A1 (en) 2014-11-06
US20140330016A1 (en) 2014-11-06
EP3199532A1 (en) 2017-08-02
HUE034770T2 (hu) 2018-02-28
PT2991976T (pt) 2017-11-14
CY1119525T1 (el) 2018-03-07
HRP20171535T1 (hr) 2017-11-17
EP2991976B1 (en) 2017-09-20
SG11201508836XA (en) 2015-11-27
US20160009685A1 (en) 2016-01-14
JP2016517886A (ja) 2016-06-20
TW201536766A (zh) 2015-10-01
AU2017200965A1 (en) 2017-03-02
DK2991976T3 (da) 2017-11-06
AU2014260011A1 (en) 2015-11-12

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